BG98813A - Терапевтични средства - Google Patents
Терапевтични средства Download PDFInfo
- Publication number
- BG98813A BG98813A BG98813A BG9881394A BG98813A BG 98813 A BG98813 A BG 98813A BG 98813 A BG98813 A BG 98813A BG 9881394 A BG9881394 A BG 9881394A BG 98813 A BG98813 A BG 98813A
- Authority
- BG
- Bulgaria
- Prior art keywords
- group
- alkyl group
- hydrogen
- formula
- halogen
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Rheumatology (AREA)
- Pharmacology & Pharmacy (AREA)
- Pain & Pain Management (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Steroid Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB919127252A GB9127252D0 (en) | 1991-12-23 | 1991-12-23 | Therapeutic agents |
PCT/EP1992/002901 WO1993013097A1 (fr) | 1991-12-23 | 1992-12-12 | Derives de naphtyridine antirhumatismaux |
CN93109454A CN1096784A (zh) | 1991-12-23 | 1993-06-22 | 含取代4(5)-氨基-1,8-二氨杂萘的治疗剂 |
Publications (1)
Publication Number | Publication Date |
---|---|
BG98813A true BG98813A (bg) | 1995-05-31 |
Family
ID=36822317
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BG98813A BG98813A (bg) | 1991-12-23 | 1994-05-31 | Терапевтични средства |
Country Status (22)
Country | Link |
---|---|
US (1) | US5464781A (fr) |
EP (1) | EP0618916B1 (fr) |
JP (1) | JP2527917B2 (fr) |
CN (1) | CN1096784A (fr) |
AT (1) | ATE171452T1 (fr) |
AU (1) | AU656832B2 (fr) |
BG (1) | BG98813A (fr) |
CA (1) | CA2125858A1 (fr) |
CZ (1) | CZ153594A3 (fr) |
DE (1) | DE69227125T2 (fr) |
FI (1) | FI943019A0 (fr) |
GB (1) | GB9127252D0 (fr) |
HR (1) | HRP921455A2 (fr) |
HU (1) | HUT66971A (fr) |
IL (1) | IL104169A0 (fr) |
IN (1) | IN174405B (fr) |
MX (1) | MX9207494A (fr) |
NO (1) | NO942376L (fr) |
NZ (1) | NZ246156A (fr) |
SI (1) | SI9200408A (fr) |
SK (1) | SK75094A3 (fr) |
WO (1) | WO1993013097A1 (fr) |
Families Citing this family (28)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9312891D0 (en) * | 1993-06-22 | 1993-08-04 | Boots Co Plc | Therapeutic agents |
GB9318931D0 (en) * | 1993-09-14 | 1993-10-27 | Boots Co Plc | Therapeutic agents |
GB9420168D0 (en) * | 1994-10-06 | 1994-11-23 | Boots Co Plc | Therapeutic agents |
AR004010A1 (es) | 1995-10-11 | 1998-09-30 | Glaxo Group Ltd | Compuestos heterociclicos |
ATE300521T1 (de) | 1996-09-25 | 2005-08-15 | Astrazeneca Ab | Chinolin-derivate die den effekt von wachstumsfaktoren wie vegf vezögern |
RS49779B (sr) | 1998-01-12 | 2008-06-05 | Glaxo Group Limited, | Biciklična heteroaromatična jedinjenja kao inhibitori protein tirozin kinaze |
US6166069A (en) * | 1998-05-12 | 2000-12-26 | American Home Products Corporation | Phenyl oxo-acetic acids useful in the treatment of insulin resistance and hyperglycemia |
ATE377597T1 (de) | 1999-07-09 | 2007-11-15 | Glaxo Group Ltd | Anilinochinazoline als protein-tyrosin- kinasehemmer |
US6933299B1 (en) | 1999-07-09 | 2005-08-23 | Smithkline Beecham Corporation | Anilinoquinazolines as protein tyrosine kinase inhibitors |
US7160889B2 (en) | 2000-04-07 | 2007-01-09 | Astrazeneca Ab | Quinazoline compounds |
US6534656B2 (en) * | 2001-05-31 | 2003-03-18 | North Carolina State University | Short synthesis of pyridine-based pharmaceutical intermediates |
JP2003329989A (ja) * | 2002-03-06 | 2003-11-19 | Nippon Telegr & Teleph Corp <Ntt> | 光送信装置 |
GB0230018D0 (en) | 2002-12-23 | 2003-01-29 | Syngenta Ltd | Fungicides |
WO2006074147A2 (fr) | 2005-01-03 | 2006-07-13 | Myriad Genetics, Inc. | Composes et utilisation therapeutique associee |
EP1660092A2 (fr) | 2003-07-03 | 2006-05-31 | Myriad Genetics, Inc. | 4-arylamino-quinazolines comme activateurs de caspases et inducteurs d'apoptose |
US8309562B2 (en) * | 2003-07-03 | 2012-11-13 | Myrexis, Inc. | Compounds and therapeutical use thereof |
BRPI0418102A (pt) | 2003-12-23 | 2007-04-27 | Pfizer | derivados de quinolina |
US8258145B2 (en) * | 2005-01-03 | 2012-09-04 | Myrexis, Inc. | Method of treating brain cancer |
WO2007076034A2 (fr) * | 2005-12-21 | 2007-07-05 | Abbott Laboratories | Composes antiviraux |
CN102702194A (zh) * | 2005-12-21 | 2012-10-03 | 雅培制药有限公司 | 抗病毒化合物 |
TW200738707A (en) * | 2005-12-21 | 2007-10-16 | Abbott Lab | Anti-viral compounds |
WO2007081517A2 (fr) | 2005-12-21 | 2007-07-19 | Abbott Laboratories | Composes anti-viraux |
EP2345652A1 (fr) | 2005-12-21 | 2011-07-20 | Abbott Laboratories | Composées antivirales |
TWI399380B (zh) | 2006-12-20 | 2013-06-21 | Abbott Lab | 抗病毒化合物 |
EP2291376A2 (fr) * | 2008-07-03 | 2011-03-09 | Merck Patent GmbH | Naphtyridininones en tant qu inhibiteurs d aurora kinase |
US8415333B2 (en) | 2009-02-24 | 2013-04-09 | Respiratorious Ab | Bronchodilating diazaheteroaryls |
WO2011063398A1 (fr) * | 2009-11-23 | 2011-05-26 | Cylene Pharamaceuticals, Inc. | Polymorphes et sels d'un inhibiteur de kinase |
SG10201507846YA (en) | 2010-04-02 | 2015-10-29 | Senomyx Inc | Sweet flavor modifier |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4466965A (en) * | 1982-07-26 | 1984-08-21 | American Hospital Supply Corporation | Phthalazine compounds, compositions and use |
NZ213986A (en) * | 1984-10-30 | 1989-07-27 | Usv Pharma Corp | Heterocyclic or aromatic compounds, and pharmaceutical compositions containing such |
EP0222839A4 (fr) * | 1985-05-17 | 1988-11-09 | Univ Australian | Composes antipaludiques. |
JPS6368568A (ja) * | 1986-09-10 | 1988-03-28 | Otsuka Pharmaceut Factory Inc | p−アミノフエノ−ル誘導体 |
DE3644825A1 (de) * | 1986-12-31 | 1988-07-14 | Basf Ag | Substituierte 1,8-naphthyridin-derivate und diese enthaltende fungizide |
JPH07116187B2 (ja) * | 1987-07-22 | 1995-12-13 | シェリング・コーポレーション | 二環式化合物、それらを薬剤として使用すること、それらの製法、およびそれらの製造に有用な中間体 |
GB8804443D0 (en) * | 1988-02-25 | 1988-03-23 | Smithkline Beckman Intercredit | Compounds |
US4978661A (en) * | 1988-09-29 | 1990-12-18 | Innocenzo Caruso | Use of 6-halo-4-quinolone compounds and pharmaceutical compositions thereof for the preparation of a medicament for the therapeutical application in rheumatoid arthritis |
GR900100380A (el) * | 1989-05-20 | 1991-10-10 | Fisons Plc | Μέ?οδος παρασκευής αντι-φλεγμονωδών παραγώγων αμινοφενόλης. |
AU634561B2 (en) * | 1989-07-27 | 1993-02-25 | Eli Lilly And Company | Naphthyridine derivatives |
JP2988739B2 (ja) * | 1990-04-16 | 1999-12-13 | 協和醗酵工業株式会社 | 1,8−ナフチリジン−2−オン誘導体 |
JP3157077B2 (ja) * | 1994-02-16 | 2001-04-16 | 内山工業株式会社 | ベアリングシール |
-
1991
- 1991-12-23 GB GB919127252A patent/GB9127252D0/en active Pending
-
1992
- 1992-10-12 US US08/244,369 patent/US5464781A/en not_active Expired - Lifetime
- 1992-12-12 CA CA002125858A patent/CA2125858A1/fr not_active Abandoned
- 1992-12-12 EP EP93900052A patent/EP0618916B1/fr not_active Expired - Lifetime
- 1992-12-12 AT AT93900052T patent/ATE171452T1/de not_active IP Right Cessation
- 1992-12-12 AU AU31587/93A patent/AU656832B2/en not_active Ceased
- 1992-12-12 JP JP5511397A patent/JP2527917B2/ja not_active Expired - Fee Related
- 1992-12-12 WO PCT/EP1992/002901 patent/WO1993013097A1/fr active IP Right Grant
- 1992-12-12 CZ CZ941535A patent/CZ153594A3/cs unknown
- 1992-12-12 NZ NZ246156A patent/NZ246156A/en unknown
- 1992-12-12 HU HU9401877A patent/HUT66971A/hu unknown
- 1992-12-12 DE DE69227125T patent/DE69227125T2/de not_active Expired - Fee Related
- 1992-12-12 SK SK750-94A patent/SK75094A3/sk unknown
- 1992-12-17 IN IN758MA1992 patent/IN174405B/en unknown
- 1992-12-18 IL IL104169A patent/IL104169A0/xx unknown
- 1992-12-22 SI SI19929200408A patent/SI9200408A/sl unknown
- 1992-12-22 MX MX9207494A patent/MX9207494A/es unknown
- 1992-12-22 HR HR921455A patent/HRP921455A2/hr not_active Application Discontinuation
-
1993
- 1993-06-22 CN CN93109454A patent/CN1096784A/zh active Pending
-
1994
- 1994-05-31 BG BG98813A patent/BG98813A/bg unknown
- 1994-06-22 FI FI943019A patent/FI943019A0/fi not_active Application Discontinuation
- 1994-06-22 NO NO942376A patent/NO942376L/no unknown
Also Published As
Publication number | Publication date |
---|---|
HU9401877D0 (en) | 1994-09-28 |
FI943019A (fi) | 1994-06-22 |
IN174405B (fr) | 1994-11-26 |
CN1096784A (zh) | 1994-12-28 |
NZ246156A (en) | 1996-01-26 |
DE69227125D1 (de) | 1998-10-29 |
FI943019A0 (fi) | 1994-06-22 |
US5464781A (en) | 1995-11-07 |
GB9127252D0 (en) | 1992-02-19 |
CZ153594A3 (en) | 1995-02-15 |
CA2125858A1 (fr) | 1993-07-08 |
DE69227125T2 (de) | 1999-02-18 |
JPH07502280A (ja) | 1995-03-09 |
HUT66971A (en) | 1995-01-30 |
ATE171452T1 (de) | 1998-10-15 |
SK75094A3 (en) | 1995-04-12 |
EP0618916A1 (fr) | 1994-10-12 |
AU3158793A (en) | 1993-07-28 |
HRP921455A2 (en) | 1994-12-31 |
NO942376L (no) | 1994-06-22 |
WO1993013097A1 (fr) | 1993-07-08 |
IL104169A0 (en) | 1993-05-13 |
SI9200408A (en) | 1993-09-30 |
AU656832B2 (en) | 1995-02-16 |
JP2527917B2 (ja) | 1996-08-28 |
NO942376D0 (fr) | 1994-06-22 |
EP0618916B1 (fr) | 1998-09-23 |
MX9207494A (es) | 1993-07-01 |
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