BG62569B1 - Пенемови производни, тяхното получаване и приложението им въвфармацевтични композиции - Google Patents

Пенемови производни, тяхното получаване и приложението им въвфармацевтични композиции Download PDF

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Publication number
BG62569B1
BG62569B1 BG99507A BG9950795A BG62569B1 BG 62569 B1 BG62569 B1 BG 62569B1 BG 99507 A BG99507 A BG 99507A BG 9950795 A BG9950795 A BG 9950795A BG 62569 B1 BG62569 B1 BG 62569B1
Authority
BG
Bulgaria
Prior art keywords
methyl
hydroxyethyl
group
alkyl
carboxylic acid
Prior art date
Application number
BG99507A
Other languages
Bulgarian (bg)
English (en)
Other versions
BG99507A (bg
Inventor
Maria Altamura
Federico M. Arcamone
Enzo Perrotta
Vittorio Pestellini
Piero Sbraci
Giuseppe Cascio
Original Assignee
Menarini Industrie Farmaceutiche Riunite S.R.L.
Istituto Lusofarmaco D'italia S.P.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Menarini Industrie Farmaceutiche Riunite S.R.L., Istituto Lusofarmaco D'italia S.P.A. filed Critical Menarini Industrie Farmaceutiche Riunite S.R.L.
Publication of BG99507A publication Critical patent/BG99507A/bg
Publication of BG62569B1 publication Critical patent/BG62569B1/bg

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/88—Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Inks, Pencil-Leads, Or Crayons (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
BG99507A 1992-09-17 1995-03-17 Пенемови производни, тяхното получаване и приложението им въвфармацевтични композиции BG62569B1 (bg)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
ITFI920181A IT1262908B (it) 1992-09-17 1992-09-17 Derivati penems; loro preparazione e composizioni farmacologiche che li contengono
PCT/EP1993/002493 WO1994006803A1 (en) 1992-09-17 1993-09-15 Penem derivatives, their preparation and pharmaceutical compositions containing them
US08/414,081 US5747483A (en) 1992-09-17 1995-03-17 Penem derivatives, their preparation and pharmaceutical compositions containing them

Publications (2)

Publication Number Publication Date
BG99507A BG99507A (bg) 1996-01-31
BG62569B1 true BG62569B1 (bg) 2000-02-29

Family

ID=26330512

Family Applications (1)

Application Number Title Priority Date Filing Date
BG99507A BG62569B1 (bg) 1992-09-17 1995-03-17 Пенемови производни, тяхното получаване и приложението им въвфармацевтични композиции

Country Status (24)

Country Link
US (1) US5747483A (no)
EP (1) EP0660837B1 (no)
JP (1) JPH08501543A (no)
AT (1) ATE203027T1 (no)
AU (1) AU674874B2 (no)
BG (1) BG62569B1 (no)
BR (1) BR1100549A (no)
CA (1) CA2144961A1 (no)
CZ (1) CZ285816B6 (no)
DE (1) DE69330430T2 (no)
DK (1) DK0660837T3 (no)
ES (1) ES2158865T3 (no)
FI (1) FI951273A0 (no)
GR (1) GR3036817T3 (no)
HU (1) HU221318B1 (no)
IT (1) IT1262908B (no)
NO (1) NO310197B1 (no)
NZ (1) NZ256013A (no)
PL (1) PL176236B1 (no)
PT (1) PT660837E (no)
RO (1) RO113644B1 (no)
RU (1) RU2126410C1 (no)
SK (1) SK280476B6 (no)
WO (1) WO1994006803A1 (no)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5408002A (en) * 1993-09-09 1995-04-18 Minnesota Mining And Manufacturing Company Azlactone-functional polymer blends, articles produced therefrom and methods for preparing both
US11084833B2 (en) 2016-10-10 2021-08-10 The Johns Hopkins University Antibacterial agents against D,D- and L,D-transpeptidases

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PH21930A (en) * 1982-11-16 1988-04-08 Ciba Geigy Ag 6-hydroxy-lower alkylpenem compounds,pharmaceutical composition containing same and method of use thereof
EP0201459A1 (de) * 1985-05-06 1986-11-12 Ciba-Geigy Ag Acylaminomethylpenemverbindungen, ihre Herstellung und sie enthaltende pharmazeutische Präparate
EP0297042A1 (de) * 1987-06-23 1988-12-28 Ciba-Geigy Ag Substituierte Penem-Verbindungen
IT1239275B (it) * 1990-05-16 1993-10-01 Menarini Farma Ind Penem ditiocarbammati, loro uso e procedimento di fabbricazione relativi
GB9011151D0 (en) * 1990-05-18 1990-07-04 Secr Defence Zeolites

Also Published As

Publication number Publication date
CZ285816B6 (cs) 1999-11-17
HUT71520A (en) 1995-12-28
FI951273A (fi) 1995-03-17
BG99507A (bg) 1996-01-31
BR1100549A (pt) 2000-03-14
ATE203027T1 (de) 2001-07-15
AU4817093A (en) 1994-04-12
AU674874B2 (en) 1997-01-16
GR3036817T3 (en) 2002-01-31
DE69330430D1 (de) 2001-08-16
US5747483A (en) 1998-05-05
ITFI920181A1 (it) 1994-03-17
ES2158865T3 (es) 2001-09-16
DK0660837T3 (da) 2001-10-15
RU2126410C1 (ru) 1999-02-20
PL176236B1 (pl) 1999-05-31
PL308145A1 (en) 1995-07-24
IT1262908B (it) 1996-07-22
RU95108539A (ru) 1997-01-10
FI951273A0 (fi) 1995-03-17
SK27195A3 (en) 1995-07-11
NZ256013A (en) 1996-11-26
CZ65795A3 (en) 1995-09-13
HU9500791D0 (en) 1995-05-29
CA2144961A1 (en) 1994-03-31
PT660837E (pt) 2002-01-30
HU221318B1 (en) 2002-09-28
DE69330430T2 (de) 2002-08-29
JPH08501543A (ja) 1996-02-20
NO950941L (no) 1995-03-13
EP0660837B1 (en) 2001-07-11
WO1994006803A1 (en) 1994-03-31
RO113644B1 (ro) 1998-09-30
SK280476B6 (sk) 2000-02-14
ITFI920181A0 (it) 1992-09-17
NO310197B1 (no) 2001-06-05
EP0660837A1 (en) 1995-07-05
NO950941D0 (no) 1995-03-13

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