BG61815B1 - Фармакологично активни енантиомери - Google Patents
Фармакологично активни енантиомери Download PDFInfo
- Publication number
- BG61815B1 BG61815B1 BG100331A BG10033196A BG61815B1 BG 61815 B1 BG61815 B1 BG 61815B1 BG 100331 A BG100331 A BG 100331A BG 10033196 A BG10033196 A BG 10033196A BG 61815 B1 BG61815 B1 BG 61815B1
- Authority
- BG
- Bulgaria
- Prior art keywords
- compound
- formula
- alk
- physiologically acceptable
- alkyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P23/00—Anaesthetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
- C07D241/06—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members
- C07D241/08—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pain & Pain Management (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Anesthesiology (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Epoxy Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT93MI001418A IT1268414B1 (it) | 1993-07-01 | 1993-07-01 | Enantiomeri farmacologicamente attivi |
| PCT/EP1994/002061 WO1995001354A1 (en) | 1993-07-01 | 1994-06-21 | Pharmacologically active enantiomers |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| BG100331A BG100331A (bg) | 1996-09-30 |
| BG61815B1 true BG61815B1 (bg) | 1998-06-30 |
Family
ID=11366510
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG100331A BG61815B1 (bg) | 1993-07-01 | 1996-02-01 | Фармакологично активни енантиомери |
Country Status (29)
| Country | Link |
|---|---|
| US (3) | US5741907A (cs) |
| EP (1) | EP0707587B1 (cs) |
| JP (1) | JP3096065B2 (cs) |
| KR (1) | KR100306018B1 (cs) |
| CN (3) | CN1046281C (cs) |
| AT (1) | ATE158796T1 (cs) |
| AU (1) | AU689478B2 (cs) |
| BG (1) | BG61815B1 (cs) |
| BR (1) | BR9406996A (cs) |
| CA (1) | CA2166470C (cs) |
| CZ (1) | CZ289526B6 (cs) |
| DE (1) | DE69405999T2 (cs) |
| DK (1) | DK0707587T3 (cs) |
| ES (1) | ES2111309T3 (cs) |
| FI (1) | FI111943B (cs) |
| GE (1) | GEP19991791B (cs) |
| GR (1) | GR3025806T3 (cs) |
| HU (1) | HU221631B1 (cs) |
| IT (1) | IT1268414B1 (cs) |
| LV (1) | LV11546B (cs) |
| NO (1) | NO305957B1 (cs) |
| NZ (1) | NZ268014A (cs) |
| PL (1) | PL181831B1 (cs) |
| RO (2) | RO116899B1 (cs) |
| RU (1) | RU2128180C1 (cs) |
| SK (1) | SK281060B6 (cs) |
| UA (1) | UA53607C2 (cs) |
| WO (1) | WO1995001354A1 (cs) |
| ZA (1) | ZA944570B (cs) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1268414B1 (it) * | 1993-07-01 | 1997-02-27 | Angelini Francesco Ist Ricerca | Enantiomeri farmacologicamente attivi |
| JP2009018992A (ja) * | 2007-07-10 | 2009-01-29 | Sumitomo Chemical Co Ltd | 光学活性ミルタザピンの製造方法 |
| RU2706700C1 (ru) | 2019-09-24 | 2019-11-20 | Общество с ограниченной ответственностью "Научно-производственная компания "СКиФФ" | Фармацевтическая композиция для коррекции поведения кошек и собак в стрессовых ситуациях |
| KR20230083318A (ko) * | 2020-10-07 | 2023-06-09 | 암젠 인크 | 7-클로로-6-플루오로-1-(2-이소프로필-4-메틸피리딘-3-일)피리도[2,3-d]피리미딘-2,4(1H,3H)-디온의 회전장애이성질체의 라세미화 및 단리 방법 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3365453A (en) * | 1963-10-28 | 1968-01-23 | Sterling Drug Inc | 1-phenyl-4-lower-alkyl-2-piperazinones |
| IT1066857B (it) * | 1965-12-15 | 1985-03-12 | Acraf | Derivati della s ipiazolo 4.3 a piridina e processi per la loro preparazione |
| SU368258A1 (ru) * | 1970-01-27 | 1973-01-26 | Днепчопетровский химико технологический институт Ф. Э. Дзержинского | Способ получения 1,4-диарил-2-карбоксиметил- 3-оксопиперазинов |
| US5303837A (en) * | 1991-03-05 | 1994-04-19 | Portola Packaging, Inc. | One-piece fitment and plug with tamper-evident band |
| US5543563A (en) * | 1992-01-17 | 1996-08-06 | Istituto Ricerca Francesco Angelini S.P.A. | Alkyl derivatives of trazodone with CNS activity |
| IT1258790B (it) * | 1992-01-17 | 1996-02-29 | Angelini Francesco Ist Ricerca | Alchil derivati del trazodone |
| IT1268414B1 (it) * | 1993-07-01 | 1997-02-27 | Angelini Francesco Ist Ricerca | Enantiomeri farmacologicamente attivi |
| US5399765A (en) * | 1994-05-23 | 1995-03-21 | Sepracor, Inc. | Enantioselective preparation of optically pure albuterol |
-
1993
- 1993-07-01 IT IT93MI001418A patent/IT1268414B1/it active IP Right Grant
-
1994
- 1994-06-21 HU HU9503876A patent/HU221631B1/hu not_active IP Right Cessation
- 1994-06-21 EP EP94919660A patent/EP0707587B1/en not_active Expired - Lifetime
- 1994-06-21 WO PCT/EP1994/002061 patent/WO1995001354A1/en active IP Right Grant
- 1994-06-21 UA UA96010331A patent/UA53607C2/uk unknown
- 1994-06-21 DK DK94919660.4T patent/DK0707587T3/da active
- 1994-06-21 GE GEAP19943025A patent/GEP19991791B/en unknown
- 1994-06-21 JP JP07503250A patent/JP3096065B2/ja not_active Expired - Fee Related
- 1994-06-21 RO RO95-02315A patent/RO116899B1/ro unknown
- 1994-06-21 AU AU70729/94A patent/AU689478B2/en not_active Ceased
- 1994-06-21 AT AT94919660T patent/ATE158796T1/de not_active IP Right Cessation
- 1994-06-21 CA CA002166470A patent/CA2166470C/en not_active Expired - Fee Related
- 1994-06-21 NZ NZ268014A patent/NZ268014A/xx not_active IP Right Cessation
- 1994-06-21 RO ROA200100015A patent/RO121031B1/ro unknown
- 1994-06-21 PL PL94312419A patent/PL181831B1/pl not_active IP Right Cessation
- 1994-06-21 US US08/564,276 patent/US5741907A/en not_active Expired - Fee Related
- 1994-06-21 BR BR9406996A patent/BR9406996A/pt not_active Application Discontinuation
- 1994-06-21 CZ CZ19953485A patent/CZ289526B6/cs not_active IP Right Cessation
- 1994-06-21 ES ES94919660T patent/ES2111309T3/es not_active Expired - Lifetime
- 1994-06-21 RU RU96104371A patent/RU2128180C1/ru not_active IP Right Cessation
- 1994-06-21 CN CN94193226A patent/CN1046281C/zh not_active Expired - Fee Related
- 1994-06-21 DE DE69405999T patent/DE69405999T2/de not_active Expired - Fee Related
- 1994-06-21 KR KR1019950705994A patent/KR100306018B1/ko not_active Expired - Fee Related
- 1994-06-21 SK SK1664-95A patent/SK281060B6/sk not_active IP Right Cessation
- 1994-06-24 ZA ZA944570A patent/ZA944570B/xx unknown
-
1995
- 1995-12-29 NO NO955345A patent/NO305957B1/no unknown
- 1995-12-29 FI FI956334A patent/FI111943B/fi active
-
1996
- 1996-01-26 LV LVP-96-17A patent/LV11546B/en unknown
- 1996-02-01 BG BG100331A patent/BG61815B1/bg unknown
-
1997
- 1997-12-22 US US08/995,988 patent/US5817815A/en not_active Expired - Fee Related
- 1997-12-30 GR GR970403452T patent/GR3025806T3/el unknown
-
1998
- 1998-05-13 US US09/076,845 patent/US5973150A/en not_active Expired - Fee Related
- 1998-07-29 CN CNB98116661XA patent/CN1136201C/zh not_active Expired - Fee Related
- 1998-07-29 CN CNB981166601A patent/CN1136200C/zh not_active Expired - Fee Related
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