BG106568A - 5-(2-заместени-5-хетероциклилсулфонилпирид-3-ил)-дихидропиразоло[4,3-d]пиримидин-7-они като фосфодиестеразни инхибитори - Google Patents
5-(2-заместени-5-хетероциклилсулфонилпирид-3-ил)-дихидропиразоло[4,3-d]пиримидин-7-они като фосфодиестеразни инхибитори Download PDFInfo
- Publication number
- BG106568A BG106568A BG106568A BG10656802A BG106568A BG 106568 A BG106568 A BG 106568A BG 106568 A BG106568 A BG 106568A BG 10656802 A BG10656802 A BG 10656802A BG 106568 A BG106568 A BG 106568A
- Authority
- BG
- Bulgaria
- Prior art keywords
- lower alkyl
- dihydro
- pyrazolo
- pyrimidin
- ethyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Reproductive Health (AREA)
- General Health & Medical Sciences (AREA)
- Endocrinology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Gynecology & Obstetrics (AREA)
- Pregnancy & Childbirth (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9924041.8A GB9924041D0 (en) | 1999-10-11 | 1999-10-11 | Pharmaceutically active compounds |
| GB0018660A GB0018660D0 (en) | 2000-07-28 | 2000-07-28 | Pharmaceutically active compounds |
| PCT/IB2000/001430 WO2001027112A1 (en) | 1999-10-11 | 2000-10-04 | 5-(2-substituted-5-heterocyclylsulphonylpyrid-3-yl)-dihydropyrazolo[4,3-d]pyrimidin-7-ones as phosphodiesterase inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BG106568A true BG106568A (bg) | 2002-12-29 |
Family
ID=26244758
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG106568A BG106568A (bg) | 1999-10-11 | 2002-04-02 | 5-(2-заместени-5-хетероциклилсулфонилпирид-3-ил)-дихидропиразоло[4,3-d]пиримидин-7-они като фосфодиестеразни инхибитори |
Country Status (34)
| Country | Link |
|---|---|
| US (1) | US6756373B1 (hu) |
| EP (1) | EP1222190A1 (hu) |
| JP (1) | JP2003511452A (hu) |
| KR (1) | KR20020038941A (hu) |
| CN (1) | CN1378547A (hu) |
| AP (1) | AP2002002455A0 (hu) |
| AR (1) | AR022665A1 (hu) |
| AU (1) | AU7547900A (hu) |
| BG (1) | BG106568A (hu) |
| BR (1) | BR0014695A (hu) |
| CA (1) | CA2387353A1 (hu) |
| CO (1) | CO5261539A1 (hu) |
| CZ (1) | CZ20021151A3 (hu) |
| DZ (1) | DZ3218A1 (hu) |
| EA (1) | EA200200240A1 (hu) |
| EE (1) | EE200200192A (hu) |
| GT (1) | GT200000168A (hu) |
| HK (1) | HK1049834A1 (hu) |
| HU (1) | HUP0203438A3 (hu) |
| IL (1) | IL149025A0 (hu) |
| IS (1) | IS6288A (hu) |
| MA (1) | MA26824A1 (hu) |
| NO (1) | NO20021695L (hu) |
| NZ (1) | NZ517324A (hu) |
| OA (1) | OA12058A (hu) |
| PA (1) | PA8504401A1 (hu) |
| PE (1) | PE20010736A1 (hu) |
| PL (1) | PL357522A1 (hu) |
| SK (1) | SK4562002A3 (hu) |
| SV (1) | SV2002000192A (hu) |
| TN (1) | TNSN00198A1 (hu) |
| TR (1) | TR200200954T2 (hu) |
| UY (1) | UY26383A1 (hu) |
| WO (1) | WO2001027112A1 (hu) |
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| DE602006003416D1 (de) | 2005-03-21 | 2008-12-11 | Pfizer Ltd | Substituierte triazolderivate als oxytocinantagonisten |
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2000
- 2000-10-04 CN CN00814083A patent/CN1378547A/zh active Pending
- 2000-10-04 DZ DZ003218A patent/DZ3218A1/fr active
- 2000-10-04 AU AU75479/00A patent/AU7547900A/en not_active Abandoned
- 2000-10-04 CA CA002387353A patent/CA2387353A1/en not_active Abandoned
- 2000-10-04 JP JP2001530330A patent/JP2003511452A/ja not_active Withdrawn
- 2000-10-04 BR BR0014695-1A patent/BR0014695A/pt not_active IP Right Cessation
- 2000-10-04 WO PCT/IB2000/001430 patent/WO2001027112A1/en not_active Application Discontinuation
- 2000-10-04 PL PL00357522A patent/PL357522A1/xx not_active Application Discontinuation
- 2000-10-04 IL IL14902500A patent/IL149025A0/xx unknown
- 2000-10-04 CZ CZ20021151A patent/CZ20021151A3/cs unknown
- 2000-10-04 TR TR2002/00954T patent/TR200200954T2/xx unknown
- 2000-10-04 NZ NZ517324A patent/NZ517324A/en unknown
- 2000-10-04 OA OA1200200101A patent/OA12058A/en unknown
- 2000-10-04 HU HU0203438A patent/HUP0203438A3/hu unknown
- 2000-10-04 KR KR1020027004589A patent/KR20020038941A/ko not_active Application Discontinuation
- 2000-10-04 SK SK456-2002A patent/SK4562002A3/sk unknown
- 2000-10-04 AP APAP/P/2002/002455A patent/AP2002002455A0/en unknown
- 2000-10-04 EP EP00964557A patent/EP1222190A1/en not_active Withdrawn
- 2000-10-04 EA EA200200240A patent/EA200200240A1/ru unknown
- 2000-10-04 EE EEP200200192A patent/EE200200192A/xx unknown
- 2000-10-06 US US09/684,228 patent/US6756373B1/en not_active Expired - Fee Related
- 2000-10-09 UY UY26383A patent/UY26383A1/es not_active Application Discontinuation
- 2000-10-10 AR ARP000105332A patent/AR022665A1/es not_active Application Discontinuation
- 2000-10-10 CO CO00077032A patent/CO5261539A1/es not_active Application Discontinuation
- 2000-10-10 GT GT200000168A patent/GT200000168A/es unknown
- 2000-10-10 PE PE2000001084A patent/PE20010736A1/es not_active Application Discontinuation
- 2000-10-10 SV SV2000000192A patent/SV2002000192A/es unknown
- 2000-10-10 PA PA20008504401A patent/PA8504401A1/es unknown
- 2000-10-10 TN TNTNSN00198A patent/TNSN00198A1/fr unknown
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2002
- 2002-02-26 IS IS6288A patent/IS6288A/is unknown
- 2002-04-02 BG BG106568A patent/BG106568A/bg unknown
- 2002-04-04 MA MA26585A patent/MA26824A1/fr unknown
- 2002-04-10 NO NO20021695A patent/NO20021695L/no not_active Application Discontinuation
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2003
- 2003-03-14 HK HK03101881.7A patent/HK1049834A1/zh unknown
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