BG105858A - Инхибитори на повишени нива моноамини за лечение на разстройства на централната нервна система - Google Patents

Инхибитори на повишени нива моноамини за лечение на разстройства на централната нервна система

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Publication number
BG105858A
BG105858A BG105858A BG10585801A BG105858A BG 105858 A BG105858 A BG 105858A BG 105858 A BG105858 A BG 105858A BG 10585801 A BG10585801 A BG 10585801A BG 105858 A BG105858 A BG 105858A
Authority
BG
Bulgaria
Prior art keywords
treatment
reuptake inhibitors
cns disorders
monoamine reuptake
compounds
Prior art date
Application number
BG105858A
Other languages
English (en)
Inventor
Mark Elliott
Harry Howard
Christopher Schmidt
Thomas Seeger
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of BG105858A publication Critical patent/BG105858A/bg

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    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
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    • C07C217/80—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of non-condensed six-membered aromatic rings
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Abstract

Изобретението се отнася до съединения, които проявяват активност като инхибитори на повишени нива серотонин, норепинефрин и допамин, до техни фармацевтично приемливи соли и до използването им при лечение на разстройства на централната нервна системаи други заболявания. Съединенията имат формула, вкоято значенията на заместителите са посочени в описанието.
BG105858A 1999-02-23 2001-08-30 Инхибитори на повишени нива моноамини за лечение на разстройства на централната нервна система BG105858A (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US12131399P 1999-02-23 1999-02-23
PCT/IB2000/000108 WO2000050380A1 (en) 1999-02-23 2000-02-02 Monoamine reuptake inhibitors for treatment of cns disorders

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BG105858A true BG105858A (bg) 2002-04-30

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