AU757272B2 - Optically active quinoline carboxylic acid derivatives with 7-pyrrolidine substituents causing optical activity and a process for the preparation thereof - Google Patents

Optically active quinoline carboxylic acid derivatives with 7-pyrrolidine substituents causing optical activity and a process for the preparation thereof Download PDF

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Publication number
AU757272B2
AU757272B2 AU46209/00A AU4620900A AU757272B2 AU 757272 B2 AU757272 B2 AU 757272B2 AU 46209/00 A AU46209/00 A AU 46209/00A AU 4620900 A AU4620900 A AU 4620900A AU 757272 B2 AU757272 B2 AU 757272B2
Authority
AU
Australia
Prior art keywords
formula
compound
optically active
carboxylic acid
acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU46209/00A
Other languages
English (en)
Other versions
AU4620900A (en
Inventor
Dong Rack Choi
Yong Ho Chung
Yoon Ho Jin
Ik Hoe Kim
Nam Doo Kim
Chi Woo Lee
Jin Soo Lee
Jung Han Shin
Wan Jin Song
Wang Yong Yang
Sung June Yoon
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
EU BIOTECH DEVELOPMENT Ltd
Original Assignee
Dong Wha Pharm Ind Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from KR1020000024657A external-priority patent/KR20010029698A/ko
Application filed by Dong Wha Pharm Ind Co Ltd filed Critical Dong Wha Pharm Ind Co Ltd
Publication of AU4620900A publication Critical patent/AU4620900A/en
Application granted granted Critical
Publication of AU757272B2 publication Critical patent/AU757272B2/en
Assigned to EU BIOTECH DEVELOPMENT LTD reassignment EU BIOTECH DEVELOPMENT LTD Alteration of Name(s) in Register under S187 Assignors: DONG WHA PHARMACEUTICAL INDUSTRIAL CO., LTD.
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/10—Spiro-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyrrole Compounds (AREA)
AU46209/00A 1999-05-20 2000-05-18 Optically active quinoline carboxylic acid derivatives with 7-pyrrolidine substituents causing optical activity and a process for the preparation thereof Ceased AU757272B2 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
KR1999/18158 1999-05-20
KR19990018158 1999-05-20
KR2000/24657 2000-05-09
KR1020000024657A KR20010029698A (ko) 1999-05-20 2000-05-09 광학활성을 유발하는 7-피롤리딘 치환체를 갖는광학활성의 퀴놀린 카르복실산 유도체 및 그의 제조방법
PCT/KR2000/000487 WO2000071541A1 (en) 1999-05-20 2000-05-18 Optically active quinoline carboxylic acid derivatives having 7-pyrrolidine substitutes causing optical activity and a process for preparing thereof

Publications (2)

Publication Number Publication Date
AU4620900A AU4620900A (en) 2000-12-12
AU757272B2 true AU757272B2 (en) 2003-02-13

Family

ID=37040873

Family Applications (1)

Application Number Title Priority Date Filing Date
AU46209/00A Ceased AU757272B2 (en) 1999-05-20 2000-05-18 Optically active quinoline carboxylic acid derivatives with 7-pyrrolidine substituents causing optical activity and a process for the preparation thereof

Country Status (11)

Country Link
US (2) US6649763B1 (enExample)
EP (1) EP1187835B1 (enExample)
JP (2) JP2003500406A (enExample)
KR (1) KR100497942B1 (enExample)
CN (1) CN1142164C (enExample)
AT (1) ATE382047T1 (enExample)
AU (1) AU757272B2 (enExample)
CA (1) CA2374767C (enExample)
DE (1) DE60037587T2 (enExample)
ES (1) ES2296618T3 (enExample)
WO (1) WO2000071541A1 (enExample)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6589978B2 (en) * 2000-06-30 2003-07-08 Hoffman-La Roche Inc. 1-sulfonyl pyrrolidine derivatives
WO2006099167A1 (en) * 2005-03-10 2006-09-21 Theravance, Inc. Biphenyl compounds useful as muscarinic receptor antagonists
US7902227B2 (en) 2007-07-27 2011-03-08 Janssen Pharmaceutica Nv. C-7 isoxazolinyl quinolone / naphthyridine derivatives useful as antibacterial agents
CN101353348A (zh) * 2008-07-28 2009-01-28 南京明生医药技术有限公司 7-[4-(胺甲基)-4-氟-3-(烷氧亚氨基)吡咯烷-1-基]取代的喹啉羧酸衍生物及其制备方法
KR101468659B1 (ko) * 2009-07-27 2014-12-05 주식회사 아리바이오 Ｒ-7-(3-아미노메틸-4-메톡시이미노-3-메틸-피롤리딘-1-일)-1-시클로프로필-6-플루오로-4-옥소-1,4-디히드로-[1,8]나프티리딘-3-카르복실산 ｌ-아스파르트산염, 이의 제조방법 및 이를 포함하는 항균용 약학적 조성물
KR20220135949A (ko) 2021-03-31 2022-10-07 주식회사 이큐인베스트먼트 차트 유사도 분석을 이용한 주식 거래 인공신경망 장치 및 방법

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0541086A1 (en) * 1991-11-08 1993-05-12 Kaken Pharmaceutical Co., Ltd. Antibacterial 6-fluoro-quinolones having an oxime group on the substituent in position 7
DK0688772T3 (da) * 1994-06-16 1999-11-01 Lg Chemical Ltd Quinolincarboxylsyrederivater med 7-(4-aminomethyl-3-oxim)-pyrrolidinsubstituenter og fremgangsmåde til deres fremstilling
IT234996Y1 (it) 1994-06-22 2000-03-31 Bocchiotti Soc Ind Elettrotec Imballaggio per profilati metallici.
DE4422237A1 (de) * 1994-06-24 1996-01-04 Gruenenthal Gmbh Verwendung von Lactamverbindungen als pharmazeutische Wirkstoffe
KR0174373B1 (ko) * 1995-08-03 1999-02-18 성재갑 7-(4-아미노메틸-4-알킬-3-알킬옥심)피롤리딘 치환체를 갖는 신규 퀴놀린 카르복실산 유도체 및 그의 제조방법
DE69802692D1 (de) * 1997-06-26 2002-01-10 Dong Wha Pharm Ind Co Ltd Derivate der chinoloncarbonsäure

Also Published As

Publication number Publication date
JP2003500406A (ja) 2003-01-07
CA2374767C (en) 2007-05-15
US6753430B2 (en) 2004-06-22
ATE382047T1 (de) 2008-01-15
AU4620900A (en) 2000-12-12
JP2006232842A (ja) 2006-09-07
US20040029915A1 (en) 2004-02-12
CA2374767A1 (en) 2000-11-30
US6649763B1 (en) 2003-11-18
EP1187835A4 (en) 2003-01-29
WO2000071541A1 (en) 2000-11-30
ES2296618T3 (es) 2008-05-01
KR100497942B1 (ko) 2005-06-29
KR20020002461A (ko) 2002-01-09
CN1358185A (zh) 2002-07-10
EP1187835B1 (en) 2007-12-26
EP1187835A1 (en) 2002-03-20
JP5276255B2 (ja) 2013-08-28
DE60037587D1 (de) 2008-02-07
DE60037587T2 (de) 2008-04-30
CN1142164C (zh) 2004-03-17

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DA3 Amendments made section 104

Free format text: THE NATURE OF THE AMENDMENT IS: THE INVENTION TITLE IN REGARD TO PATENT APPLICATION NUMBER 46209/00 SHOULD READ: OPTICALLY ACTIVE QUINOLINE CARBOXYLIC ACID DERIVATIVES WITH 7-PYRROLIDINE SUBSTITUENTS CAUSING OPTICAL ACTIVITY AND A PROCESS FOR THE PREPARATION THEREOF

FGA Letters patent sealed or granted (standard patent)