AU2017302307A1 - Sodium bicarbonate in situ conversion driven transdermal delivery of amine drug - Google Patents

Sodium bicarbonate in situ conversion driven transdermal delivery of amine drug Download PDF

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Publication number
AU2017302307A1
AU2017302307A1 AU2017302307A AU2017302307A AU2017302307A1 AU 2017302307 A1 AU2017302307 A1 AU 2017302307A1 AU 2017302307 A AU2017302307 A AU 2017302307A AU 2017302307 A AU2017302307 A AU 2017302307A AU 2017302307 A1 AU2017302307 A1 AU 2017302307A1
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AU
Australia
Prior art keywords
composition
adhesive
active agent
transdermal
transdermal patch
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2017302307A
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English (en)
Inventor
Amit K. Jain
Eun Soo Lee
Appala Sagi
Parminder Singh
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Corium LLC
Original Assignee
Corium LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Corium LLC filed Critical Corium LLC
Publication of AU2017302307A1 publication Critical patent/AU2017302307A1/en
Assigned to Corium, LLC. reassignment Corium, LLC. Amend patent request/document other than specification (104) Assignors: CORIUM INTERNATIONAL, INC.
Priority to AU2023203616A priority Critical patent/AU2023203616A1/en
Priority to AU2025205205A priority patent/AU2025205205A1/en
Abandoned legal-status Critical Current

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
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    • A61K31/13—Amines
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    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
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    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/18—Sulfonamides
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    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/192—Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
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    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
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    • A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
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  • Dermatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Emergency Medicine (AREA)
  • Psychiatry (AREA)
  • Inorganic Chemistry (AREA)
  • Urology & Nephrology (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Addiction (AREA)
  • Pain & Pain Management (AREA)
  • Polymers & Plastics (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AU2017302307A 2016-07-27 2017-07-26 Sodium bicarbonate in situ conversion driven transdermal delivery of amine drug Abandoned AU2017302307A1 (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
AU2023203616A AU2023203616A1 (en) 2016-07-27 2023-06-09 Sodium bicarbonate in situ conversion driven transdermal delivery of amine drug
AU2025205205A AU2025205205A1 (en) 2016-07-27 2025-07-08 Sodium bicarbonate in situ conversion driven transdermal delivery of amine drug

Applications Claiming Priority (17)

Application Number Priority Date Filing Date Title
US201662367542P 2016-07-27 2016-07-27
US201662367502P 2016-07-27 2016-07-27
US62/367,542 2016-07-27
US62/367,502 2016-07-27
US201662423133P 2016-11-16 2016-11-16
US62/423,133 2016-11-16
US201762444745P 2017-01-10 2017-01-10
US201762444763P 2017-01-10 2017-01-10
US62/444,763 2017-01-10
US62/444,745 2017-01-10
US201762457794P 2017-02-10 2017-02-10
US62/457,794 2017-02-10
US201762504391P 2017-05-10 2017-05-10
US201762504408P 2017-05-10 2017-05-10
US62/504,408 2017-05-10
US62/504,391 2017-05-10
PCT/US2017/044049 WO2018022816A1 (en) 2016-07-27 2017-07-26 Sodium bicarbonate in situ conversion driven transdermal delivery of amine drug

Related Child Applications (1)

Application Number Title Priority Date Filing Date
AU2023203616A Division AU2023203616A1 (en) 2016-07-27 2023-06-09 Sodium bicarbonate in situ conversion driven transdermal delivery of amine drug

Publications (1)

Publication Number Publication Date
AU2017302307A1 true AU2017302307A1 (en) 2019-02-14

Family

ID=59523314

Family Applications (7)

Application Number Title Priority Date Filing Date
AU2017302307A Abandoned AU2017302307A1 (en) 2016-07-27 2017-07-26 Sodium bicarbonate in situ conversion driven transdermal delivery of amine drug
AU2017301928A Active AU2017301928B2 (en) 2016-07-27 2017-07-26 Donepezil transdermal delivery system
AU2017302306A Abandoned AU2017302306A1 (en) 2016-07-27 2017-07-26 Transdermal formulation and delivery method of low solubility or unstable unionized neutral drugs by in situ salt-to-neutral drug conversion of salt drug
AU2023203618A Active AU2023203618B2 (en) 2016-07-27 2023-06-09 Transdermal formulation and delivery method of low solubility or unstable unionized neutral drugs by in situ salt-to-neutral drug conversion of salt drug
AU2023203616A Abandoned AU2023203616A1 (en) 2016-07-27 2023-06-09 Sodium bicarbonate in situ conversion driven transdermal delivery of amine drug
AU2023204240A Abandoned AU2023204240A1 (en) 2016-07-27 2023-07-03 Donepezil transdermal delivery system
AU2025205205A Abandoned AU2025205205A1 (en) 2016-07-27 2025-07-08 Sodium bicarbonate in situ conversion driven transdermal delivery of amine drug

Family Applications After (6)

Application Number Title Priority Date Filing Date
AU2017301928A Active AU2017301928B2 (en) 2016-07-27 2017-07-26 Donepezil transdermal delivery system
AU2017302306A Abandoned AU2017302306A1 (en) 2016-07-27 2017-07-26 Transdermal formulation and delivery method of low solubility or unstable unionized neutral drugs by in situ salt-to-neutral drug conversion of salt drug
AU2023203618A Active AU2023203618B2 (en) 2016-07-27 2023-06-09 Transdermal formulation and delivery method of low solubility or unstable unionized neutral drugs by in situ salt-to-neutral drug conversion of salt drug
AU2023203616A Abandoned AU2023203616A1 (en) 2016-07-27 2023-06-09 Sodium bicarbonate in situ conversion driven transdermal delivery of amine drug
AU2023204240A Abandoned AU2023204240A1 (en) 2016-07-27 2023-07-03 Donepezil transdermal delivery system
AU2025205205A Abandoned AU2025205205A1 (en) 2016-07-27 2025-07-08 Sodium bicarbonate in situ conversion driven transdermal delivery of amine drug

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