AU2016367306B2 - Monomaleimide-functionalized platinum compounds for cancer therapy - Google Patents

Monomaleimide-functionalized platinum compounds for cancer therapy Download PDF

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Publication number
AU2016367306B2
AU2016367306B2 AU2016367306A AU2016367306A AU2016367306B2 AU 2016367306 B2 AU2016367306 B2 AU 2016367306B2 AU 2016367306 A AU2016367306 A AU 2016367306A AU 2016367306 A AU2016367306 A AU 2016367306A AU 2016367306 B2 AU2016367306 B2 AU 2016367306B2
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AU
Australia
Prior art keywords
alkyl
alkylene
cancer
compound
moiety
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AU2016367306A
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English (en)
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AU2016367306A1 (en
Inventor
Walter Berger
Petra Heffeter
Bernhard K. Keppler
Christian KOWOL
Josef Mayr
Verena PICHLER
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Medizinische Universitaet Wien
Universitaet Wien
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Medizinische Universitaet Wien
Universitaet Wien
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Publication of AU2016367306A1 publication Critical patent/AU2016367306A1/en
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F15/00—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table
    • C07F15/0006—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table compounds of the platinum group
    • C07F15/0086—Platinum compounds
    • C07F15/0093—Platinum compounds without a metal-carbon linkage
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/555—Heterocyclic compounds containing heavy metals, e.g. hemin, hematin, melarsoprol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AU2016367306A 2015-12-09 2016-12-09 Monomaleimide-functionalized platinum compounds for cancer therapy Ceased AU2016367306B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP15198739.3 2015-12-09
EP15198739 2015-12-09
PCT/EP2016/080453 WO2017097986A1 (en) 2015-12-09 2016-12-09 Monomaleimide-functionalized platinum compounds for cancer therapy

Publications (2)

Publication Number Publication Date
AU2016367306A1 AU2016367306A1 (en) 2018-06-14
AU2016367306B2 true AU2016367306B2 (en) 2021-04-22

Family

ID=54849106

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2016367306A Ceased AU2016367306B2 (en) 2015-12-09 2016-12-09 Monomaleimide-functionalized platinum compounds for cancer therapy

Country Status (21)

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US (2) US10723748B2 (https=)
EP (1) EP3386997B1 (https=)
JP (1) JP6867652B2 (https=)
CN (1) CN108368143B (https=)
AU (1) AU2016367306B2 (https=)
CA (1) CA3004630A1 (https=)
CY (1) CY1124529T1 (https=)
DK (1) DK3386997T3 (https=)
ES (1) ES2898704T3 (https=)
HR (1) HRP20211466T1 (https=)
HU (1) HUE056897T2 (https=)
IL (1) IL259864B (https=)
LT (1) LT3386997T (https=)
MX (1) MX377528B (https=)
PL (1) PL3386997T3 (https=)
PT (1) PT3386997T (https=)
RS (1) RS62412B1 (https=)
SG (1) SG11201804885TA (https=)
SI (1) SI3386997T1 (https=)
SM (1) SMT202100709T1 (https=)
WO (1) WO2017097986A1 (https=)

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TWI808055B (zh) 2016-05-11 2023-07-11 美商滬亞生物國際有限公司 Hdac 抑制劑與 pd-1 抑制劑之組合治療
CN109171001A (zh) * 2018-09-14 2019-01-11 上海烟草集团有限责任公司 草酸钠在降低卷烟烟气中TSNAs释放量中的应用
JP2023508996A (ja) * 2019-12-31 2023-03-06 キネート バイオファーマ インク． Ｃｄｋ１２／１３阻害剤を用いる癌の処置
CN114163479B (zh) * 2020-09-11 2025-05-16 上海海聚生物科技有限公司 一类治疗癌症用的铂类化合物及其制备方法
US20230339997A1 (en) * 2020-09-11 2023-10-26 Shanghai Haiju Biological Technology Co., Ltd. Class of platinum compounds for treating cancer, and method for preparation thereof
CN114539320B (zh) * 2020-11-25 2026-01-27 北京大学 辐射激活的四价铂配合物及其用途

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Also Published As

Publication number Publication date
AU2016367306A1 (en) 2018-06-14
ES2898704T3 (es) 2022-03-08
HRP20211466T1 (hr) 2021-12-24
CN108368143A (zh) 2018-08-03
MX2018006953A (es) 2019-05-16
US10723748B2 (en) 2020-07-28
US11572379B2 (en) 2023-02-07
SG11201804885TA (en) 2018-07-30
IL259864A (en) 2018-07-31
SI3386997T1 (sl) 2021-11-30
CN108368143B (zh) 2022-02-01
WO2017097986A1 (en) 2017-06-15
EP3386997A1 (en) 2018-10-17
CA3004630A1 (en) 2017-06-15
LT3386997T (lt) 2021-12-10
US20180354979A1 (en) 2018-12-13
SMT202100709T1 (it) 2022-01-10
JP6867652B2 (ja) 2021-05-12
EP3386997B1 (en) 2021-06-30
HUE056897T2 (hu) 2022-03-28
JP2018538292A (ja) 2018-12-27
MX377528B (es) 2025-03-10
PL3386997T3 (pl) 2021-12-13
DK3386997T3 (da) 2021-09-20
IL259864B (en) 2022-07-01
PT3386997T (pt) 2021-11-04
RS62412B1 (sr) 2021-10-29
CY1124529T1 (el) 2022-07-22
US20210002313A1 (en) 2021-01-07

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