IL259864B - Monomaleimide-functionalized platinum compounds for cancer therapy - Google Patents

Monomaleimide-functionalized platinum compounds for cancer therapy

Info

Publication number
IL259864B
IL259864B IL259864A IL25986418A IL259864B IL 259864 B IL259864 B IL 259864B IL 259864 A IL259864 A IL 259864A IL 25986418 A IL25986418 A IL 25986418A IL 259864 B IL259864 B IL 259864B
Authority
IL
Israel
Prior art keywords
alkyl
compound
alkylene
cancer
moiety
Prior art date
Application number
IL259864A
Other languages
English (en)
Hebrew (he)
Other versions
IL259864A (en
Original Assignee
Univ Wien Med
Univ Wien
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Wien Med, Univ Wien filed Critical Univ Wien Med
Publication of IL259864A publication Critical patent/IL259864A/en
Publication of IL259864B publication Critical patent/IL259864B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F15/00Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table
    • C07F15/0006Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table compounds of the platinum group
    • C07F15/0086Platinum compounds
    • C07F15/0093Platinum compounds without a metal-carbon linkage
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/555Heterocyclic compounds containing heavy metals, e.g. hemin, hematin, melarsoprol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
IL259864A 2015-12-09 2016-12-09 Monomaleimide-functionalized platinum compounds for cancer therapy IL259864B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP15198739 2015-12-09
PCT/EP2016/080453 WO2017097986A1 (en) 2015-12-09 2016-12-09 Monomaleimide-functionalized platinum compounds for cancer therapy

Publications (2)

Publication Number Publication Date
IL259864A IL259864A (en) 2018-07-31
IL259864B true IL259864B (en) 2022-07-01

Family

ID=54849106

Family Applications (1)

Application Number Title Priority Date Filing Date
IL259864A IL259864B (en) 2015-12-09 2016-12-09 Monomaleimide-functionalized platinum compounds for cancer therapy

Country Status (21)

Country Link
US (2) US10723748B2 (https=)
EP (1) EP3386997B1 (https=)
JP (1) JP6867652B2 (https=)
CN (1) CN108368143B (https=)
AU (1) AU2016367306B2 (https=)
CA (1) CA3004630A1 (https=)
CY (1) CY1124529T1 (https=)
DK (1) DK3386997T3 (https=)
ES (1) ES2898704T3 (https=)
HR (1) HRP20211466T1 (https=)
HU (1) HUE056897T2 (https=)
IL (1) IL259864B (https=)
LT (1) LT3386997T (https=)
MX (1) MX377528B (https=)
PL (1) PL3386997T3 (https=)
PT (1) PT3386997T (https=)
RS (1) RS62412B1 (https=)
SG (1) SG11201804885TA (https=)
SI (1) SI3386997T1 (https=)
SM (1) SMT202100709T1 (https=)
WO (1) WO2017097986A1 (https=)

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TWI808055B (zh) 2016-05-11 2023-07-11 美商滬亞生物國際有限公司 Hdac 抑制劑與 pd-1 抑制劑之組合治療
CN109171001A (zh) * 2018-09-14 2019-01-11 上海烟草集团有限责任公司 草酸钠在降低卷烟烟气中TSNAs释放量中的应用
JP2023508996A (ja) * 2019-12-31 2023-03-06 キネート バイオファーマ インク. Cdk12/13阻害剤を用いる癌の処置
CN114163479B (zh) * 2020-09-11 2025-05-16 上海海聚生物科技有限公司 一类治疗癌症用的铂类化合物及其制备方法
US20230339997A1 (en) * 2020-09-11 2023-10-26 Shanghai Haiju Biological Technology Co., Ltd. Class of platinum compounds for treating cancer, and method for preparation thereof
CN114539320B (zh) * 2020-11-25 2026-01-27 北京大学 辐射激活的四价铂配合物及其用途

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Also Published As

Publication number Publication date
AU2016367306A1 (en) 2018-06-14
ES2898704T3 (es) 2022-03-08
HRP20211466T1 (hr) 2021-12-24
CN108368143A (zh) 2018-08-03
MX2018006953A (es) 2019-05-16
US10723748B2 (en) 2020-07-28
US11572379B2 (en) 2023-02-07
SG11201804885TA (en) 2018-07-30
IL259864A (en) 2018-07-31
SI3386997T1 (sl) 2021-11-30
CN108368143B (zh) 2022-02-01
WO2017097986A1 (en) 2017-06-15
EP3386997A1 (en) 2018-10-17
CA3004630A1 (en) 2017-06-15
LT3386997T (lt) 2021-12-10
US20180354979A1 (en) 2018-12-13
SMT202100709T1 (it) 2022-01-10
JP6867652B2 (ja) 2021-05-12
EP3386997B1 (en) 2021-06-30
HUE056897T2 (hu) 2022-03-28
JP2018538292A (ja) 2018-12-27
MX377528B (es) 2025-03-10
PL3386997T3 (pl) 2021-12-13
DK3386997T3 (da) 2021-09-20
PT3386997T (pt) 2021-11-04
RS62412B1 (sr) 2021-10-29
AU2016367306B2 (en) 2021-04-22
CY1124529T1 (el) 2022-07-22
US20210002313A1 (en) 2021-01-07

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