AU2015205374B2 - Bicyclic heterocyclyl derivatives as IRAK4 inhibitors - Google Patents

Bicyclic heterocyclyl derivatives as IRAK4 inhibitors Download PDF

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Publication number
AU2015205374B2
AU2015205374B2 AU2015205374A AU2015205374A AU2015205374B2 AU 2015205374 B2 AU2015205374 B2 AU 2015205374B2 AU 2015205374 A AU2015205374 A AU 2015205374A AU 2015205374 A AU2015205374 A AU 2015205374A AU 2015205374 B2 AU2015205374 B2 AU 2015205374B2
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Prior art keywords
pyridin
oxazole
carboxamide
mmol
piperidin
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AU2015205374A1 (en
Inventor
Venkateshwar Rao Gummadi
Susanta Samajdar
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Aurigene Oncology Ltd
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Aurigene Oncology Ltd
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Priority to AU2018267569A priority Critical patent/AU2018267569B2/en
Priority to AU2019283795A priority patent/AU2019283795B2/en
Priority to AU2021203761A priority patent/AU2021203761B2/en
Assigned to AURIGENE ONCOLOGY LIMITED reassignment AURIGENE ONCOLOGY LIMITED Request to Amend Deed and Register Assignors: AURIGENE DISCOVERY TECHNOLOGIES LIMITED
Priority to AU2023222987A priority patent/AU2023222987B2/en
Priority to AU2025226775A priority patent/AU2025226775A1/en
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    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
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AU2015205374A 2014-01-13 2015-01-12 Bicyclic heterocyclyl derivatives as IRAK4 inhibitors Active AU2015205374B2 (en)

Priority Applications (5)

Application Number Priority Date Filing Date Title
AU2018267569A AU2018267569B2 (en) 2014-01-13 2018-11-20 Bicyclic heterocyclyl derivatives as IRAK4 inhibitors
AU2019283795A AU2019283795B2 (en) 2014-01-13 2019-12-17 Bicyclic heterocyclyl derivatives as IRAK4 inhibitors
AU2021203761A AU2021203761B2 (en) 2014-01-13 2021-06-08 Bicyclic heterocyclyl derivatives as IRAK4 inhibitors
AU2023222987A AU2023222987B2 (en) 2014-01-13 2023-09-01 Bicyclic heterocyclyl derivatives as IRAK4 inhibitors
AU2025226775A AU2025226775A1 (en) 2014-01-13 2025-09-04 Bicyclic heterocyclyl derivatives as IRAK4 inhibitors

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
IN158CH2014 2014-01-13
IN158/CHE/2014 2014-01-13
IN3000CH2014 2014-06-20
IN3000/CHE/2014 2014-06-20
PCT/IB2015/050217 WO2015104688A1 (en) 2014-01-13 2015-01-12 Bicyclic heterocyclyl derivatives as irak4 inhibitors

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AU2018267569A Division AU2018267569B2 (en) 2014-01-13 2018-11-20 Bicyclic heterocyclyl derivatives as IRAK4 inhibitors

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AU2015205374A1 AU2015205374A1 (en) 2016-07-28
AU2015205374B2 true AU2015205374B2 (en) 2018-08-23

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AU2015205374A Active AU2015205374B2 (en) 2014-01-13 2015-01-12 Bicyclic heterocyclyl derivatives as IRAK4 inhibitors
AU2018267569A Active AU2018267569B2 (en) 2014-01-13 2018-11-20 Bicyclic heterocyclyl derivatives as IRAK4 inhibitors
AU2019283795A Active AU2019283795B2 (en) 2014-01-13 2019-12-17 Bicyclic heterocyclyl derivatives as IRAK4 inhibitors
AU2021203761A Active AU2021203761B2 (en) 2014-01-13 2021-06-08 Bicyclic heterocyclyl derivatives as IRAK4 inhibitors
AU2023222987A Active AU2023222987B2 (en) 2014-01-13 2023-09-01 Bicyclic heterocyclyl derivatives as IRAK4 inhibitors
AU2025226775A Pending AU2025226775A1 (en) 2014-01-13 2025-09-04 Bicyclic heterocyclyl derivatives as IRAK4 inhibitors

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AU2018267569A Active AU2018267569B2 (en) 2014-01-13 2018-11-20 Bicyclic heterocyclyl derivatives as IRAK4 inhibitors
AU2019283795A Active AU2019283795B2 (en) 2014-01-13 2019-12-17 Bicyclic heterocyclyl derivatives as IRAK4 inhibitors
AU2021203761A Active AU2021203761B2 (en) 2014-01-13 2021-06-08 Bicyclic heterocyclyl derivatives as IRAK4 inhibitors
AU2023222987A Active AU2023222987B2 (en) 2014-01-13 2023-09-01 Bicyclic heterocyclyl derivatives as IRAK4 inhibitors
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