HUE052252T2 - Eljárás IRAK4 inhibitorként rák kezelésére alkalmas oxazolo[4,5-b]piridin és tiazolo[4,5-b]piridin származékok elõállítására - Google Patents

Eljárás IRAK4 inhibitorként rák kezelésére alkalmas oxazolo[4,5-b]piridin és tiazolo[4,5-b]piridin származékok elõállítására

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Publication number
HUE052252T2
HUE052252T2 HUE18190333A HUE18190333A HUE052252T2 HU E052252 T2 HUE052252 T2 HU E052252T2 HU E18190333 A HUE18190333 A HU E18190333A HU E18190333 A HUE18190333 A HU E18190333A HU E052252 T2 HUE052252 T2 HU E052252T2
Authority
HU
Hungary
Prior art keywords
pyridine
oxazolo
thiazolo
preparing
treating cancer
Prior art date
Application number
HUE18190333A
Other languages
English (en)
Inventor
Venkateshwar Gummadi
Susanta Samajdar
Original Assignee
Aurigene Discovery Tech Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aurigene Discovery Tech Ltd filed Critical Aurigene Discovery Tech Ltd
Publication of HUE052252T2 publication Critical patent/HUE052252T2/hu

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    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
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    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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HUE18190333A 2014-01-13 2015-01-12 Eljárás IRAK4 inhibitorként rák kezelésére alkalmas oxazolo[4,5-b]piridin és tiazolo[4,5-b]piridin származékok elõállítására HUE052252T2 (hu)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN158CH2014 2014-01-13
IN3000CH2014 2014-06-20

Publications (1)

Publication Number Publication Date
HUE052252T2 true HUE052252T2 (hu) 2021-04-28

Family

ID=53523587

Family Applications (2)

Application Number Title Priority Date Filing Date
HUE15735499A HUE041926T2 (hu) 2014-01-13 2015-01-12 IRAK4 inhibitor biciklusos heterociklilszármazékok
HUE18190333A HUE052252T2 (hu) 2014-01-13 2015-01-12 Eljárás IRAK4 inhibitorként rák kezelésére alkalmas oxazolo[4,5-b]piridin és tiazolo[4,5-b]piridin származékok elõállítására

Family Applications Before (1)

Application Number Title Priority Date Filing Date
HUE15735499A HUE041926T2 (hu) 2014-01-13 2015-01-12 IRAK4 inhibitor biciklusos heterociklilszármazékok

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US (6) US9732095B2 (hu)
EP (4) EP3466955B1 (hu)
JP (5) JP6479850B2 (hu)
KR (3) KR102574390B1 (hu)
CN (2) CN111362966B (hu)
AU (5) AU2015205374B2 (hu)
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DK (3) DK3094329T3 (hu)
EA (2) EA031913B1 (hu)
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HR (2) HRP20181795T1 (hu)
HU (2) HUE041926T2 (hu)
IL (6) IL302878B1 (hu)
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PH (2) PH12016501344A1 (hu)
PL (3) PL3094329T3 (hu)
PT (3) PT3094329T (hu)
RS (3) RS61448B1 (hu)
SG (2) SG10201811204RA (hu)
SI (2) SI3094329T1 (hu)
TR (1) TR201815683T4 (hu)
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Families Citing this family (42)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB201311891D0 (en) 2013-07-03 2013-08-14 Glaxosmithkline Ip Dev Ltd Novel compound
GB201311888D0 (en) 2013-07-03 2013-08-14 Glaxosmithkline Ip Dev Ltd Novel compounds
SG11201605408RA (en) 2014-01-10 2016-07-28 Aurigene Discovery Tech Ltd Indazole compounds as irak4 inhibitors
SI3094329T1 (sl) 2014-01-13 2019-02-28 Aurigene Discovery Technologies Limited Biciklični heterociklilni derivati kot inhibitorji IRAK4
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