AU2012351942B2 - Fluorinated estrogen receptor modulators and uses thereof - Google Patents

Fluorinated estrogen receptor modulators and uses thereof Download PDF

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Publication number
AU2012351942B2
AU2012351942B2 AU2012351942A AU2012351942A AU2012351942B2 AU 2012351942 B2 AU2012351942 B2 AU 2012351942B2 AU 2012351942 A AU2012351942 A AU 2012351942A AU 2012351942 A AU2012351942 A AU 2012351942A AU 2012351942 B2 AU2012351942 B2 AU 2012351942B2
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substituted
unsubstituted
compound
pharmaceutically acceptable
cancer
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AU2012351942A1 (en
Inventor
Celine Bonnefous
Steven P. Govek
Mehmet Kahraman
Andiliy G. Lai
Johnny Y. Nagasawa
Nicholas D. Smith
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Seragon Pharmaceuticals Inc
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Seragon Pharmaceuticals Inc
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    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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  • Health & Medical Sciences (AREA)
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  • Diabetes (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Psychiatry (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Oncology (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Hospice & Palliative Care (AREA)
  • Addiction (AREA)
  • Obesity (AREA)
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AU2012351942A 2011-12-14 2012-12-14 Fluorinated estrogen receptor modulators and uses thereof Ceased AU2012351942B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161570756P 2011-12-14 2011-12-14
US61/570,756 2011-12-14
PCT/US2012/069933 WO2013090836A1 (en) 2011-12-14 2012-12-14 Fluorinated estrogen receptor modulators and uses thereof

Publications (2)

Publication Number Publication Date
AU2012351942A1 AU2012351942A1 (en) 2014-06-12
AU2012351942B2 true AU2012351942B2 (en) 2017-07-06

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AU2012351942A Ceased AU2012351942B2 (en) 2011-12-14 2012-12-14 Fluorinated estrogen receptor modulators and uses thereof

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US (2) US9193714B2 (cg-RX-API-DMAC7.html)
EP (2) EP2791133B1 (cg-RX-API-DMAC7.html)
JP (2) JP2015500346A (cg-RX-API-DMAC7.html)
KR (1) KR20140101399A (cg-RX-API-DMAC7.html)
CN (1) CN104114551B (cg-RX-API-DMAC7.html)
AU (1) AU2012351942B2 (cg-RX-API-DMAC7.html)
BR (1) BR112014014124A2 (cg-RX-API-DMAC7.html)
CA (1) CA2857057A1 (cg-RX-API-DMAC7.html)
EA (1) EA029559B1 (cg-RX-API-DMAC7.html)
HK (1) HK1198165A1 (cg-RX-API-DMAC7.html)
IL (1) IL232793A (cg-RX-API-DMAC7.html)
MX (1) MX357496B (cg-RX-API-DMAC7.html)
PH (1) PH12014501351A1 (cg-RX-API-DMAC7.html)
SG (1) SG11201403002RA (cg-RX-API-DMAC7.html)
WO (2) WO2013090836A1 (cg-RX-API-DMAC7.html)

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US9193714B2 (en) 2011-12-14 2015-11-24 Seragon Pharmaceuticals, Inc. Fluorinated estrogen receptor modulators and uses thereof
MD20140054A2 (ro) 2011-12-16 2014-10-31 Olema Pharmaceuticals, Inc. Compuşi noi de benzopiran, compoziţii şi utilizări ale acestora
BR112015030595A2 (pt) 2013-06-19 2017-07-25 Seragon Pharmaceuticals Inc moduladores de receptor de estrogênio de azetidina e usos dos mesmos
BR112015031903A8 (pt) 2013-06-19 2019-12-31 Seragon Pharmaceuticals Inc composto, sal farmaceuticamente aceitável, composição farmacêutica e uso de um composto
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