AU2005318959B2 - Crystalline forms of (R)-8-chloro-1-methyl- 2,3,4,5-tetrahydro-1H-3-benzazepine hydrochloride - Google Patents

Crystalline forms of (R)-8-chloro-1-methyl- 2,3,4,5-tetrahydro-1H-3-benzazepine hydrochloride Download PDF

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AU2005318959B2
AU2005318959B2 AU2005318959A AU2005318959A AU2005318959B2 AU 2005318959 B2 AU2005318959 B2 AU 2005318959B2 AU 2005318959 A AU2005318959 A AU 2005318959A AU 2005318959 A AU2005318959 A AU 2005318959A AU 2005318959 B2 AU2005318959 B2 AU 2005318959B2
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disorder
compound according
pharmaceutical composition
compound
treatment
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AU2005318959A1 (en
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Rajesh Kumar Agarwal
Iii William L. Betts
James A. Henshilwood
Yuan-Hon Kiang
Noah Post
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Arena Pharmaceuticals Inc
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/14—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D223/16—Benzazepines; Hydrogenated benzazepines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
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    • A61P3/04—Anorexiants; Antiobesity agents
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  • Diabetes (AREA)
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  • Endocrinology (AREA)
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  • Obesity (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pulmonology (AREA)
  • Heart & Thoracic Surgery (AREA)
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  • Hospice & Palliative Care (AREA)
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  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
AU2005318959A 2004-12-21 2005-12-20 Crystalline forms of (R)-8-chloro-1-methyl- 2,3,4,5-tetrahydro-1H-3-benzazepine hydrochloride Expired AU2005318959B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US63822104P 2004-12-21 2004-12-21
US60/638,221 2004-12-21
PCT/US2005/046983 WO2006069363A2 (en) 2004-12-21 2005-12-20 Crystalline forms of (r)-8-chloro-1-methyl- 2,3,4,5-tetrahydro-1h-3-benzazepine hydrochloride

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AU2005318959A1 AU2005318959A1 (en) 2006-06-29
AU2005318959B2 true AU2005318959B2 (en) 2011-12-15

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AU2005318959A Expired AU2005318959B2 (en) 2004-12-21 2005-12-20 Crystalline forms of (R)-8-chloro-1-methyl- 2,3,4,5-tetrahydro-1H-3-benzazepine hydrochloride

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US (4) US8168624B2 (enExample)
EP (3) EP2149562A1 (enExample)
JP (3) JP5270167B2 (enExample)
KR (1) KR101281919B1 (enExample)
CN (2) CN101084193B (enExample)
AT (1) ATE442359T1 (enExample)
AU (1) AU2005318959B2 (enExample)
BR (1) BRPI0519726B8 (enExample)
CA (1) CA2589988C (enExample)
CU (1) CU20070138A7 (enExample)
CY (1) CY1109599T1 (enExample)
DE (1) DE602005016603D1 (enExample)
DK (1) DK1838677T3 (enExample)
EA (2) EA017894B1 (enExample)
ES (1) ES2332009T3 (enExample)
HR (1) HRP20090640T1 (enExample)
IL (1) IL183844A (enExample)
MA (1) MA29147B1 (enExample)
ME (1) ME01090B (enExample)
NI (1) NI200700160A (enExample)
NZ (2) NZ589756A (enExample)
PL (1) PL1838677T3 (enExample)
PT (1) PT1838677E (enExample)
RS (1) RS50996B (enExample)
SI (1) SI1838677T1 (enExample)
TN (1) TNSN07235A1 (enExample)
WO (1) WO2006069363A2 (enExample)
ZA (1) ZA200705125B (enExample)

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CN116270646A (zh) 2015-10-16 2023-06-23 艾伯维公司 制备咪唑并[1,2-a]吡咯并[2,3-e]吡嗪类化合物及其固态形式的方法
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