CY1109599T1 - Κρυσταλλικες μορφες υδροχλωρικης (r)-8-χλωρο-1-μεθυλο-2,3,4,5-τετραϋδρο-1η-3-βενζαζεπινης - Google Patents

Κρυσταλλικες μορφες υδροχλωρικης (r)-8-χλωρο-1-μεθυλο-2,3,4,5-τετραϋδρο-1η-3-βενζαζεπινης

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Publication number
CY1109599T1
CY1109599T1 CY20091101162T CY091101162T CY1109599T1 CY 1109599 T1 CY1109599 T1 CY 1109599T1 CY 20091101162 T CY20091101162 T CY 20091101162T CY 091101162 T CY091101162 T CY 091101162T CY 1109599 T1 CY1109599 T1 CY 1109599T1
Authority
CY
Cyprus
Prior art keywords
tetrahydro
chloro
methyl
benzazepine
hydrochloric
Prior art date
Application number
CY20091101162T
Other languages
English (en)
Inventor
Rajesh Kumar Agarwal
Iii William L Betts
James A Henshilwood
Yuan-Hon Kiang
Noah Post
Original Assignee
Arena Pharmaceuticals, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36602366&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY1109599(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Arena Pharmaceuticals, Inc. filed Critical Arena Pharmaceuticals, Inc.
Publication of CY1109599T1 publication Critical patent/CY1109599T1/el

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/14—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D223/16—Benzazepines; Hydrogenated benzazepines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/16—Central respiratory analeptics
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
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    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/32—Alcohol-abuse
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    • A61P25/36—Opioid-abuse
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    • A61P3/04—Anorexiants; Antiobesity agents
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    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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    • A61P7/12—Antidiuretics, e.g. drugs for diabetes insipidus
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    • A61P9/00—Drugs for disorders of the cardiovascular system

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  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Obesity (AREA)
  • Pulmonology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
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  • Anesthesiology (AREA)
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  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)

Abstract

Η παρούσα εφεύρεση αφορά σε κρυσταλλικές μορφές (R)-8-χλωρο-1-μεθυλο-2,3,4,5-τετραϋδρο-1Η-3-βενζαζεπίνης, σε συνθέσεις που τις περιέχουν, σε σκευάσματα και χρήσεις αυτών.
CY20091101162T 2004-12-21 2009-11-10 Κρυσταλλικες μορφες υδροχλωρικης (r)-8-χλωρο-1-μεθυλο-2,3,4,5-τετραϋδρο-1η-3-βενζαζεπινης CY1109599T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US63822104P 2004-12-21 2004-12-21
EP05855526A EP1838677B1 (en) 2004-12-21 2005-12-20 Crystalline forms of (r)-8-chloro-1-methyl- 2,3,4,5-tetrahydro-1h-3-benzazepine hydrochloride

Publications (1)

Publication Number Publication Date
CY1109599T1 true CY1109599T1 (el) 2014-08-13

Family

ID=36602366

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20091101162T CY1109599T1 (el) 2004-12-21 2009-11-10 Κρυσταλλικες μορφες υδροχλωρικης (r)-8-χλωρο-1-μεθυλο-2,3,4,5-τετραϋδρο-1η-3-βενζαζεπινης

Country Status (29)

Country Link
US (4) US8168624B2 (el)
EP (3) EP1838677B1 (el)
JP (3) JP5270167B2 (el)
KR (1) KR101281919B1 (el)
CN (2) CN101084193B (el)
AT (1) ATE442359T1 (el)
AU (1) AU2005318959B2 (el)
BR (1) BRPI0519726B8 (el)
CA (1) CA2589988C (el)
CU (1) CU20070138A7 (el)
CY (1) CY1109599T1 (el)
DE (1) DE602005016603D1 (el)
DK (1) DK1838677T3 (el)
EA (2) EA201200954A1 (el)
ES (1) ES2332009T3 (el)
HK (2) HK1102812A1 (el)
HR (1) HRP20090640T1 (el)
IL (1) IL183844A (el)
MA (1) MA29147B1 (el)
ME (1) ME01090B (el)
NI (1) NI200700160A (el)
NZ (2) NZ555981A (el)
PL (1) PL1838677T3 (el)
PT (1) PT1838677E (el)
RS (1) RS50996B (el)
SI (1) SI1838677T1 (el)
TN (1) TNSN07235A1 (el)
WO (1) WO2006069363A2 (el)
ZA (1) ZA200705125B (el)

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