AU2001272476A1 - Piperidines for use as orexin receptor antagonists - Google Patents

Piperidines for use as orexin receptor antagonists

Info

Publication number
AU2001272476A1
AU2001272476A1 AU2001272476A AU7247601A AU2001272476A1 AU 2001272476 A1 AU2001272476 A1 AU 2001272476A1 AU 2001272476 A AU2001272476 A AU 2001272476A AU 7247601 A AU7247601 A AU 7247601A AU 2001272476 A1 AU2001272476 A1 AU 2001272476A1
Authority
AU
Australia
Prior art keywords
optionally substituted
phenyl
heteroatoms selected
heteroaryl group
group containing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2001272476A
Other languages
English (en)
Inventor
Clive Leslie Branch
Christopher Norbert Johnson
Geoffrey Stemp
Kevin Thewlis
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SmithKline Beecham Ltd
Original Assignee
SmithKline Beecham Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0014823A external-priority patent/GB0014823D0/en
Priority claimed from GB0027704A external-priority patent/GB0027704D0/en
Application filed by SmithKline Beecham Ltd filed Critical SmithKline Beecham Ltd
Publication of AU2001272476A1 publication Critical patent/AU2001272476A1/en
Abandoned legal-status Critical Current

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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07D211/26—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by nitrogen atoms
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AU2001272476A 2000-06-16 2001-06-13 Piperidines for use as orexin receptor antagonists Abandoned AU2001272476A1 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GB0014823A GB0014823D0 (en) 2000-06-16 2000-06-16 Compounds
GB0014823 2000-06-16
GB0027704A GB0027704D0 (en) 2000-11-11 2000-11-11 Compounds
GB0027704 2000-11-11
PCT/EP2001/006752 WO2001096302A1 (fr) 2000-06-16 2001-06-13 Piperidines utiles en tant qu'antagonistes du recepteur d'orexine

Publications (1)

Publication Number Publication Date
AU2001272476A1 true AU2001272476A1 (en) 2001-12-24

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Family Applications (1)

Application Number Title Priority Date Filing Date
AU2001272476A Abandoned AU2001272476A1 (en) 2000-06-16 2001-06-13 Piperidines for use as orexin receptor antagonists

Country Status (10)

Country Link
US (1) US6677354B2 (fr)
EP (1) EP1289955B1 (fr)
JP (1) JP4611608B2 (fr)
AT (1) ATE293101T1 (fr)
AU (1) AU2001272476A1 (fr)
CA (1) CA2450922C (fr)
DE (1) DE60110066T2 (fr)
ES (1) ES2238458T3 (fr)
PT (1) PT1289955E (fr)
WO (1) WO2001096302A1 (fr)

Families Citing this family (138)

* Cited by examiner, † Cited by third party
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EP1353918B1 (fr) * 2000-11-28 2005-01-12 Smithkline Beecham Plc Derives de la morpholine utilises comme antagonistes des recepteurs de l'orexine
HUP0400048A3 (en) * 2001-05-05 2008-10-28 Smithkline Beecham Plc N-aroyl cyclic amines and pharmaceutical compositions containing them
WO2002089800A2 (fr) * 2001-05-05 2002-11-14 Smithkline Beecham P.L.C. Derives d'amines cycliques n-aroyl utilises comme antagonistes du recepteur d'orexine
GB0115862D0 (en) * 2001-06-28 2001-08-22 Smithkline Beecham Plc Compounds
US7470710B2 (en) 2001-06-28 2008-12-30 Smithkline Beecham P.L.C. N-aroyl cyclic amine derivatives as orexin receptor antagonists
GB0124463D0 (en) * 2001-10-11 2001-12-05 Smithkline Beecham Plc Compounds
GB0126292D0 (en) * 2001-11-01 2002-01-02 Smithkline Beecham Plc Compounds
GB0127145D0 (en) 2001-11-10 2002-01-02 Smithkline Beecham Compounds
US20090286791A1 (en) * 2001-11-27 2009-11-19 Takeda Pharmaceutical Company Limited Amide Compounds
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