AR228937A1 - Procedimiento para preparar derivados de pentapeptidos de tyr-ala-gly-me-nh2 o lev-nh2 o cys(et)-nh2 o cys-(p-metoxibencilo) - Google Patents

Procedimiento para preparar derivados de pentapeptidos de tyr-ala-gly-me-nh2 o lev-nh2 o cys(et)-nh2 o cys-(p-metoxibencilo)

Info

Publication number
AR228937A1
AR228937A1 AR269298A AR26929877A AR228937A1 AR 228937 A1 AR228937 A1 AR 228937A1 AR 269298 A AR269298 A AR 269298A AR 26929877 A AR26929877 A AR 26929877A AR 228937 A1 AR228937 A1 AR 228937A1
Authority
AR
Argentina
Prior art keywords
cys
metoxibencilo
pentapeptides
lev
tyr
Prior art date
Application number
AR269298A
Other languages
English (en)
Spanish (es)
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Application granted granted Critical
Publication of AR228937A1 publication Critical patent/AR228937A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
    • C07K14/70—Enkephalins
    • C07K14/702—Enkephalins with at least 1 amino acid in D-form
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Zoology (AREA)
  • Toxicology (AREA)
  • Neurology (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AR269298A 1976-09-27 1977-09-22 Procedimiento para preparar derivados de pentapeptidos de tyr-ala-gly-me-nh2 o lev-nh2 o cys(et)-nh2 o cys-(p-metoxibencilo) AR228937A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US72672476A 1976-09-27 1976-09-27
US05/807,849 US4259234A (en) 1976-09-27 1977-06-20 Analgesic compounds

Publications (1)

Publication Number Publication Date
AR228937A1 true AR228937A1 (es) 1983-05-13

Family

ID=27111374

Family Applications (1)

Application Number Title Priority Date Filing Date
AR269298A AR228937A1 (es) 1976-09-27 1977-09-22 Procedimiento para preparar derivados de pentapeptidos de tyr-ala-gly-me-nh2 o lev-nh2 o cys(et)-nh2 o cys-(p-metoxibencilo)

Country Status (27)

Country Link
US (1) US4259234A (ro)
JP (1) JPS5340736A (ro)
AR (1) AR228937A1 (ro)
AT (1) AT359219B (ro)
AU (1) AU513702B2 (ro)
CA (1) CA1201710A (ro)
CH (2) CH636847A5 (ro)
CS (1) CS204011B2 (ro)
DD (1) DD132862A5 (ro)
DE (1) DE2741393A1 (ro)
DK (1) DK148904C (ro)
ES (1) ES462658A1 (ro)
FR (1) FR2365553A1 (ro)
GB (1) GB1586521A (ro)
GR (1) GR69224B (ro)
HK (1) HK52681A (ro)
HU (1) HU180723B (ro)
IE (1) IE45576B1 (ro)
IL (1) IL52872A (ro)
MY (1) MY8200150A (ro)
NL (1) NL7710502A (ro)
NZ (1) NZ185084A (ro)
PL (1) PL111136B1 (ro)
PT (1) PT67026B (ro)
RO (1) RO80379B (ro)
SE (1) SE438339B (ro)
SU (1) SU753358A3 (ro)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4261888A (en) * 1976-04-12 1981-04-14 Sandoz Ltd. Organic compounds
ZA775285B (en) * 1976-09-01 1978-07-26 A Kastin Novel methionine enkephalin derivatives
HU178001B (en) * 1976-09-16 1982-02-28 Gyogyszekutato Intezet Process for preparing new pentapeptides with morphine-like activity and derivatives thereof
US4322342A (en) * 1977-06-20 1982-03-30 Eli Lilly And Company Analgesic compounds
EP0000559B1 (en) * 1977-07-22 1983-10-05 The Wellcome Foundation Limited Pentapeptide-n-alkylamides and their acid addition salts, methods for preparation of these compounds and pharmaceutical formulations containing them
US4264491A (en) * 1977-10-03 1981-04-28 Eli Lilly And Company Analgesic compounds
FR2424253A1 (fr) * 1978-04-27 1979-11-23 Brun Lab Sa Le Nouveaux derives de peptides analogues des enkephalines, leur procede de preparation et leur application therapeutique
DE2933947A1 (de) * 1979-08-22 1981-03-12 Hoechst Ag, 6000 Frankfurt Neue peptidamide und verfahren zu ihrer herstellung.
US4254024A (en) * 1979-10-16 1981-03-03 Pennwalt Corporation Tetrapeptides and derivatives having opiate activity
US4351763A (en) * 1979-12-17 1982-09-28 Eli Lilly And Company Pharmacologically active peptides
US4283329A (en) * 1979-12-17 1981-08-11 Eli Lilly And Company Pharmacologically active peptides
US4265808A (en) * 1979-12-17 1981-05-05 Eli Lilly And Company Pharmacologically active peptides
US4251439A (en) * 1979-12-17 1981-02-17 Eli Lilly And Company Pharmacologically active peptides
US4283330A (en) * 1979-12-17 1981-08-11 Eli Lilly And Company Pharmacologically active peptides
FR2488253A1 (fr) * 1980-08-08 1982-02-12 Roques Bernard Nouveaux peptides et leur application en therapeutique
US4322339A (en) * 1980-10-20 1982-03-30 Eli Lilly And Company Pharmacologically active peptides
ATE16495T1 (de) * 1981-06-22 1985-11-15 Ici Plc Peptide und pseudopeptide, die zwei substituenten am n-terminus aufweisen.
US4430327A (en) 1982-05-18 1984-02-07 Eli Lilly And Company Method for treating pregnant females for pain and anxiety
DE3915755A1 (de) * 1989-05-13 1990-11-29 Bayer Ag Fungizide mittel sowie substituierte aminosaeureamid-derivate und deren herstellung
DE4102042A1 (de) * 1991-01-24 1992-07-30 Bayer Ag Substituierte aminosaeureamid-derivate deren herstellung und verwendung als fungizide
JPH09173654A (ja) * 1995-12-21 1997-07-08 Ritsuwa Yo 積 木
EP1297830A1 (en) * 2001-09-28 2003-04-02 Flamma Fabbrica Lombarda Ammino Acidi S.p.a. Use of alpha- or beta-amino acids, of the corresponding esters or of dipeptides of these amino acids with histidine derivatives in the prevention or treatment of tissue damage caused by a atmospheric ozone

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1532181A (en) * 1976-02-02 1978-11-15 Beckman Instruments Inc Pentapetides and a method of preparing them
FI770219A (ro) * 1976-02-02 1977-08-03 Sandoz Ag
NZ183712A (en) * 1976-04-08 1979-10-25 Ici Ltd Polypeptide analogues of enkephalins, and pharmaceutical compositions
ZA775285B (en) * 1976-09-01 1978-07-26 A Kastin Novel methionine enkephalin derivatives
HU178001B (en) * 1976-09-16 1982-02-28 Gyogyszekutato Intezet Process for preparing new pentapeptides with morphine-like activity and derivatives thereof
US4178371A (en) * 1977-12-15 1979-12-11 Reckitt & Colman Products Limited Tetrapeptide derivatives

Also Published As

Publication number Publication date
SU753358A3 (ru) 1980-07-30
AU513702B2 (en) 1980-12-18
NZ185084A (en) 1980-11-14
MY8200150A (en) 1982-12-31
GB1586521A (en) 1981-03-18
DK424577A (da) 1978-03-28
CH643533A5 (de) 1984-06-15
ES462658A1 (es) 1978-11-01
RO80379B (ro) 1983-04-30
CA1201710A (en) 1986-03-11
ATA685977A (de) 1980-03-15
AU2856577A (en) 1979-03-15
DD132862A5 (de) 1978-11-15
PL201049A1 (pl) 1979-01-29
CS204011B2 (en) 1981-03-31
CH636847A5 (de) 1983-06-30
IL52872A (en) 1983-07-31
DK148904C (da) 1986-04-14
PT67026B (en) 1979-02-14
FR2365553B1 (ro) 1980-11-14
AT359219B (de) 1980-10-27
RO80379A (ro) 1983-04-29
HU180723B (en) 1983-04-29
PT67026A (en) 1977-10-01
SE438339B (sv) 1985-04-15
IE45576B1 (en) 1982-10-06
DK148904B (da) 1985-11-11
DE2741393C2 (ro) 1988-03-10
DE2741393A1 (de) 1978-03-30
JPS6254800B2 (ro) 1987-11-17
JPS5340736A (en) 1978-04-13
US4259234A (en) 1981-03-31
SE7710755L (sv) 1978-03-28
PL111136B1 (en) 1980-08-30
HK52681A (en) 1981-11-06
NL7710502A (nl) 1978-03-29
IE45576L (en) 1978-03-27
GR69224B (ro) 1982-05-10
FR2365553A1 (fr) 1978-04-21

Similar Documents

Publication Publication Date Title
AR228937A1 (es) Procedimiento para preparar derivados de pentapeptidos de tyr-ala-gly-me-nh2 o lev-nh2 o cys(et)-nh2 o cys-(p-metoxibencilo)
SE7811689L (sv) Forfarande for framstellning av maytansinoider
ES494635A0 (es) Procedimiento de preparacion de derivados de tiadiazol
RO76807A (ro) Procedeu pentru prepararea unor derivati de hidantoina
AR228940A1 (es) Procedimiento para preparar derivados de 4-desacetil vlb c-3 carboxi-hidrazida
NO151895C (no) Fremgangsmaate for fremstilling av pyrido-indolderivater
IT1142606B (it) Fabbricazione perfezionata di glicoletilenico da gas sintetico
RO72258A (ro) Procedeu pentru prepararea unor derivati ai n-fosfonometilglicinei
AR222691A1 (es) Procedimiento de preparacion de derivados hidroxi-de 2-isopropilamino-pirimidina
DK313878A (da) Indolderivater og fremgangsmaade til fremstilling deraf
MX5215E (es) Procedimiento de preparacion de derivados de tienopiridina
NO784382L (no) Fremgangsmaate for fremstilling av tiazoldin-derivater
AR211570A1 (es) Procedimiento de preparacion de nuevos derivados de 8-oxi-5-(2-hidroxi-3-aminopropoxi)-carbostirilo
AR231289A1 (es) Procedimiento para preparar derivados de quinolil-4-1-piperidilo-4-2-etanol o quinolil-4-1-piperidil-4-3-propanol
ES493569A0 (es) Procedimiento de preparar derivados isoquinolinicos
NO802435L (no) Fremgangsmaate til fremstilling av tetrahydrokinolinderivater
RO77027A (ro) Procedeu pentru prepararea unor derivati ai bis(nitrozoureido)-poliolilor
AR219746A1 (es) Procedimiento de preparacion de derivados de cromenilpropano
NO780389L (no) Fremgangsmaate for fremstilling av erytromycin-derivater
RO76166A (ro) Procedeu pentru prepararea unor derivati ai ergolinei
NO792659L (no) Fremgangsmaate for fremstilling av karbostyrilderivater
ES491004A0 (es) Procedimiento de preparacion de nuevos derivados halogenadosde isopropilamino-pirimidina
ES495745A0 (es) Procedimiento de preparacion de derivados de la piridina.
NO801724L (no) Fremgangsmaate for fremstilling av ergopeptin-derivater
AR220140A1 (es) Procedimiento para la preparacion de derivados de 1-(2-metilfenil)-tetrahidro-s-triazin-2-tiono con utiles propiedades pesticidas