AR121070A1 - Inhibidores de péptidos del receptor de interleucina-23 y su uso para tratar enfermedades inflamatorias - Google Patents

Inhibidores de péptidos del receptor de interleucina-23 y su uso para tratar enfermedades inflamatorias

Info

Publication number
AR121070A1
AR121070A1 ARP210100106A ARP210100106A AR121070A1 AR 121070 A1 AR121070 A1 AR 121070A1 AR P210100106 A ARP210100106 A AR P210100106A AR P210100106 A ARP210100106 A AR P210100106A AR 121070 A1 AR121070 A1 AR 121070A1
Authority
AR
Argentina
Prior art keywords
interleukin
peptide inhibitors
inflammatory diseases
treat inflammatory
receptor peptide
Prior art date
Application number
ARP210100106A
Other languages
English (en)
Spanish (es)
Inventor
Chengzao Sun
Brian Troy Frederick
Sandeep Somani
Gregory Thomas Bourne
Raymond Patch
Ashok Bhandari
Raffaele Ingenito
Roberto Costante
Danila Branca
Elisabetta Bianchi
Original Assignee
Janssen Biotech Inc
Protagonist Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Biotech Inc, Protagonist Therapeutics Inc filed Critical Janssen Biotech Inc
Publication of AR121070A1 publication Critical patent/AR121070A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/64Cyclic peptides containing only normal peptide links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/705Receptors; Cell surface antigens; Cell surface determinants
    • C07K14/715Receptors; Cell surface antigens; Cell surface determinants for cytokines; for lymphokines; for interferons
    • C07K14/7155Receptors; Cell surface antigens; Cell surface determinants for cytokines; for lymphokines; for interferons for interleukins [IL]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/08Linear peptides containing only normal peptide links having 12 to 20 amino acids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Immunology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Toxicology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Zoology (AREA)
  • Cell Biology (AREA)
  • Dermatology (AREA)
  • Epidemiology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Medicinal Preparation (AREA)
ARP210100106A 2020-01-15 2021-01-15 Inhibidores de péptidos del receptor de interleucina-23 y su uso para tratar enfermedades inflamatorias AR121070A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US202062961624P 2020-01-15 2020-01-15

Publications (1)

Publication Number Publication Date
AR121070A1 true AR121070A1 (es) 2022-04-13

Family

ID=76864704

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP210100106A AR121070A1 (es) 2020-01-15 2021-01-15 Inhibidores de péptidos del receptor de interleucina-23 y su uso para tratar enfermedades inflamatorias

Country Status (32)

Country Link
US (2) US11845808B2 (https=)
EP (2) EP4613761A3 (https=)
JP (2) JP7441955B2 (https=)
KR (1) KR20220141807A (https=)
CN (5) CN118005736A (https=)
AR (1) AR121070A1 (https=)
AU (1) AU2021207653A1 (https=)
CA (1) CA3167751A1 (https=)
CL (2) CL2022001893A1 (https=)
CO (1) CO2022009931A2 (https=)
CR (1) CR20220332A (https=)
DK (1) DK4090670T3 (https=)
DO (1) DOP2022000147A (https=)
EC (1) ECSP22063238A (https=)
ES (1) ES3036287T3 (https=)
FI (1) FI4090670T3 (https=)
HR (1) HRP20250769T1 (https=)
HU (1) HUE072238T2 (https=)
IL (1) IL294680A (https=)
JO (1) JOP20220169A1 (https=)
LT (1) LT4090670T (https=)
MA (1) MA58373B1 (https=)
MX (1) MX2022008741A (https=)
PE (1) PE20230370A1 (https=)
PH (1) PH12022551750A1 (https=)
PL (1) PL4090670T3 (https=)
PT (1) PT4090670T (https=)
RS (1) RS66991B1 (https=)
SI (1) SI4090670T1 (https=)
SM (1) SMT202500254T1 (https=)
TW (2) TWI882061B (https=)
WO (1) WO2021146441A1 (https=)

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CN114341161A (zh) * 2019-07-10 2022-04-12 领导医疗有限公司 白细胞介素-23受体的肽抑制剂及其用于治疗炎症性疾病的用途
HRP20250769T1 (hr) * 2020-01-15 2025-08-29 Janssen Biotech, Inc. Peptidni inhibitori receptora za interleukin-23 i njihova uporaba u liječenju upalnih bolesti
AU2021209086A1 (en) 2020-01-15 2022-08-04 Janssen Biotech, Inc. Peptide inhibitors of interleukin-23 receptor and their use to treat inflammatory diseases
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CA3226539A1 (en) * 2021-07-14 2023-01-19 Janssen Biotech, Inc. Peptide inhibitors of interleukin-23 receptor
WO2023288019A2 (en) 2021-07-14 2023-01-19 Janssen Biotech, Inc. Lipidated peptide inhibitors of interleukin-23 receptor
WO2023004414A1 (en) * 2021-07-23 2023-01-26 Colorado Chromatography, Llc A method for preparing hexahydrocannabinol
CN118354781A (zh) 2021-12-01 2024-07-16 西兰制药公司 白介素-23受体的肽抑制剂
IL314629A (en) 2022-02-01 2024-09-01 Janssen Pharmaceutica Nv Peptide inhibitors of the interleukin-23 receptor and pharmaceutical preparations thereof
WO2023177452A1 (en) * 2022-03-14 2023-09-21 Colorado Chromatography, Llc Hydrogenation of cannabigerol and cannabichromene
CA3260606A1 (en) 2022-06-30 2024-01-04 Sanofi NEW PEPTIDES FOR USE AS SELECTIVE IL-23 RECEPTOR ANTAGONISTS
AU2023386710A1 (en) * 2022-11-21 2025-07-10 Janssen Pharmaceutica Nv Synthesis of a cyclic peptide
KR20250111134A (ko) * 2022-11-30 2025-07-22 상하이 한서 바이오메디컬 컴퍼니 리미티드 폴리펩티드 억제제, 이의 제조 방법 및 응용
EP4652182A1 (en) * 2023-01-16 2025-11-26 Janssen Pharmaceutica NV Peptide inhibitors of interleukin-23 receptor
EP4652180A2 (en) * 2023-01-16 2025-11-26 Janssen Pharmaceutica NV Peptide inhibitors of interleukin-23 receptor
EP4652179A1 (en) * 2023-01-16 2025-11-26 Janssen Pharmaceutica NV Lipidated peptide inhibitors of interleukin-23 receptor
KR20250139359A (ko) 2023-01-31 2025-09-23 얀센 파마슈티카 엔브이 인터류킨-23 수용체의 결정질 펩티드 억제제의 제조 방법
EP4676595A1 (en) * 2023-03-03 2026-01-14 Janssen Pharmaceutica NV Interleukin-23 receptor antagonist peptides for use in the treatment of psoriasis
WO2024227437A1 (zh) * 2023-05-04 2024-11-07 西藏海思科制药有限公司 白介素-23受体的肽抑制剂制备及其用途
EP4471048A1 (en) 2023-06-01 2024-12-04 Zealand Pharma A/S Peptide inhibitors of interleukin-23 receptor
EP4471049A1 (en) 2023-06-01 2024-12-04 Zealand Pharma A/S Peptide inhibitors of interleukin-23 receptor
CN121909205A (zh) * 2023-09-08 2026-04-21 赛诺菲 作为选择性il-23受体抑制剂的新型肽
WO2025163534A1 (en) 2024-01-31 2025-08-07 Janssen Pharmaceutica Nv Crystal form of a peptide inhibitor of interleukin-23 receptor
WO2025243217A1 (en) * 2024-05-22 2025-11-27 Janssen Pharmaceutica Nv Crystal forms of peptide molecules
WO2026013260A1 (en) 2024-07-12 2026-01-15 Zealand Pharma A/S Peptide inhibitors of interleukin-23 receptor
WO2026026816A1 (zh) * 2024-07-30 2026-02-05 西藏海思科制药有限公司 白介素-23受体的肽抑制剂及其用途
WO2026046292A1 (zh) * 2024-08-28 2026-03-05 西藏海思科制药有限公司 白介素-23受体的肽抑制剂的药物组合物及其制备方法和用途
WO2026057052A1 (zh) * 2024-09-14 2026-03-19 深圳信立泰药业股份有限公司 一种il-23受体抑制剂及其制备方法和用途
CN120905324A (zh) * 2025-10-10 2025-11-07 北京元延医药科技股份有限公司 白细胞介素-23受体肽抑制剂及其手性中间体的制法

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