AR018633A1 - Derivados de benzo(b)tiepin-1,1-dioxido, procedimiento para su preparacion, medicamentos conteniendo estos compuestos y su empleo - Google Patents

Derivados de benzo(b)tiepin-1,1-dioxido, procedimiento para su preparacion, medicamentos conteniendo estos compuestos y su empleo

Info

Publication number
AR018633A1
AR018633A1 ARP990102715A ARP990102715A AR018633A1 AR 018633 A1 AR018633 A1 AR 018633A1 AR P990102715 A ARP990102715 A AR P990102715A AR P990102715 A ARP990102715 A AR P990102715A AR 018633 A1 AR018633 A1 AR 018633A1
Authority
AR
Argentina
Prior art keywords
radical
compounds
preparation
alkyl
tiepin
Prior art date
Application number
ARP990102715A
Other languages
English (en)
Spanish (es)
Original Assignee
Gompel Marie
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gompel Marie filed Critical Gompel Marie
Publication of AR018633A1 publication Critical patent/AR018633A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D337/00Heterocyclic compounds containing rings of more than six members having one sulfur atom as the only ring hetero atom
    • C07D337/02Seven-membered rings
    • C07D337/06Seven-membered rings condensed with carbocyclic rings or ring systems
    • C07D337/08Seven-membered rings condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/351Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom not condensed with another ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/38Heterocyclic compounds having sulfur as a ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/04Drugs for disorders of the urinary system for urolithiasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06086Dipeptides with the first amino acid being basic
    • CCHEMISTRY; METALLURGY
    • C08ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08GMACROMOLECULAR COMPOUNDS OBTAINED OTHERWISE THAN BY REACTIONS ONLY INVOLVING UNSATURATED CARBON-TO-CARBON BONDS
    • C08G65/00Macromolecular compounds obtained by reactions forming an ether link in the main chain of the macromolecule
    • C08G65/02Macromolecular compounds obtained by reactions forming an ether link in the main chain of the macromolecule from cyclic ethers by opening of the heterocyclic ring
    • C08G65/32Polymers modified by chemical after-treatment
    • C08G65/329Polymers modified by chemical after-treatment with organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
ARP990102715A 1998-06-10 1999-06-08 Derivados de benzo(b)tiepin-1,1-dioxido, procedimiento para su preparacion, medicamentos conteniendo estos compuestos y su empleo AR018633A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19825804A DE19825804C2 (de) 1998-06-10 1998-06-10 1,4-Benzothiepin-1,1-dioxidderivate, Verfahren zu deren Herstellung und diese Verbindungen enthaltende Arzneimittel

Publications (1)

Publication Number Publication Date
AR018633A1 true AR018633A1 (es) 2001-11-28

Family

ID=7870440

Family Applications (2)

Application Number Title Priority Date Filing Date
ARP990102716A AR018634A1 (es) 1998-06-10 1999-06-08 Derivados de benzo(b)tiepin-1,1,-dioxido, procedimiento para su preparacion, medicamentos conteniendo estos compuestos, procedimiento para la preparacion de medicamentos y su empleo para la preparacion de medicamentos.
ARP990102715A AR018633A1 (es) 1998-06-10 1999-06-08 Derivados de benzo(b)tiepin-1,1-dioxido, procedimiento para su preparacion, medicamentos conteniendo estos compuestos y su empleo

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ARP990102716A AR018634A1 (es) 1998-06-10 1999-06-08 Derivados de benzo(b)tiepin-1,1,-dioxido, procedimiento para su preparacion, medicamentos conteniendo estos compuestos, procedimiento para la preparacion de medicamentos y su empleo para la preparacion de medicamentos.

Country Status (26)

Country Link
US (1) US6387944B1 (US06387944-20020514-C00002.png)
EP (2) EP1086092B1 (US06387944-20020514-C00002.png)
JP (2) JP4374426B2 (US06387944-20020514-C00002.png)
KR (2) KR100681721B1 (US06387944-20020514-C00002.png)
CN (2) CN1127497C (US06387944-20020514-C00002.png)
AR (2) AR018634A1 (US06387944-20020514-C00002.png)
AT (2) ATE227715T1 (US06387944-20020514-C00002.png)
AU (2) AU753275B2 (US06387944-20020514-C00002.png)
BR (2) BR9912188B1 (US06387944-20020514-C00002.png)
CA (2) CA2334775C (US06387944-20020514-C00002.png)
CZ (2) CZ297989B6 (US06387944-20020514-C00002.png)
DE (3) DE19825804C2 (US06387944-20020514-C00002.png)
DK (2) DK1086092T3 (US06387944-20020514-C00002.png)
ES (2) ES2182535T3 (US06387944-20020514-C00002.png)
HK (2) HK1039490A1 (US06387944-20020514-C00002.png)
HU (2) HU229761B1 (US06387944-20020514-C00002.png)
ID (2) ID28695A (US06387944-20020514-C00002.png)
IL (1) IL140078A (US06387944-20020514-C00002.png)
NO (1) NO327075B1 (US06387944-20020514-C00002.png)
NZ (1) NZ508681A (US06387944-20020514-C00002.png)
PL (2) PL196074B1 (US06387944-20020514-C00002.png)
PT (2) PT1086092E (US06387944-20020514-C00002.png)
RU (2) RU2215001C2 (US06387944-20020514-C00002.png)
TR (2) TR200003634T2 (US06387944-20020514-C00002.png)
WO (2) WO1999064410A1 (US06387944-20020514-C00002.png)
ZA (2) ZA200007060B (US06387944-20020514-C00002.png)

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DK1345895T3 (da) * 2000-12-21 2007-05-07 Sanofi Aventis Deutschland Hidtil ukendt diphenylazetidioner, fremgangsmåde til deres fremstilling, lægemidler indeholdende disse forbindelser og deres anvendelse til behandling af lipidstofskifteforstyrrelser
MXPA04001328A (es) * 2001-08-22 2004-05-05 Aventis Pharma Gmbh Productos en combinacion de derivados de 1,4-benzotiepina-1,1-dioxido con otros ingredientes activos, y su uso.
GB0121337D0 (en) 2001-09-04 2001-10-24 Astrazeneca Ab Chemical compounds
GB0121622D0 (en) 2001-09-07 2001-10-31 Astrazeneca Ab Chemical compounds
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CN1582151A (zh) 2001-09-08 2005-02-16 阿斯特拉曾尼卡有限公司 用于治疗高脂血症、具有回肠胆汁酸转运(ibat)抑制活性的苯并硫氮杂䓬和苯并硫杂二氮杂䓬衍生物
GB0209467D0 (en) 2002-04-25 2002-06-05 Astrazeneca Ab Chemical compounds
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CN107375932B (zh) 2011-10-28 2021-12-21 夏尔人类遗传性治疗公司 用于治疗小儿胆汁淤积性肝病的胆汁酸再循环抑制剂
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KR20220082931A (ko) 2014-06-25 2022-06-17 이에이 파마 가부시키가이샤 고형 제제 및 그의 착색 방지 또는 착색 감소 방법
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US11014898B1 (en) 2020-12-04 2021-05-25 Albireo Ab Benzothiazepine compounds and their use as bile acid modulators
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Also Published As

Publication number Publication date
ID28695A (id) 2001-06-28
AU753275B2 (en) 2002-10-10
IL140078A0 (en) 2002-02-10
CZ20004592A3 (cs) 2001-04-11
HK1036799A1 (en) 2002-01-18
CA2334773A1 (en) 1999-12-16
JP2002517490A (ja) 2002-06-18
HU228570B1 (en) 2013-04-29
CZ20004591A3 (cs) 2001-04-11
KR20010052682A (ko) 2001-06-25
NO20006251L (no) 2001-02-07
ZA200007060B (en) 2001-07-18
DE59908522D1 (de) 2004-03-18
HUP0102256A1 (hu) 2001-12-28
HUP0102554A3 (en) 2002-12-28
NZ508681A (en) 2002-06-28
PT1086113E (pt) 2004-06-30
JP2002517491A (ja) 2002-06-18
JP4374426B2 (ja) 2009-12-02
TR200003632T2 (tr) 2001-04-20
NO20006251D0 (no) 2000-12-08
PT1086092E (pt) 2003-03-31
ATE227715T1 (de) 2002-11-15
ZA200007061B (en) 2001-07-18
CN1305487A (zh) 2001-07-25
BR9911123A (pt) 2006-01-03
DE19825804C2 (de) 2000-08-24
CA2334775A1 (en) 1999-12-16
PL344827A1 (en) 2001-11-19
WO1999064409A2 (de) 1999-12-16
EP1086092A1 (de) 2001-03-28
HK1039490A1 (en) 2002-04-26
CN1305469A (zh) 2001-07-25
DK1086092T3 (da) 2003-03-10
NO327075B1 (no) 2009-04-20
KR20010052701A (ko) 2001-06-25
KR100562184B1 (ko) 2006-03-20
PL345901A1 (en) 2002-01-14
EP1086113A2 (de) 2001-03-28
ATE259372T1 (de) 2004-02-15
JP3374129B2 (ja) 2003-02-04
DE59903411D1 (de) 2002-12-19
AU4501999A (en) 1999-12-30
IL140078A (en) 2004-08-31
BR9912188B1 (pt) 2010-12-14
US6387944B1 (en) 2002-05-14
ES2215387T3 (es) 2004-10-01
HUP0102256A3 (en) 2002-04-29
HUP0102554A1 (hu) 2001-10-28
CA2334775C (en) 2009-10-13
EP1086113B1 (de) 2004-02-11
CZ297989B6 (cs) 2007-05-16
WO1999064409A3 (de) 2000-03-02
RU2220141C2 (ru) 2003-12-27
AU752633B2 (en) 2002-09-26
HU229761B1 (hu) 2014-06-30
EP1086092B1 (de) 2002-11-13
DE19825804A1 (de) 1999-12-16
CZ297925B6 (cs) 2007-05-02
RU2215001C2 (ru) 2003-10-27
CA2334773C (en) 2009-05-26
PL196057B1 (pl) 2007-11-30
AU4503199A (en) 1999-12-30
TR200003634T2 (tr) 2001-06-21
BR9912188A (pt) 2001-04-10
CN1127497C (zh) 2003-11-12
AR018634A1 (es) 2001-11-28
WO1999064410A1 (de) 1999-12-16
BR9911123B1 (pt) 2010-12-14
ID26876A (id) 2001-02-15
ES2182535T3 (es) 2003-03-01
DK1086113T3 (da) 2004-05-24
KR100681721B1 (ko) 2007-02-15
PL196074B1 (pl) 2007-12-31
CN1152039C (zh) 2004-06-02

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