AR009052A1 - Tienopirimidinas, un procedimiento para su preparacion, empleo de las mismas para preparar un medicamento, preparaciones farmaceuticas que lascontienen y un procedimiento para obtener estas preparaciones farmaceuticas - Google Patents

Tienopirimidinas, un procedimiento para su preparacion, empleo de las mismas para preparar un medicamento, preparaciones farmaceuticas que lascontienen y un procedimiento para obtener estas preparaciones farmaceuticas

Info

Publication number
AR009052A1
AR009052A1 ARP970103649A ARP970103649A AR009052A1 AR 009052 A1 AR009052 A1 AR 009052A1 AR P970103649 A ARP970103649 A AR P970103649A AR P970103649 A ARP970103649 A AR P970103649A AR 009052 A1 AR009052 A1 AR 009052A1
Authority
AR
Argentina
Prior art keywords
pharmaceutical preparations
procedure
hal
prepare
preparation
Prior art date
Application number
ARP970103649A
Other languages
English (en)
Spanish (es)
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of AR009052A1 publication Critical patent/AR009052A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/02Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Hospice & Palliative Care (AREA)
  • Gynecology & Obstetrics (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ARP970103649A 1996-08-12 1997-08-12 Tienopirimidinas, un procedimiento para su preparacion, empleo de las mismas para preparar un medicamento, preparaciones farmaceuticas que lascontienen y un procedimiento para obtener estas preparaciones farmaceuticas AR009052A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19632423A DE19632423A1 (de) 1996-08-12 1996-08-12 Thienopyrimidine

Publications (1)

Publication Number Publication Date
AR009052A1 true AR009052A1 (es) 2000-03-08

Family

ID=7802392

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP970103649A AR009052A1 (es) 1996-08-12 1997-08-12 Tienopirimidinas, un procedimiento para su preparacion, empleo de las mismas para preparar un medicamento, preparaciones farmaceuticas que lascontienen y un procedimiento para obtener estas preparaciones farmaceuticas

Country Status (28)

Country Link
US (1) US6110920A (https=)
EP (1) EP0920431B1 (https=)
JP (1) JP4405593B2 (https=)
KR (1) KR100502271B1 (https=)
CN (1) CN1081638C (https=)
AR (1) AR009052A1 (https=)
AT (1) ATE233265T1 (https=)
AU (1) AU725227B2 (https=)
BR (1) BR9711062A (https=)
CA (1) CA2263561C (https=)
CZ (1) CZ287772B6 (https=)
DE (2) DE19632423A1 (https=)
DK (1) DK0920431T3 (https=)
ES (1) ES2191192T3 (https=)
HU (1) HUP0001607A3 (https=)
IL (1) IL128504A (https=)
NO (1) NO990643L (https=)
NZ (1) NZ334600A (https=)
PL (1) PL190174B1 (https=)
PT (1) PT920431E (https=)
RU (1) RU2199541C2 (https=)
SI (1) SI0920431T1 (https=)
SK (1) SK282823B6 (https=)
TR (1) TR199900308T2 (https=)
TW (1) TW359672B (https=)
UA (1) UA55421C2 (https=)
WO (1) WO1998006722A1 (https=)
ZA (1) ZA977156B (https=)

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US6339106B1 (en) 1999-08-11 2002-01-15 Sepracor, Inc. Methods and compositions for the treatment and prevention of sexual dysfunction
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US6399826B1 (en) 1999-08-11 2002-06-04 Sepracor Inc. Salts of sibutramine metabolites, methods of making sibutramine metabolites and intermediates useful in the same, and methods of treating pain
DE19950647A1 (de) * 1999-10-21 2001-04-26 Merck Patent Gmbh Imidazolderivate als Phosphodiesterase VII-Hemmer
DE10031585A1 (de) * 2000-06-29 2002-01-10 Merck Patent Gmbh 2-Aminoalkyl-thieno[2,3-d]pyrimidine
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US6610887B2 (en) 2001-04-13 2003-08-26 Sepracor Inc. Methods of preparing didesmethylsibutramine and other sibutramine derivatives
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WO2003035653A1 (en) * 2001-10-26 2003-05-01 Nippon Soda Co.,Ltd. Pyridothienopyrimidine compound and salt thereof
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US7276529B2 (en) 2002-03-20 2007-10-02 Celgene Corporation Methods of the treatment or prevention of exercise-induced asthma using (+)-2-[1-(3-ethoxy-4-methoxyphenyl)-2-methylsulfonylethyl]-4-acetylaminoisoindoline-1,3-dione
US7208516B2 (en) 2002-03-20 2007-04-24 Celgene Corporation Methods of the treatment of psoriatic arthritis using (+)-2-[1-(3-ethoxy-4-methoxyphenyl)-2-methylsulfonylethyl]-4-acetylaminoisoindoline-1,3-dione
US7893101B2 (en) 2002-03-20 2011-02-22 Celgene Corporation Solid forms comprising (+)-2-[1-(3-ethoxy-4-methoxyphenyl)-2-methylsulfonylethyl]-4-acetylaminoisoindoline-1,3-dione, compositions thereof, and uses thereof
TW200410975A (en) * 2002-09-26 2004-07-01 Nihon Nohyaku Co Ltd New pesticide and method for using it, new substituted thienopyrimidine derivative, its intermediate, and method for producing it
GB0320300D0 (en) * 2003-08-29 2003-10-01 Cancer Rec Tech Ltd Pyrimidothiophene compounds
DE10351436A1 (de) * 2003-11-04 2005-06-09 Merck Patent Gmbh Verwendung von Thienopyrimidinen
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KR20220049612A (ko) 2014-01-21 2022-04-21 얀센 파마슈티카 엔.브이. 대사 조절형 글루탐산 작동성 수용체 제2아형의 양성 알로스테릭 조절제 또는 오르토스테릭 작동제를 포함하는 조합 및 그 용도
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JP7514005B2 (ja) 2017-06-21 2024-07-10 シャイ・セラピューティクス・エルエルシー がん、炎症性疾患、ラソパシー、及び線維性疾患の治療のためのrasスーパーファミリーと相互作用する化合物
JP7453210B2 (ja) 2018-08-07 2024-03-19 フィルメニッヒ インコーポレイテッド 5-置換4-アミノ-1H-ベンゾ[c][1,2,6]チアジアジン2,2-ジオキシド並びにその配合物及び使用
JP7407461B2 (ja) 2018-12-19 2024-01-04 シャイ・セラピューティクス・エルエルシー がん、炎症性疾患、ras病、及び線維性疾患の処置のためのrasスーパーファミリーと相互作用する化合物
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Also Published As

Publication number Publication date
IL128504A (en) 2003-01-12
JP4405593B2 (ja) 2010-01-27
ZA977156B (en) 1998-02-19
NO990643D0 (no) 1999-02-11
IL128504A0 (en) 2000-01-31
SI0920431T1 (en) 2003-08-31
SK16499A3 (en) 1999-06-11
CA2263561C (en) 2007-02-20
TR199900308T2 (xx) 1999-04-21
EP0920431B1 (de) 2003-02-26
DK0920431T3 (da) 2003-06-02
AU4203597A (en) 1998-03-06
PT920431E (pt) 2003-07-31
ATE233265T1 (de) 2003-03-15
US6110920A (en) 2000-08-29
CZ287772B6 (en) 2001-01-17
CZ44899A3 (cs) 1999-05-12
DE19632423A1 (de) 1998-02-19
HUP0001607A2 (hu) 2000-10-28
EP0920431A1 (de) 1999-06-09
KR100502271B1 (ko) 2005-07-22
RU2199541C2 (ru) 2003-02-27
HK1021731A1 (en) 2000-06-30
HUP0001607A3 (en) 2002-09-30
PL190174B1 (pl) 2005-11-30
UA55421C2 (uk) 2003-04-15
CN1227560A (zh) 1999-09-01
CA2263561A1 (en) 1998-02-19
KR20000029932A (ko) 2000-05-25
WO1998006722A1 (de) 1998-02-19
AU725227B2 (en) 2000-10-12
JP2000516223A (ja) 2000-12-05
DE59709404D1 (en) 2003-04-03
ES2191192T3 (es) 2003-09-01
TW359672B (en) 1999-06-01
CN1081638C (zh) 2002-03-27
NO990643L (no) 1999-02-11
NZ334600A (en) 2000-07-28
PL331538A1 (en) 1999-07-19
SK282823B6 (sk) 2002-12-03
BR9711062A (pt) 1999-08-17

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