AR008820A1 - Comprimido dotado de recubrimiento laminar de maleato de trimebutina, destinado ala administracion por via oral, y un procedimiento para prepararlo - Google Patents
Comprimido dotado de recubrimiento laminar de maleato de trimebutina, destinado ala administracion por via oral, y un procedimiento para prepararloInfo
- Publication number
- AR008820A1 AR008820A1 ARP970103538A ARP970103538A AR008820A1 AR 008820 A1 AR008820 A1 AR 008820A1 AR P970103538 A ARP970103538 A AR P970103538A AR P970103538 A ARP970103538 A AR P970103538A AR 008820 A1 AR008820 A1 AR 008820A1
- Authority
- AR
- Argentina
- Prior art keywords
- preparing
- intended
- trimebutine maleate
- administration
- procedure
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/235—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group
- A61K31/24—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group having an amino or nitro group
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
Abstract
Comprimido dotado de recubrimiento laminar de maleato de trimebutina destinado a la administracion por vía oral, caracterizado por comprender: -unnucleo que comprende de 30 a 60% de maleato de trimebutina, y excipientes adaptados a lapreparacion de dicho nucleo siendo éstos apropiados a la estabilidad y a la liberacion del principio activo, - un recubrimiento laminar hidrosoluble, de eficacia transitoria pero suficiente para preservar ladesintegracion al nucleo y de laliberacion p rematura del principio activo en el medio bucal. Un procedimiento para la fabricacion de comprimidos queconsiste en un primer momento en preparar un compuesto apropiado y después someterlo a compresion para obtener los nucleos que sondotados a continuacion de envolvente laminar.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9609956A FR2752162B1 (fr) | 1996-08-07 | 1996-08-07 | Comprime de maleate de trimebutine pellicule |
Publications (1)
Publication Number | Publication Date |
---|---|
AR008820A1 true AR008820A1 (es) | 2000-02-23 |
Family
ID=9494890
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP970103538A AR008820A1 (es) | 1996-08-07 | 1997-08-04 | Comprimido dotado de recubrimiento laminar de maleato de trimebutina, destinado ala administracion por via oral, y un procedimiento para prepararlo |
Country Status (27)
Country | Link |
---|---|
EP (1) | EP0942718B1 (es) |
JP (1) | JP2000515535A (es) |
KR (1) | KR100539642B1 (es) |
CN (1) | CN1206986C (es) |
AR (1) | AR008820A1 (es) |
AT (1) | ATE300297T1 (es) |
AU (1) | AU3697097A (es) |
BR (1) | BR9711032B1 (es) |
CA (1) | CA2256751C (es) |
CO (1) | CO4900042A1 (es) |
CZ (1) | CZ294195B6 (es) |
DZ (1) | DZ2272A1 (es) |
EA (1) | EA001506B1 (es) |
ES (2) | ES2244002T3 (es) |
FR (1) | FR2752162B1 (es) |
GR (1) | GR1002907B (es) |
HK (1) | HK1020888A1 (es) |
HU (1) | HU228040B1 (es) |
IT (1) | IT1294671B1 (es) |
MX (2) | MXPA98010007A (es) |
OA (1) | OA10968A (es) |
PL (1) | PL188839B1 (es) |
PT (2) | PT942718E (es) |
TN (1) | TNSN97134A1 (es) |
TR (1) | TR199900261T2 (es) |
UA (1) | UA52682C2 (es) |
WO (1) | WO1998005320A1 (es) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PE20001302A1 (es) | 1998-11-27 | 2000-11-30 | Hoffmann La Roche | Preparaciones de una combinacion farmaceutica que contiene carvedilol e hidroclorotiazida |
FR2834889B1 (fr) | 2002-01-18 | 2004-04-02 | Roquette Freres | Forme pharmaceutique solide orodispersible |
US20030181488A1 (en) | 2002-03-07 | 2003-09-25 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Administration form for the oral application of 3-[(2-{[4-(hexyloxycarbonylamino-imino-methyl)-phenylamino]-methyl}-1-methyl-1H-benzimidazol-5-carbonyl)-pyridin-2-yl-amino]-propionic acid ethyl ester and the salts thereof |
US7125563B2 (en) * | 2002-04-12 | 2006-10-24 | Dava Pharmaceuticals, Inc. | Sustained release pharmaceutical preparations and methods for producing the same |
EP1726621A1 (en) * | 2005-05-26 | 2006-11-29 | Cytec Surface Specialties, S.A. | Thermosetting powder compositions |
CN100393311C (zh) * | 2006-01-26 | 2008-06-11 | 孙伟丰 | 马来酸曲美布汀分散片 |
CN1927185B (zh) * | 2006-10-19 | 2010-05-19 | 开开援生制药股份有限公司 | 具速释部分的马来酸曲美布汀缓释片及其制备工艺 |
BRPI0916689A2 (pt) | 2008-07-28 | 2015-11-17 | Takeda Pharmaceutical | composição farmacêutica estabilizada, preparação sólida, e, métodos para estabilizar uma composição farmacêutica, e para estabilizar uma preparação sólida. |
KR101048487B1 (ko) * | 2008-08-19 | 2011-07-11 | 한국콜마 주식회사 | 말레인산트리메부틴 서방정 |
KR101220829B1 (ko) * | 2010-07-16 | 2013-01-10 | 안국약품 주식회사 | 트리메부틴 함유 서방성 정제 |
CN102462657A (zh) * | 2010-11-15 | 2012-05-23 | 杭州赛利药物研究所有限公司 | 马来酸曲美布汀栓剂及其制备方法 |
WO2014148520A1 (ja) * | 2013-03-21 | 2014-09-25 | 大正製薬株式会社 | 固形製剤 |
RU2536254C1 (ru) * | 2013-11-26 | 2014-12-20 | Общество С Ограниченной Ответственностью "Валента-Интеллект" | Таблетки-ретард с тримебутином |
CN107205984B (zh) * | 2015-01-26 | 2019-11-12 | 第一三共株式会社 | 吡咯甲酰胺的固体组合物 |
RU2706166C2 (ru) * | 2017-11-20 | 2019-11-14 | Общество С Ограниченной Ответственностью "Валента - Интеллект" | Новые полиморфные формы тримебутина малеата, способ получения и применения |
RU2770300C2 (ru) * | 2019-10-17 | 2022-04-15 | Общество С Ограниченной Ответственностью "Валента - Интеллект" | Новые полиморфные формы тримебутина малеата, способ получения и применения |
RU2770301C2 (ru) * | 2019-10-17 | 2022-04-15 | Общество С Ограниченной Ответственностью "Валента - Интеллект" | Новые полиморфные формы тримебутина малеата, способ получения и применения |
CN113171353B (zh) * | 2021-04-25 | 2022-10-21 | 海南普利制药股份有限公司 | 一种马来酸曲美布汀片 |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS6045845B2 (ja) * | 1979-10-31 | 1985-10-12 | 田辺製薬株式会社 | 医薬物質含有マイクロカプセルの製法 |
JPS57197214A (en) * | 1981-05-29 | 1982-12-03 | Tanabe Seiyaku Co Ltd | Rapid-releasing microcapsule and its preparation |
JPS5858146A (ja) * | 1981-10-05 | 1983-04-06 | Tanabe Seiyaku Co Ltd | 速放性マイクロカプセル |
JPS5858145A (ja) * | 1981-10-05 | 1983-04-06 | Tanabe Seiyaku Co Ltd | 速放性マイクロカプセル |
JPS5916821A (ja) * | 1982-07-16 | 1984-01-28 | Tanabe Seiyaku Co Ltd | 非凝集性マイクロカプセルの製法 |
FR2640876B1 (es) * | 1988-12-28 | 1993-09-24 | Jouveinal Sa | |
JPH03275622A (ja) * | 1990-03-26 | 1991-12-06 | Teisan Seiyaku Kk | マレイン酸トリメブチンを含有する経口固形製剤 |
JP2836493B2 (ja) * | 1994-08-04 | 1998-12-14 | 田辺製薬株式会社 | 苦味隠蔽されたマレイン酸トリメブチン含有製剤 |
-
1996
- 1996-08-07 FR FR9609956A patent/FR2752162B1/fr not_active Expired - Lifetime
-
1997
- 1997-07-11 EA EA199900102A patent/EA001506B1/ru not_active IP Right Cessation
- 1997-07-11 KR KR10-1999-7001031A patent/KR100539642B1/ko not_active IP Right Cessation
- 1997-07-11 HU HU9902878A patent/HU228040B1/hu unknown
- 1997-07-11 PT PT97933713T patent/PT942718E/pt unknown
- 1997-07-11 JP JP10507659A patent/JP2000515535A/ja not_active Ceased
- 1997-07-11 BR BRPI9711032-9A patent/BR9711032B1/pt not_active IP Right Cessation
- 1997-07-11 AT AT97933713T patent/ATE300297T1/de active
- 1997-07-11 WO PCT/FR1997/001281 patent/WO1998005320A1/fr active IP Right Grant
- 1997-07-11 AU AU36970/97A patent/AU3697097A/en not_active Abandoned
- 1997-07-11 TR TR1999/00261T patent/TR199900261T2/xx unknown
- 1997-07-11 PL PL97331517A patent/PL188839B1/pl unknown
- 1997-07-11 ES ES97933713T patent/ES2244002T3/es not_active Expired - Lifetime
- 1997-07-11 EP EP97933713A patent/EP0942718B1/fr not_active Expired - Lifetime
- 1997-07-11 CZ CZ1999376A patent/CZ294195B6/cs not_active IP Right Cessation
- 1997-07-11 MX MXPA98010007A patent/MXPA98010007A/es active IP Right Grant
- 1997-07-11 CA CA002256751A patent/CA2256751C/en not_active Expired - Lifetime
- 1997-07-11 CN CNB971967903A patent/CN1206986C/zh not_active Expired - Lifetime
- 1997-07-18 GR GR970100284A patent/GR1002907B/el unknown
- 1997-07-21 DZ DZ970122A patent/DZ2272A1/fr active
- 1997-07-24 ES ES009701642A patent/ES2130081B1/es not_active Expired - Fee Related
- 1997-07-25 PT PT102031A patent/PT102031B/pt active IP Right Grant
- 1997-08-04 AR ARP970103538A patent/AR008820A1/es active IP Right Grant
- 1997-08-05 TN TNTNSN97134A patent/TNSN97134A1/fr unknown
- 1997-08-06 CO CO97045253A patent/CO4900042A1/es unknown
- 1997-08-06 IT IT97GE000067A patent/IT1294671B1/it active IP Right Grant
- 1997-08-07 MX MX9706053A patent/MX9706053A/es unknown
- 1997-11-07 UA UA99031234A patent/UA52682C2/uk unknown
-
1999
- 1999-01-29 OA OA9900020A patent/OA10968A/fr unknown
-
2000
- 2000-01-03 HK HK00100007A patent/HK1020888A1/xx not_active IP Right Cessation
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG | Grant, registration |