AP2014008137A0 - Camsylate salt - Google Patents

Camsylate salt

Info

Publication number
AP2014008137A0
AP2014008137A0 AP2014008137A AP2014008137A AP2014008137A0 AP 2014008137 A0 AP2014008137 A0 AP 2014008137A0 AP 2014008137 A AP2014008137 A AP 2014008137A AP 2014008137 A AP2014008137 A AP 2014008137A AP 2014008137 A0 AP2014008137 A0 AP 2014008137A0
Authority
AP
ARIPO
Prior art keywords
camsylate salt
camsylate
salt
Prior art date
Application number
AP2014008137A
Other languages
English (en)
Inventor
Craig Robert Stewart
Martin Hans Bohlin
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of AP2014008137A0 publication Critical patent/AP2014008137A0/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/10Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
AP2014008137A 2012-06-21 2013-06-20 Camsylate salt AP2014008137A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261662592P 2012-06-21 2012-06-21
PCT/GB2013/051606 WO2013190302A1 (en) 2012-06-21 2013-06-20 Camsylate salt

Publications (1)

Publication Number Publication Date
AP2014008137A0 true AP2014008137A0 (en) 2014-12-31

Family

ID=48746084

Family Applications (2)

Application Number Title Priority Date Filing Date
AP2014008137A AP2014008137A0 (en) 2012-06-21 2013-06-20 Camsylate salt
AP2017009693A AP2017009693A0 (en) 2012-06-21 2013-06-20 Camsylate salt

Family Applications After (1)

Application Number Title Priority Date Filing Date
AP2017009693A AP2017009693A0 (en) 2012-06-21 2013-06-20 Camsylate salt

Country Status (42)

Country Link
US (1) US10548882B2 (zh)
EP (2) EP2864316B1 (zh)
JP (2) JP2015520221A (zh)
KR (1) KR102123708B1 (zh)
CN (2) CN104411697B (zh)
AP (2) AP2014008137A0 (zh)
AR (2) AR091495A1 (zh)
AU (2) AU2013279109B2 (zh)
BR (2) BR122016014302B1 (zh)
CA (1) CA2875589C (zh)
CL (1) CL2014003374A1 (zh)
CO (1) CO7151486A2 (zh)
CR (2) CR20140571A (zh)
CY (1) CY1119505T1 (zh)
DK (1) DK2864316T3 (zh)
DO (1) DOP2014000268A (zh)
EC (1) ECSP14032215A (zh)
ES (1) ES2618939T3 (zh)
HK (1) HK1206349A1 (zh)
HR (1) HRP20170359T1 (zh)
HU (1) HUE033376T2 (zh)
IL (1) IL236131A0 (zh)
IN (1) IN2014DN10088A (zh)
LT (1) LT2864316T (zh)
MA (2) MA39259B1 (zh)
ME (1) ME02633B (zh)
MX (1) MX354214B (zh)
NI (1) NI201400146A (zh)
NZ (2) NZ727045A (zh)
PE (1) PE20150670A1 (zh)
PH (2) PH12014502803B1 (zh)
PL (1) PL2864316T3 (zh)
PT (1) PT2864316T (zh)
RS (1) RS55815B1 (zh)
RU (1) RU2638175C2 (zh)
SG (1) SG11201407934UA (zh)
SI (1) SI2864316T1 (zh)
TN (1) TN2014000491A1 (zh)
TW (2) TWI639591B (zh)
UA (1) UA114196C2 (zh)
WO (1) WO2013190302A1 (zh)
ZA (1) ZA201500408B (zh)

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US8415483B2 (en) 2010-12-22 2013-04-09 Astrazeneca Ab Compounds and their use as BACE inhibitors
US9650336B2 (en) 2011-10-10 2017-05-16 Astrazeneca Ab Mono-fluoro beta-secretase inhibitors
US9000184B2 (en) 2012-06-20 2015-04-07 Astrazeneca Ab Cyclohexane-1,2′-naphthalene-1′,2″-imidazol compounds and their use as BACE inhibitors
US9000185B2 (en) 2012-06-20 2015-04-07 Astrazeneca Ab Cycloalkyl ether compounds and their use as BACE inhibitors
US9000183B2 (en) 2012-06-20 2015-04-07 Astrazeneca Ab Cyclohexane-1,2′-indene-1′,2″-imidazol compounds and their use as BACE inhibitors
US9000182B2 (en) 2012-06-20 2015-04-07 Astrazeneca Ab 2H-imidazol-4-amine compounds and their use as BACE inhibitors
TW201629025A (zh) 2014-10-07 2016-08-16 阿斯特捷利康公司 化合物及其作為bace抑制劑之用途
JP6546410B2 (ja) * 2015-02-23 2019-07-17 ローム株式会社 電力供給装置、acアダプタ、acチャージャ、電子機器および電力供給システム
TW201742625A (zh) 2016-03-15 2017-12-16 阿斯特捷利康公司 組合療法
TW201740944A (zh) * 2016-03-15 2017-12-01 美國禮來大藥廠 組合療法
US20220175749A1 (en) * 2019-03-14 2022-06-09 Astrazeneca Ab Lanabecestat for weight loss

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KR100452491B1 (ko) * 2001-03-29 2004-10-12 한미약품 주식회사 신규한 결정형 암로디핀 캠실레이트 염 및 그의 제조방법
WO2002098462A1 (fr) 2001-06-01 2002-12-12 Ono Pharmaceutical Co., Ltd. Remedes contenant un inhibiteur d'aldose reductase en tant qu'agent actif destines a des troubles de demyelinisation ou des troubles associes a la demyelinisation
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WO2007100536A1 (en) 2006-02-24 2007-09-07 Wyeth DIHYDROSPIRO[DIBENZO[A,D][7]ANNULENE-5,4'-IMIDAZOL] COMPOUNDS FOR THE INHIBITION OF β-SECRETASE
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WO2008092877A2 (en) 2007-02-01 2008-08-07 Glaxo Group Limited 8-oxa-1, 4-diazaspiro [4,5] dec-3-en-1-yl and 1,4, 8-triazaspiro [4,5] dec- 3-en-1-yl acetamides as glyti transporter inhibitors in treatment of neurological and neuropsychiatric disorders
RU2009144998A (ru) 2007-05-07 2011-06-20 Шеринг Корпорейшн (US) Модуляторы гамма-секретазы
WO2009100169A1 (en) 2008-02-06 2009-08-13 Glaxo Group Limited Dual pharmacophores - pde4-muscarinic antagonistics
FR2929943B1 (fr) * 2008-04-15 2010-09-24 Inst Rech Developpement Ird Sels de quinoleines 2-substituees
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AR077365A1 (es) 2009-07-02 2011-08-24 Astrazeneca Ab Derivados de imidazol para el tratamiento de enfermedades mediadas por la inhibicion de la formacion de abeta
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WO2011106414A1 (en) 2010-02-24 2011-09-01 Dillard Lawrence W Inhibitors of beta-secretase
AR080865A1 (es) 2010-03-31 2012-05-16 Array Biopharma Inc Derivados de espirotetrahidronaftaleno, composiciones farmaceuticas que los contienen, proceso de preparacion y uso de los mismos para tratar enfermedades neurodegenerativas,tal como alzheimer.
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US8415483B2 (en) 2010-12-22 2013-04-09 Astrazeneca Ab Compounds and their use as BACE inhibitors
US9650336B2 (en) 2011-10-10 2017-05-16 Astrazeneca Ab Mono-fluoro beta-secretase inhibitors
US9000183B2 (en) 2012-06-20 2015-04-07 Astrazeneca Ab Cyclohexane-1,2′-indene-1′,2″-imidazol compounds and their use as BACE inhibitors
US9000182B2 (en) 2012-06-20 2015-04-07 Astrazeneca Ab 2H-imidazol-4-amine compounds and their use as BACE inhibitors
US9000185B2 (en) 2012-06-20 2015-04-07 Astrazeneca Ab Cycloalkyl ether compounds and their use as BACE inhibitors
US9000184B2 (en) 2012-06-20 2015-04-07 Astrazeneca Ab Cyclohexane-1,2′-naphthalene-1′,2″-imidazol compounds and their use as BACE inhibitors

Also Published As

Publication number Publication date
MX354214B (es) 2018-02-19
IL236131A0 (en) 2015-02-01
PL2864316T3 (pl) 2017-09-29
US20140031379A1 (en) 2014-01-30
AU2013279109B2 (en) 2017-08-31
CR20160202A (es) 2016-07-26
TN2014000491A1 (en) 2016-03-30
BR122016014302B1 (pt) 2022-08-23
AU2013279109A1 (en) 2015-01-15
CA2875589A1 (en) 2013-12-27
ZA201500408B (en) 2016-10-26
PT2864316T (pt) 2017-02-24
HUE033376T2 (en) 2017-11-28
MA37666B1 (fr) 2016-12-30
PH12014502803A1 (en) 2015-02-23
US10548882B2 (en) 2020-02-04
RS55815B1 (sr) 2017-08-31
EP2864316B1 (en) 2016-12-14
JP2015520221A (ja) 2015-07-16
CY1119505T1 (el) 2018-03-07
RU2014148305A (ru) 2016-08-10
AR091495A1 (es) 2015-02-11
JP6509393B2 (ja) 2019-05-08
SG11201407934UA (en) 2015-01-29
TW201730177A (zh) 2017-09-01
EP3064494A1 (en) 2016-09-07
NI201400146A (es) 2016-09-21
CR20140571A (es) 2015-02-04
TW201406745A (zh) 2014-02-16
MA39259B1 (fr) 2018-09-28
AR105176A2 (es) 2017-09-13
MX2014014709A (es) 2015-03-04
MA39259A1 (fr) 2017-12-29
AP2017009693A0 (en) 2017-01-31
CA2875589C (en) 2020-08-25
MA37666A1 (fr) 2016-04-29
AU2017254965B2 (en) 2019-05-09
CN106279102A (zh) 2017-01-04
KR102123708B1 (ko) 2020-06-16
BR122016014302A2 (pt) 2019-08-27
DK2864316T3 (en) 2017-03-20
PH12014502803B1 (en) 2015-02-23
AU2017254965A1 (en) 2017-11-23
LT2864316T (lt) 2017-03-27
ECSP14032215A (es) 2015-12-31
ES2618939T3 (es) 2017-06-22
HK1206349A1 (zh) 2016-01-08
TWI588140B (zh) 2017-06-21
HRP20170359T1 (hr) 2017-05-05
PH12016500498A1 (en) 2017-04-10
SI2864316T1 (sl) 2017-04-26
IN2014DN10088A (zh) 2015-08-21
NZ702742A (en) 2016-12-23
ME02633B (me) 2017-06-20
KR20150023388A (ko) 2015-03-05
BR112014031531A2 (pt) 2017-06-27
RU2638175C2 (ru) 2017-12-12
DOP2014000268A (es) 2015-04-15
CN104411697A (zh) 2015-03-11
JP2018104448A (ja) 2018-07-05
CN104411697B (zh) 2016-08-10
TWI639591B (zh) 2018-11-01
NZ727045A (en) 2018-06-29
WO2013190302A1 (en) 2013-12-27
UA114196C2 (uk) 2017-05-10
CO7151486A2 (es) 2014-12-29
PE20150670A1 (es) 2015-06-03
BR112014031531B1 (pt) 2022-08-02
EP2864316A1 (en) 2015-04-29
CL2014003374A1 (es) 2015-02-27

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