ZA974336B - Vitamin D3 analogs. - Google Patents

Vitamin D3 analogs.

Info

Publication number
ZA974336B
ZA974336B ZA9704336A ZA974336A ZA974336B ZA 974336 B ZA974336 B ZA 974336B ZA 9704336 A ZA9704336 A ZA 9704336A ZA 974336 A ZA974336 A ZA 974336A ZA 974336 B ZA974336 B ZA 974336B
Authority
ZA
South Africa
Prior art keywords
analogs
vitamin
Prior art date
Application number
ZA9704336A
Other languages
English (en)
Inventor
Andrew David Batcho
Graeme Findlay Bryce
Bernard Michael Hennessy
Jerome Anthony Iacobelli
Milan Radoje Uskokovic
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of ZA974336B publication Critical patent/ZA974336B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C401/00Irradiation products of cholesterol or its derivatives; Vitamin D derivatives, 9,10-seco cyclopenta[a]phenanthrene or analogues obtained by chemical preparation without irradiation
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/02Nutrients, e.g. vitamins, minerals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nutrition Science (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
ZA9704336A 1996-05-23 1997-05-19 Vitamin D3 analogs. ZA974336B (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US1818696P 1996-05-23 1996-05-23
US1815396P 1996-05-23 1996-05-23
US3990097P 1997-03-19 1997-03-19

Publications (1)

Publication Number Publication Date
ZA974336B true ZA974336B (en) 1997-11-24

Family

ID=27360973

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA9704336A ZA974336B (en) 1996-05-23 1997-05-19 Vitamin D3 analogs.

Country Status (29)

Country Link
EP (2) EP0808833B1 (fr)
JP (1) JP2859247B2 (fr)
KR (1) KR100783856B1 (fr)
CN (1) CN1176072C (fr)
AR (1) AR007241A1 (fr)
AT (1) ATE277008T1 (fr)
AU (1) AU723929B2 (fr)
BR (1) BR9703384A (fr)
CA (1) CA2205275C (fr)
CO (1) CO4950531A1 (fr)
CZ (1) CZ157897A3 (fr)
DE (1) DE69730774T2 (fr)
DK (1) DK0808833T3 (fr)
ES (1) ES2227635T3 (fr)
HR (1) HRP970273A2 (fr)
HU (1) HUP9700926A3 (fr)
IL (1) IL120843A0 (fr)
MA (1) MA24251A1 (fr)
NO (1) NO972304L (fr)
NZ (1) NZ314839A (fr)
PE (1) PE70198A1 (fr)
PL (1) PL320132A1 (fr)
PT (1) PT808833E (fr)
SG (1) SG70009A1 (fr)
TR (1) TR199700415A2 (fr)
TW (1) TW445252B (fr)
UY (1) UY24561A1 (fr)
YU (1) YU20197A (fr)
ZA (1) ZA974336B (fr)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5939408A (en) 1996-05-23 1999-08-17 Hoffman-La Roche Inc. Vitamin D3 analogs
AU737376B2 (en) * 1997-02-25 2001-08-16 Regents Of The University Of Michigan, The Methods and compositions for preventing and treating chronological aging in human skin
AU743514B2 (en) * 1997-05-16 2002-01-24 Women & Infants Hospital Cyclic ether vitamin D3 compounds, 1alpha (OH) 3-EPI-vitamin D3 compounds and uses thereof
JP2002506429A (ja) * 1997-05-16 2002-02-26 ウィメン アンド インファンツ ホスピタル 3−エピビタミンd2化合物及びその使用法
EP0957098A1 (fr) * 1998-05-14 1999-11-17 F. Hoffmann-La Roche Ag Intermédiaires pour la synthèse de métabolites de la 3-épi vitamine D3 et analogues
US6603030B1 (en) 1999-04-22 2003-08-05 Hoffman-La Roche Inc. Process for producing phosphineoxide vitamin D precursors
EP3146969B1 (fr) * 1999-04-23 2018-06-20 Leo Pharma A/S Pommade pour le traitement topique du psoriasis
US6255501B1 (en) 1999-04-26 2001-07-03 Hoffman-La Roche Inc. Process for preparing antiosteoporotic agents
WO2001040177A2 (fr) * 1999-12-02 2001-06-07 Women And Infants Hospital Esters de vitamine d3 et utilisation de ces ceux-ci
GB2407499B (en) * 2003-11-03 2008-02-27 Bioxell Spa Vitamin D3 analogue for use in the treatment of BPH
CH698144B1 (fr) * 2003-09-24 2009-05-29 Bioxell Spa Analogue de la vitamine D3
SG110107A1 (en) 2003-09-24 2005-04-28 Bioxell Spa Compound and use in treatment
EP1737468A2 (fr) 2004-03-01 2007-01-03 Bioxell S.p.a. Methodes permettant de traiter la cystite interstitielle et composes et compositions connexes
EP1812011A1 (fr) 2004-11-12 2007-08-01 Bioxell S.p.a. Emploi combiné de dérivés de vitamine d et d'agents antiproliférants pour le traitement de cancers de la vessie
JP5449767B2 (ja) * 2005-04-25 2014-03-19 サイトクロマ インコーポレイテッド 1α,25−ジヒドロキシビタミンD3の低血漿カルシウム上昇性16,23−ジエン−25−オキシムアナログ
KR20080050420A (ko) * 2005-08-18 2008-06-05 비옥셀 에스.피.에이. 1α-플루오로-25-히드록시-16-23E-디엔-26,27-비스호모-20-에피-콜레칼시페롤의 합성
WO2008091686A2 (fr) * 2007-01-25 2008-07-31 Bioxell S.P.A. SYNTHÈSE DU 1α-FLUORO-25-HYDROXY-16-23E-DIÈNE-26,27-BISHOMO-20-ÉPI-CHOLÉCALCIFÉROL
JP5480131B2 (ja) 2007-05-30 2014-04-23 シトクロマ インコーポレイテッド ホスフィンオキシドビタミンd前駆物質の製造方法
ES2366077B2 (es) * 2010-03-30 2012-06-25 Universidade De Vigo Compuestos quirales, procedimientos de obtención y uso.
SG189427A1 (en) * 2010-10-25 2013-05-31 Teijin Pharma Ltd 23-yne-vitamin d3 derivative
CN105348164B (zh) * 2015-10-29 2017-03-29 无锡福祈制药有限公司 一种1α‑羟基维生素D2的制备方法
CN106748942B (zh) * 2016-11-28 2018-06-29 无锡福祈制药有限公司 度骨化醇类似物wxfq-65及其合成方法
ES2731558B2 (es) * 2018-05-15 2020-03-18 Univ Santiago Compostela Compuestos de interés farmacéutico
CN109738252B (zh) * 2019-01-23 2021-03-09 深圳天辰医疗科技有限公司 25-羟基-维生素d解离液
CN109696435B (zh) * 2019-01-25 2021-03-09 深圳天辰医疗科技有限公司 维生素d的测定方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA8923B (en) * 1988-01-20 1989-09-27 Hoffmann La Roche 16-dehydro-vitamin d3-derivatives
GB8914963D0 (en) * 1989-06-29 1989-08-23 Leo Pharm Prod Ltd Chemical compounds
GB9017890D0 (en) * 1990-08-15 1990-09-26 Leo Pharm Prod Ltd Chemical compounds i
GB9206648D0 (en) * 1992-03-26 1992-05-06 Leo Pharm Prod Ltd Chemical compounds
ES2091515T3 (es) * 1992-05-20 1996-11-01 Hoffmann La Roche Analogos fluorados de la vitamina d3.
US5428029A (en) * 1993-11-24 1995-06-27 Hoffmann-La Roche Inc. Vitamin D3 fluorinated analogs
JP3228488B2 (ja) * 1993-12-24 2001-11-12 株式会社クラレ 20−エピステロイド誘導体およびその製造方法

Also Published As

Publication number Publication date
CZ157897A3 (en) 1997-12-17
EP1464640A2 (fr) 2004-10-06
NO972304L (no) 1997-11-24
EP1464640A3 (fr) 2005-01-12
KR100783856B1 (ko) 2008-05-09
PL320132A1 (en) 1997-11-24
ATE277008T1 (de) 2004-10-15
IL120843A0 (en) 1997-09-30
SG70009A1 (en) 2000-01-25
TR199700415A3 (tr) 1997-12-21
KR970074765A (ko) 1997-12-10
TR199700415A2 (xx) 1997-12-21
CA2205275A1 (fr) 1997-11-23
NZ314839A (en) 2000-01-28
BR9703384A (pt) 1998-09-15
NO972304D0 (no) 1997-05-21
PE70198A1 (es) 1998-11-26
EP0808833A3 (fr) 1998-11-25
HUP9700926A2 (hu) 1998-01-28
HRP970273A2 (en) 1998-04-30
CA2205275C (fr) 2007-04-03
DE69730774D1 (de) 2004-10-28
ES2227635T3 (es) 2005-04-01
CN1175573A (zh) 1998-03-11
AR007241A1 (es) 1999-10-27
AU2357797A (en) 1997-11-27
AU723929B2 (en) 2000-09-07
CO4950531A1 (es) 2000-09-01
PT808833E (pt) 2004-11-30
UY24561A1 (es) 2000-12-29
JP2859247B2 (ja) 1999-02-17
EP0808833B1 (fr) 2004-09-22
DK0808833T3 (da) 2005-01-31
EP0808833A2 (fr) 1997-11-26
MA24251A1 (fr) 1998-04-01
TW445252B (en) 2001-07-11
HUP9700926A3 (en) 1999-05-28
YU20197A (sh) 1999-09-27
MX9703774A (es) 1998-06-30
JPH1045713A (ja) 1998-02-17
DE69730774T2 (de) 2005-09-29
CN1176072C (zh) 2004-11-17
HU9700926D0 (en) 1997-07-28

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