ZA931677B - Process for the preparation of beta-phenylisoserine and analogues thereof - Google Patents
Process for the preparation of beta-phenylisoserine and analogues thereofInfo
- Publication number
- ZA931677B ZA931677B ZA931677A ZA931677A ZA931677B ZA 931677 B ZA931677 B ZA 931677B ZA 931677 A ZA931677 A ZA 931677A ZA 931677 A ZA931677 A ZA 931677A ZA 931677 B ZA931677 B ZA 931677B
- Authority
- ZA
- South Africa
- Prior art keywords
- pct
- general formula
- phenylisoserine
- analogues
- beta
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
- C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C227/14—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof
- C07C227/18—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof by reactions involving amino or carboxyl groups, e.g. hydrolysis of esters or amides, by formation of halides, salts or esters
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C227/22—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from lactams, cyclic ketones or cyclic oximes, e.g. by reactions involving Beckmann rearrangement
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Epoxy Compounds (AREA)
- Steroid Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9202821A FR2688499B1 (fr) | 1992-03-10 | 1992-03-10 | Procede de preparation de la beta-phenylisoserine et de ses analogues. |
Publications (1)
Publication Number | Publication Date |
---|---|
ZA931677B true ZA931677B (en) | 1993-10-06 |
Family
ID=9427518
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ZA931677A ZA931677B (en) | 1992-03-10 | 1993-03-09 | Process for the preparation of beta-phenylisoserine and analogues thereof |
Country Status (25)
Country | Link |
---|---|
US (2) | US5608102A (de) |
EP (1) | EP0630365B1 (de) |
JP (1) | JP3278768B2 (de) |
KR (1) | KR100272650B1 (de) |
AT (1) | ATE159512T1 (de) |
AU (1) | AU667886B2 (de) |
CA (1) | CA2130333C (de) |
CZ (1) | CZ283613B6 (de) |
DE (1) | DE69314779T2 (de) |
DK (1) | DK0630365T3 (de) |
ES (1) | ES2109509T3 (de) |
FI (1) | FI113640B (de) |
FR (1) | FR2688499B1 (de) |
GE (1) | GEP19981430B (de) |
GR (1) | GR3025117T3 (de) |
HU (1) | HU213621B (de) |
MX (1) | MX9301268A (de) |
NO (1) | NO304515B1 (de) |
NZ (1) | NZ249899A (de) |
PL (1) | PL171551B1 (de) |
RU (1) | RU2103258C1 (de) |
SK (1) | SK281297B6 (de) |
TW (1) | TW252971B (de) |
WO (1) | WO1993017997A1 (de) |
ZA (1) | ZA931677B (de) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2195844C (en) * | 1994-07-26 | 2001-10-09 | Ezio Bombardelli | Semi-synthetic taxanes with anti-tumoural activity |
US6765015B2 (en) * | 1995-12-13 | 2004-07-20 | Xechem International, Inc. | Halogenated paclitaxel derivatives |
EP1019347B1 (de) | 1997-08-21 | 2003-03-19 | Florida State University | Verfahren zur synthese von taxanen |
EP1105118A4 (de) * | 1997-11-19 | 2003-02-26 | Xechem Inc | Halogenierte paclitaxel-derivate |
ITMI991483A1 (it) * | 1999-07-06 | 2001-01-06 | Indena Spa | Derivati tassanici e procedimenti per la loro preparazione |
CA2385528C (en) | 1999-10-01 | 2013-12-10 | Immunogen, Inc. | Compositions and methods for treating cancer using immunoconjugates and chemotherapeutic agents |
JP2002080435A (ja) * | 2000-06-26 | 2002-03-19 | Kanegafuchi Chem Ind Co Ltd | 3−アミノ−2−ヒドロキシプロピオン酸誘導体の製造法 |
JP4142444B2 (ja) | 2001-03-07 | 2008-09-03 | 第一三共株式会社 | 2−アゼチジノン誘導体の製造方法 |
EP1961735B1 (de) * | 2007-02-22 | 2009-11-18 | Indena S.P.A. | Verfahren zur Herstellung von (2r,3s)-3-Phenylisoserin-Methylester-Acetatsalz |
ES2389518T3 (es) | 2008-01-18 | 2012-10-26 | Indena S.P.A. | Formas sólidas de ortataxel |
CN102408356A (zh) * | 2011-09-28 | 2012-04-11 | 北京东方协和医药生物技术有限公司 | 一种多西他赛手性侧链中间体的制备方法 |
MX2016010095A (es) * | 2014-02-03 | 2017-02-15 | Quadriga Biosciences Inc | Beta-aminoacidos beta-sustituidos y sus analogos como agentes quimioterapeuticos. |
CN111100026A (zh) * | 2019-12-30 | 2020-05-05 | 重庆市碚圣医药科技股份有限公司 | 一种紫杉醇恶唑环侧链中间体的制备方法 |
CN112574134A (zh) * | 2020-12-30 | 2021-03-30 | 重庆市碚圣医药科技股份有限公司 | 一种多西紫杉醇侧链的合成方法 |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2629819B1 (fr) * | 1988-04-06 | 1990-11-16 | Rhone Poulenc Sante | Procede de preparation de derives de la baccatine iii et de la desacetyl-10 baccatine iii |
IT1231751B (it) * | 1989-04-12 | 1991-12-21 | Sigma Tau Ind Farmaceuti | Procedimento per la produzione di r(+) amminocarnitina e s(-) amminocarnitina |
US5175315A (en) * | 1989-05-31 | 1992-12-29 | Florida State University | Method for preparation of taxol using β-lactam |
US5304670A (en) * | 1989-08-23 | 1994-04-19 | Centre National De La Recherche Scientifique | Process for the enantioselective preparation of phenylisoserine derivatives |
FR2658510B1 (fr) * | 1990-02-21 | 1992-04-30 | Rhone Poulenc Sante | Nouveau derive de la beta-phenylisoserine, sa preparation et son emploi. |
US5294737A (en) * | 1992-02-27 | 1994-03-15 | The Research Foundation State University Of New York | Process for the production of chiral hydroxy-β-lactams and hydroxyamino acids derived therefrom |
-
1992
- 1992-03-10 FR FR9202821A patent/FR2688499B1/fr not_active Expired - Fee Related
-
1993
- 1993-03-08 AT AT93918746T patent/ATE159512T1/de active
- 1993-03-08 NZ NZ249899A patent/NZ249899A/en not_active IP Right Cessation
- 1993-03-08 DK DK93918746.4T patent/DK0630365T3/da active
- 1993-03-08 EP EP93918746A patent/EP0630365B1/de not_active Expired - Lifetime
- 1993-03-08 MX MX9301268A patent/MX9301268A/es unknown
- 1993-03-08 CA CA002130333A patent/CA2130333C/fr not_active Expired - Lifetime
- 1993-03-08 ES ES93918746T patent/ES2109509T3/es not_active Expired - Lifetime
- 1993-03-08 PL PL93305059A patent/PL171551B1/pl unknown
- 1993-03-08 US US08/295,677 patent/US5608102A/en not_active Expired - Lifetime
- 1993-03-08 HU HU9402590A patent/HU213621B/hu unknown
- 1993-03-08 GE GEAP19932472A patent/GEP19981430B/en unknown
- 1993-03-08 RU RU94045799A patent/RU2103258C1/ru active
- 1993-03-08 AU AU37557/93A patent/AU667886B2/en not_active Expired
- 1993-03-08 WO PCT/FR1993/000224 patent/WO1993017997A1/fr active IP Right Grant
- 1993-03-08 DE DE69314779T patent/DE69314779T2/de not_active Expired - Lifetime
- 1993-03-08 SK SK1085-94A patent/SK281297B6/sk not_active IP Right Cessation
- 1993-03-08 KR KR1019940703156A patent/KR100272650B1/ko not_active IP Right Cessation
- 1993-03-08 CZ CZ942185A patent/CZ283613B6/cs not_active IP Right Cessation
- 1993-03-08 JP JP51539493A patent/JP3278768B2/ja not_active Expired - Lifetime
- 1993-03-09 ZA ZA931677A patent/ZA931677B/xx unknown
- 1993-03-10 TW TW082101775A patent/TW252971B/zh not_active IP Right Cessation
-
1994
- 1994-09-05 NO NO943280A patent/NO304515B1/no not_active IP Right Cessation
- 1994-09-09 FI FI944169A patent/FI113640B/fi not_active IP Right Cessation
-
1996
- 1996-08-23 US US08/697,420 patent/US5763628A/en not_active Expired - Lifetime
-
1997
- 1997-10-23 GR GR970401615T patent/GR3025117T3/el unknown
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