ZA200603472B - Bicyclo[3.1.1]heptane substituted benzimidazolone and quinazolinone derivatives as agonists on human ORL1 receptors - Google Patents
Bicyclo[3.1.1]heptane substituted benzimidazolone and quinazolinone derivatives as agonists on human ORL1 receptors Download PDFInfo
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- ZA200603472B ZA200603472B ZA200603472A ZA200603472A ZA200603472B ZA 200603472 B ZA200603472 B ZA 200603472B ZA 200603472 A ZA200603472 A ZA 200603472A ZA 200603472 A ZA200603472 A ZA 200603472A ZA 200603472 B ZA200603472 B ZA 200603472B
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WO (1) | WO2005032547A1 (fr) |
ZA (1) | ZA200603472B (fr) |
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CN101273026A (zh) * | 2005-09-30 | 2008-09-24 | 霍夫曼-拉罗奇有限公司 | 作为mch受体拮抗剂的茚满衍生物 |
DE102007009235A1 (de) * | 2007-02-22 | 2008-09-18 | Grünenthal GmbH | Spirocyclische Cyclohexan-Derivate |
RU2488585C2 (ru) * | 2007-08-31 | 2013-07-27 | Пэдью Фарма Л.П. | Замещенные пиперидиновые соединения хиноксалинового типа и их применение |
CN102675226B (zh) * | 2012-05-24 | 2014-04-23 | 西南大学 | 3-取代-1-甲基-2,4-喹唑啉二酮类化合物及其制备方法和应用 |
CN104755465A (zh) * | 2012-08-24 | 2015-07-01 | 武田药品工业株式会社 | 杂环化合物 |
WO2014102589A1 (fr) * | 2012-12-27 | 2014-07-03 | Purdue Pharma L.P. | Composés de pipéridine du type quinazolin-4(3h)-one et utilisations de ceux-ci |
CN103420944A (zh) * | 2013-07-26 | 2013-12-04 | 江西农业大学 | 一种合成顺式氢化诺卜基甲酰胺类化合物的方法 |
GB201820165D0 (en) | 2018-12-11 | 2019-01-23 | Ucb Biopharma Sprl | Therapeutic agents |
CN115124441B (zh) * | 2022-06-30 | 2024-04-02 | 南京林业大学 | 一类诺卜酸酰肼类化合物的制备方法和产品及其应用 |
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FR2097031A1 (en) | 1970-07-29 | 1972-03-03 | Berri Balzac | 2-aminoethoxyethyl-6,6-dimethyl nor pinane derivs - local anaesthetics spasmolytics and anticholinergics |
CN1258294A (zh) | 1997-05-30 | 2000-06-28 | 万有制药株式会社 | 2-氧代咪唑衍生物 |
IL137149A0 (en) | 1998-01-19 | 2001-07-24 | Pfizer | 4-(2-keto-1-benzimidazolinyl) piperidine compounds as orl1-receptor agonists |
US6340681B1 (en) * | 1999-07-16 | 2002-01-22 | Pfizer Inc | 2-benzimidazolylamine compounds as ORL-1-receptor agonists |
DE60022226D1 (de) | 1999-12-06 | 2005-09-29 | Euro Celtique Sa | Benzimidazolverbindungen die nociceptinrezeptoraffinität haben |
US8067603B2 (en) * | 2003-09-25 | 2011-11-29 | Solvay Pharmaceuticals B.V. | Benzimidazolone and quinazolinone derivatives as agonists on human ORL1 receptors |
AR046756A1 (es) * | 2003-12-12 | 2005-12-21 | Solvay Pharm Gmbh | Derivados de hidronopol como agonistas de receptores orl-1 humanos. |
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RU2357964C2 (ru) | 2009-06-10 |
AU2004277346B2 (en) | 2009-02-19 |
SA04250319B1 (ar) | 2008-07-19 |
MXPA06002065A (es) | 2006-05-19 |
WO2005032547A1 (fr) | 2005-04-14 |
CN1838951A (zh) | 2006-09-27 |
TW200519102A (en) | 2005-06-16 |
RU2006110519A (ru) | 2006-07-27 |
AU2004277346A1 (en) | 2005-04-14 |
UA83870C2 (ru) | 2008-08-26 |
EP1670457A1 (fr) | 2006-06-21 |
JP2007507470A (ja) | 2007-03-29 |
US20050075355A1 (en) | 2005-04-07 |
BRPI0414494A (pt) | 2006-11-14 |
US7851630B2 (en) | 2010-12-14 |
AR045843A1 (es) | 2005-11-16 |
CA2534833A1 (fr) | 2005-04-14 |
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