ZA200403684B - Macrolides. - Google Patents

Macrolides.

Info

Publication number
ZA200403684B
ZA200403684B ZA200403684A ZA200403684A ZA200403684B ZA 200403684 B ZA200403684 B ZA 200403684B ZA 200403684 A ZA200403684 A ZA 200403684A ZA 200403684 A ZA200403684 A ZA 200403684A ZA 200403684 B ZA200403684 B ZA 200403684B
Authority
ZA
South Africa
Prior art keywords
macrolides
Prior art date
Application number
ZA200403684A
Other languages
English (en)
Inventor
Sulejman Alihodzic
Andrea Berdik
Stefano Biondi
Federica Damiani
Miljenko Dumic
Antun Hutinec
Sergio Luciuro
Zorica Marusic-Istuk
Alfredo Paio
Anna Quaglia
Vlado Stimac
Daniele Andreotti
Ilaria Bientinesi
Manuela Ciraco
Marko Djerek
Vesna Erakovic
Gorjana Lazarevski
Natasa Marsic
Stjepan Mutak
Drazen Pavlovic
Wolfgang Schoenfeld
Jessica Tibasco
Original Assignee
Glaxo Group Ltd
Pliva Istrazivacki Inst D O O
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd, Pliva Istrazivacki Inst D O O filed Critical Glaxo Group Ltd
Publication of ZA200403684B publication Critical patent/ZA200403684B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Steroid Compounds (AREA)
ZA200403684A 2001-11-14 2004-05-13 Macrolides. ZA200403684B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0127349.9A GB0127349D0 (en) 2001-11-14 2001-11-14 Macrolides

Publications (1)

Publication Number Publication Date
ZA200403684B true ZA200403684B (en) 2005-09-13

Family

ID=9925777

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200403684A ZA200403684B (en) 2001-11-14 2004-05-13 Macrolides.

Country Status (20)

Country Link
US (1) US7202221B2 (pt)
EP (1) EP1453846B1 (pt)
JP (1) JP2005515978A (pt)
CN (1) CN1307194C (pt)
AR (1) AR037371A1 (pt)
AT (1) ATE362479T1 (pt)
BR (1) BR0214132A (pt)
CA (1) CA2466975A1 (pt)
DE (1) DE60220180T2 (pt)
EA (1) EA007433B1 (pt)
ES (1) ES2287332T3 (pt)
GB (1) GB0127349D0 (pt)
HR (1) HRP20040433A2 (pt)
HU (1) HUP0402225A3 (pt)
IL (1) IL161710A0 (pt)
PL (1) PL371472A1 (pt)
RS (1) RS41904A (pt)
UA (1) UA77210C2 (pt)
WO (1) WO2003042228A1 (pt)
ZA (1) ZA200403684B (pt)

Families Citing this family (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6995143B2 (en) * 2002-02-28 2006-02-07 Basilea Pharmaceutica Ag Macrolides with antibacterial activity
US7135573B2 (en) 2002-05-13 2006-11-14 Enanta Pharmaceuticals, Inc. Processes for the preparation of O-(6-Pyrazol-1-yl-pyridin-3-ylmethyl)-hydroxylamine
US6764998B1 (en) 2003-06-18 2004-07-20 Enanta Pharmaceuticals, Inc. 6,11-4C-bicyclic 9a-azalide derivatives
US7910558B2 (en) 2002-05-13 2011-03-22 Enanta Pharmaceuticals, Inc. Bridged macrocyclic compounds and processes for the preparation thereof
US7022679B2 (en) 2002-05-13 2006-04-04 Enanta Pharmaceuticals, Inc. Processes for the preparation of 6-11 bicyclic erythromycin derivatives
CN1652784A (zh) * 2002-05-14 2005-08-10 加利福尼亚大学董事会 取代的喹诺酮羧酸、它们的衍生物、作用部位、以及其用途
US7091196B2 (en) 2002-09-26 2006-08-15 Rib-X Pharmaceuticals, Inc. Bifunctional heterocyclic compounds and methods of making and using same
GB0225384D0 (en) * 2002-10-31 2002-12-11 Glaxo Group Ltd Novel compounds
US6645941B1 (en) 2003-03-26 2003-11-11 Enanta Pharmaceuticals, Inc. 6,11-3C-bicyclic 9a-azalide derivatives
GB0310980D0 (en) * 2003-05-13 2003-06-18 Glaxo Group Ltd Novel compounds
GB0310979D0 (en) * 2003-05-13 2003-06-18 Glaxo Group Ltd Novel compounds
CA2525455A1 (en) * 2003-05-13 2004-11-25 Glaxo Group Limited Novel 14 and 15 membered-ring compounds
GB0310986D0 (en) * 2003-05-13 2003-06-18 Glaxo Group Ltd Novel compounds
GB0310984D0 (en) * 2003-05-13 2003-06-18 Glaxo Group Ltd Novel compounds
WO2005030227A1 (en) 2003-09-23 2005-04-07 Enanta Pharmaceuticals, Inc. 9a, 11-3C-BICYCLIC 9a-AZALIDE DERIVATIVES
WO2005070113A2 (en) 2004-01-09 2005-08-04 Enanta Pharmaceuticals, Inc. 9n-substituted 6-11 bicyclic erythromycin derivatives
EP2716647A3 (en) 2004-02-27 2014-08-20 Rib-X Pharmaceuticals, Inc. Macrocyclic compounds and methods of making and using the same
ATE439367T1 (de) * 2004-05-06 2009-08-15 Glaxosmithkline Zagreb Estergebundene makrolide, die sich für die behandlung von mikrobiellen infektionen eignen
US20080249033A1 (en) * 2004-05-06 2008-10-09 Sulejman Alihodzic Carbamate Linked Macrolides Useful For The Treatment Of Microbial Infections
WO2006047167A2 (en) * 2004-10-21 2006-05-04 Janssen Pharmaceutica, N.V. 9 alkyl and 9 alkylidenyl 6-0 alkyl-11, 12 carbamate ketolide antimicrobials
GB0424958D0 (en) * 2004-11-11 2004-12-15 Glaxo Group Ltd Novel compounds
GB0424951D0 (en) * 2004-11-11 2004-12-15 Glaxo Group Ltd Novel compounds
GB0424961D0 (en) * 2004-11-11 2004-12-15 Glaxo Group Ltd Novel compounds
GB0424959D0 (en) * 2004-11-11 2004-12-15 Glaxo Group Ltd Novel compounds
ES2428874T3 (es) * 2006-08-09 2013-11-12 Basilea Pharmaceutica Ag Nuevos macrólidos útiles contra las enfermedades inflamatorias y alérgicas
EP2056844A4 (en) 2006-08-24 2010-11-24 Wockhardt Research Center NEW MACROLIDS AND KETOLIDS WITH ANTIMICROBIAL EFFECT
US8410065B2 (en) 2008-02-08 2013-04-02 Basilea Pharmaceutica Ag Macrolides and their use
CA2763246C (en) 2009-05-27 2013-10-29 Wockhardt Research Centre Ketolide compounds having antimicrobial activity
CA2820451C (en) 2010-12-09 2017-12-12 Wockhardt Limited Ketolide compounds
JPWO2012105562A1 (ja) * 2011-01-31 2014-07-03 Meiji Seikaファルマ株式会社 新規マクロライド誘導体
CN103619849B (zh) 2011-03-01 2016-05-25 沃克哈特有限公司 酮内酯中间体的制备方法

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0126344A2 (en) 1983-05-20 1984-11-28 Abbott Laboratories Tripeptide esters of therapeutic agents
US4742049A (en) * 1986-06-04 1988-05-03 Abbott Laboratories Semisynthetic erythromycin antibiotics
JPH04504259A (ja) 1989-03-28 1992-07-30 アボツト・ラボラトリーズ エリスロマイシン誘導体
CA2064634C (en) * 1991-04-04 1998-08-04 James V. Heck 9-deoxo-8a-aza-8a-homoerythromycin a derivatives modified at the 4"- and8a-positions
IL126625A0 (en) 1996-05-07 1999-08-17 Abbott Lab 6-o-substituted erythromycin compounds and method for making same
EP0895999A1 (en) * 1997-08-06 1999-02-10 Pfizer Products Inc. C-4" substituted macrolide antibiotics
US6262030B1 (en) * 1998-11-03 2001-07-17 Pfizer Inc. Erythromycin derivatives
AP2001002302A0 (en) 1999-05-24 2001-10-25 Pfizer Prod Inc 13-Methyl erythromycin derivatives.
EP1206476B1 (en) 1999-08-24 2006-01-04 Abbott Laboratories 9a-azalides with antibacterial activity
US6946446B2 (en) * 2000-02-24 2005-09-20 Abbott Laboratories Anti-infective agents useful against multidrug-resistant strains of bacteria
DK1259923T3 (da) 2000-02-24 2006-05-01 Abbott Lab Antiinfektionsmiddel, der er anvendeligt mod multilægemiddelresistente bakteriestammer
JP2002173498A (ja) 2000-09-27 2002-06-21 Hokuriku Seiyaku Co Ltd エリスロマイシン誘導体
GB0025688D0 (en) * 2000-10-19 2000-12-06 Glaxo Group Ltd Macrolides

Also Published As

Publication number Publication date
HUP0402225A2 (hu) 2005-02-28
CN1612888A (zh) 2005-05-04
AR037371A1 (es) 2004-11-03
BR0214132A (pt) 2004-09-14
CA2466975A1 (en) 2003-05-22
RS41904A (en) 2006-10-27
DE60220180T2 (de) 2008-01-17
EP1453846A1 (en) 2004-09-08
CN1307194C (zh) 2007-03-28
UA77210C2 (en) 2006-11-15
US20050080025A1 (en) 2005-04-14
DE60220180D1 (de) 2007-06-28
WO2003042228A1 (en) 2003-05-22
EA007433B1 (ru) 2006-10-27
GB0127349D0 (en) 2002-01-02
ATE362479T1 (de) 2007-06-15
US7202221B2 (en) 2007-04-10
JP2005515978A (ja) 2005-06-02
HUP0402225A3 (en) 2006-01-30
ES2287332T3 (es) 2007-12-16
IL161710A0 (en) 2004-09-27
EA200400536A1 (ru) 2004-12-30
PL371472A1 (en) 2005-06-13
HRP20040433A2 (en) 2005-04-30
EP1453846B1 (en) 2007-05-16

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