ZA200302191B - Alpha-aryl ethanolamines and their use as beta-3 adrenergic receptor agonists. - Google Patents

Alpha-aryl ethanolamines and their use as beta-3 adrenergic receptor agonists. Download PDF

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Publication number
ZA200302191B
ZA200302191B ZA200302191A ZA200302191A ZA200302191B ZA 200302191 B ZA200302191 B ZA 200302191B ZA 200302191 A ZA200302191 A ZA 200302191A ZA 200302191 A ZA200302191 A ZA 200302191A ZA 200302191 B ZA200302191 B ZA 200302191B
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South Africa
Prior art keywords
phenoxy
pyridin
ethylamino
thiazol
ethylamine
Prior art date
Application number
ZA200302191A
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English (en)
Inventor
Day Robert Francis
Lafontaine Jennifer Anne
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Pfizer Prod Inc
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Publication of ZA200302191B publication Critical patent/ZA200302191B/en

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    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
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    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
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    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
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    • C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D263/32—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
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    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
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ZA200302191A 2000-10-20 2003-03-19 Alpha-aryl ethanolamines and their use as beta-3 adrenergic receptor agonists. ZA200302191B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US24227400P 2000-10-20 2000-10-20

Publications (1)

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ZA200302191B true ZA200302191B (en) 2004-08-27

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ZA200302191A ZA200302191B (en) 2000-10-20 2003-03-19 Alpha-aryl ethanolamines and their use as beta-3 adrenergic receptor agonists.

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US (2) US6566377B2 (sk)
EP (1) EP1326861A1 (sk)
JP (1) JP2004511555A (sk)
KR (1) KR20030044013A (sk)
CN (1) CN1469876A (sk)
AP (1) AP2001002307A0 (sk)
AR (1) AR035716A1 (sk)
AU (1) AU2001292161A1 (sk)
BG (1) BG107652A (sk)
BR (1) BR0114836A (sk)
CA (1) CA2423792A1 (sk)
CR (1) CR6935A (sk)
CZ (1) CZ20031012A3 (sk)
DO (1) DOP2001000270A (sk)
EA (1) EA200300305A1 (sk)
EC (1) ECSP034562A (sk)
EE (1) EE200300191A (sk)
GT (1) GT200100210A (sk)
HR (1) HRP20030297A2 (sk)
HU (1) HUP0301382A2 (sk)
IL (1) IL154911A0 (sk)
IS (1) IS6748A (sk)
MA (1) MA26954A1 (sk)
MX (1) MXPA03003455A (sk)
NO (1) NO20031573L (sk)
PA (1) PA8530401A1 (sk)
PE (1) PE20020541A1 (sk)
PL (1) PL362076A1 (sk)
SK (1) SK4612003A3 (sk)
SV (1) SV2003000697A (sk)
TN (1) TNSN01148A1 (sk)
UY (1) UY26974A1 (sk)
WO (1) WO2002032897A1 (sk)
ZA (1) ZA200302191B (sk)

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