ZA200204663B - Substituted norbornylamino derivatives, method for the production thereof, use thereof as a medicament or a dignostic reagent and medicaments containing said compounds. - Google Patents

Substituted norbornylamino derivatives, method for the production thereof, use thereof as a medicament or a dignostic reagent and medicaments containing said compounds. Download PDF

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Publication number
ZA200204663B
ZA200204663B ZA200204663A ZA200204663A ZA200204663B ZA 200204663 B ZA200204663 B ZA 200204663B ZA 200204663 A ZA200204663 A ZA 200204663A ZA 200204663 A ZA200204663 A ZA 200204663A ZA 200204663 B ZA200204663 B ZA 200204663B
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Prior art keywords
exo
methanoinden
endo
amine
alkyl
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ZA200204663A
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English (en)
Inventor
Uwe Heinelt
Hans-Jochen Lang
Heinz-Werner Kleemann
Jan-Robert Schwark
Klaus With
Hans-Willi Jansen
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Aventis Pharma Gmbh
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Publication of ZA200204663B publication Critical patent/ZA200204663B/en

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    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/26—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
    • C07C317/32—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
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    • C07C211/34—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of a saturated carbon skeleton
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    • C07C211/43—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C07C211/44—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to only one six-membered aromatic ring
    • C07C211/49—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to only one six-membered aromatic ring having at least two amino groups bound to the carbon skeleton
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    • C07C215/02—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C215/22—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated
    • C07C215/28—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings
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    • C07C217/56—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups bound to carbon atoms of at least one six-membered aromatic ring and amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups linked to the six-membered aromatic ring, or to the condensed ring system containing that ring, by carbon chains not further substituted by singly-bound oxygen atoms
    • C07C217/58—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups bound to carbon atoms of at least one six-membered aromatic ring and amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups linked to the six-membered aromatic ring, or to the condensed ring system containing that ring, by carbon chains not further substituted by singly-bound oxygen atoms with amino groups and the six-membered aromatic ring, or the condensed ring system containing that ring, bound to the same carbon atom of the carbon chain
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    • C07C217/56—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups bound to carbon atoms of at least one six-membered aromatic ring and amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups linked to the six-membered aromatic ring, or to the condensed ring system containing that ring, by carbon chains not further substituted by singly-bound oxygen atoms
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    • C07C257/10—Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. amidines
    • C07C257/18—Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. amidines having carbon atoms of amidino groups bound to carbon atoms of six-membered aromatic rings
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    • C07C323/31—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton
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ZA200204663A 1999-12-14 2002-06-11 Substituted norbornylamino derivatives, method for the production thereof, use thereof as a medicament or a dignostic reagent and medicaments containing said compounds. ZA200204663B (en)

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Application Number Priority Date Filing Date Title
DE19960204A DE19960204A1 (de) 1999-12-14 1999-12-14 Substituierte Norlbornylamino-Derivate, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament

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ZA200204663B true ZA200204663B (en) 2003-09-29

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ZA200204663A ZA200204663B (en) 1999-12-14 2002-06-11 Substituted norbornylamino derivatives, method for the production thereof, use thereof as a medicament or a dignostic reagent and medicaments containing said compounds.

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PL356235A1 (en) 2004-06-28
BR0016360A (pt) 2002-10-01
AU1525401A (en) 2001-06-25
CN1210251C (zh) 2005-07-13
HK1049655B (zh) 2005-10-14
IL150228A0 (en) 2002-12-01
ATE338022T1 (de) 2006-09-15
NZ519511A (en) 2004-08-27
WO2001044164A1 (de) 2001-06-21
US6825231B2 (en) 2004-11-30
HUP0204360A2 (en) 2003-05-28
HK1049655A1 (en) 2003-05-23
RU2002118700A (ru) 2004-01-20
SK8202002A3 (en) 2002-10-08
NO20022801D0 (no) 2002-06-12
EE200200292A (et) 2003-08-15
CA2394130A1 (en) 2001-06-21
EP1255724B1 (de) 2006-08-30
CN1379756A (zh) 2002-11-13
RU2260584C2 (ru) 2005-09-20
JP2003517033A (ja) 2003-05-20
HUP0204360A3 (en) 2005-04-28
HRP20020517A2 (en) 2004-08-31
KR20030004308A (ko) 2003-01-14
AR032434A1 (es) 2003-11-12
YU30302A (sh) 2005-06-10
CZ20022006A3 (cs) 2002-09-11
EP1255724A1 (de) 2002-11-13
NO20022801L (no) 2002-08-09
US20010023257A1 (en) 2001-09-20
MXPA02003763A (es) 2002-09-30
AU778888B2 (en) 2004-12-23
DE50013410D1 (de) 2006-10-12

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