ZA200108176B - N-(2-Phenyl-4-amino-butyl)-1-naphthamides as neurokinin-1 receptor antagonists. - Google Patents
N-(2-Phenyl-4-amino-butyl)-1-naphthamides as neurokinin-1 receptor antagonists. Download PDFInfo
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- ZA200108176B ZA200108176B ZA200108176A ZA200108176A ZA200108176B ZA 200108176 B ZA200108176 B ZA 200108176B ZA 200108176 A ZA200108176 A ZA 200108176A ZA 200108176 A ZA200108176 A ZA 200108176A ZA 200108176 B ZA200108176 B ZA 200108176B
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- compound
- compound according
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Classifications
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Landscapes
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- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Pulmonology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Rheumatology (AREA)
- Immunology (AREA)
- Hospice & Palliative Care (AREA)
- Otolaryngology (AREA)
- Psychology (AREA)
- Cardiology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Dermatology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9907571.5A GB9907571D0 (en) | 1999-04-06 | 1999-04-06 | Compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200108176B true ZA200108176B (en) | 2003-01-06 |
Family
ID=10850835
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200108176A ZA200108176B (en) | 1999-04-06 | 2001-10-04 | N-(2-Phenyl-4-amino-butyl)-1-naphthamides as neurokinin-1 receptor antagonists. |
Country Status (25)
| Country | Link |
|---|---|
| US (3) | US6476077B1 (zh) |
| EP (1) | EP1169302B1 (zh) |
| JP (1) | JP2002541137A (zh) |
| KR (1) | KR20010102580A (zh) |
| CN (2) | CN1534017A (zh) |
| AT (1) | ATE277893T1 (zh) |
| AU (1) | AU3569200A (zh) |
| BG (1) | BG106074A (zh) |
| BR (1) | BR0009582A (zh) |
| CA (1) | CA2368240A1 (zh) |
| CZ (1) | CZ20013574A3 (zh) |
| DE (1) | DE60014343T2 (zh) |
| EE (1) | EE200100520A (zh) |
| GB (1) | GB9907571D0 (zh) |
| HK (1) | HK1044145A1 (zh) |
| HU (1) | HUP0200707A3 (zh) |
| IL (1) | IL145645A0 (zh) |
| IS (1) | IS6087A (zh) |
| NO (1) | NO20014855L (zh) |
| PL (1) | PL350568A1 (zh) |
| SK (1) | SK13012001A3 (zh) |
| TR (1) | TR200102875T2 (zh) |
| UA (1) | UA67839C2 (zh) |
| WO (1) | WO2000059873A1 (zh) |
| ZA (1) | ZA200108176B (zh) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9907571D0 (en) * | 1999-04-06 | 1999-05-26 | Zeneca Ltd | Compounds |
| GB0019008D0 (en) * | 2000-08-04 | 2000-09-27 | Astrazeneca Ab | Therapeutic compounds |
| SE0201938D0 (sv) * | 2002-06-20 | 2002-06-20 | Astrazeneca Ab | New process |
| ES2299734T3 (es) * | 2002-11-05 | 2008-06-01 | Astrazeneca Ab | Disposicion de bloqueo para una tapa de un recipiente y recipiente correspondiente. |
| ES2286470T3 (es) * | 2002-12-20 | 2007-12-01 | Astrazeneca Ab | Compuestos de 4-aril-4-(naft-1-ilmetilamino)metil-piperidina y su uso. |
| US20080045610A1 (en) * | 2004-09-23 | 2008-02-21 | Alexander Michalow | Methods for regulating neurotransmitter systems by inducing counteradaptations |
| US20060069086A1 (en) * | 2004-09-23 | 2006-03-30 | Alexander Michalow | Methods for regulating neurotransmitter systems by inducing counteradaptations |
| NO2729147T3 (zh) | 2011-07-04 | 2018-02-03 | ||
| RU2743206C2 (ru) | 2015-05-18 | 2021-02-16 | Кэнди Терапьютикс Лимитед | Двойные антагонисты рецептора нейрокинин-1/нейрокинин-3 для лечения заболеваний, зависимых от половых гормонов |
| JP2021514976A (ja) | 2018-02-26 | 2021-06-17 | オスペダーレ・サン・ラッファエーレ・エッセエッレエッレ | 眼痛の治療における使用のためのｎｋ−１拮抗薬 |
| MX2020009438A (es) | 2018-03-14 | 2022-05-11 | Kandy Therapeutics Ltd | Formulacion farmaceutica novedosa que comprende antagonistas del receptor dual nk-1/nk-3. |
| RU2697414C1 (ru) | 2018-05-11 | 2019-08-14 | Общество с ограниченной ответственностью "АЙ БИ ДИ Терапевтикс" | Новый антагонист тахикининовых рецепторов и его применение |
| EP4117673A1 (en) | 2020-03-11 | 2023-01-18 | Ospedale San Raffaele S.r.l. | Treatment of stem cell deficiency |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FI97540C (fi) | 1989-11-06 | 1997-01-10 | Sanofi Sa | Menetelmä terapeuttisesti käyttökelpoisten, aromaattisesti substituoitujen piperidiini- ja piperatsiinijohdannaisten valmistamiseksi |
| EP0702681A1 (en) | 1993-06-07 | 1996-03-27 | Merck & Co. Inc. | Spiro-substituted azacycles as neurokinin antagonists |
| PT777659E (pt) * | 1994-08-15 | 2001-09-28 | Merck Sharp & Dohme | Derivados de morfolina e sua utilizacao como agentes terapeuticos |
| AU5522498A (en) * | 1996-12-13 | 1998-07-03 | Merck & Co., Inc. | Substituted aryl piperazines as modulators of chemokine receptor activity |
| GB9907571D0 (en) * | 1999-04-06 | 1999-05-26 | Zeneca Ltd | Compounds |
| HUP0400252A3 (en) * | 2001-03-21 | 2011-09-28 | Pharmacopeia Drug Discovery | Aryl and biaryl compounds having mch modulatory activity, pharmaceutical compositions containing them and process for producing them |
-
1999
- 1999-04-06 GB GBGB9907571.5A patent/GB9907571D0/en not_active Ceased
-
2000
- 2000-03-04 UA UA2001117535A patent/UA67839C2/uk unknown
- 2000-04-03 CA CA002368240A patent/CA2368240A1/en not_active Abandoned
- 2000-04-03 IL IL14564500A patent/IL145645A0/xx unknown
- 2000-04-03 PL PL00350568A patent/PL350568A1/xx unknown
- 2000-04-03 WO PCT/GB2000/001252 patent/WO2000059873A1/en not_active Application Discontinuation
- 2000-04-03 JP JP2000609386A patent/JP2002541137A/ja active Pending
- 2000-04-03 DE DE60014343T patent/DE60014343T2/de not_active Expired - Fee Related
- 2000-04-03 CZ CZ20013574A patent/CZ20013574A3/cs unknown
- 2000-04-03 US US09/937,981 patent/US6476077B1/en not_active Expired - Fee Related
- 2000-04-03 EP EP00914298A patent/EP1169302B1/en not_active Expired - Lifetime
- 2000-04-03 CN CNA2004100053467A patent/CN1534017A/zh active Pending
- 2000-04-03 TR TR2001/02875T patent/TR200102875T2/xx unknown
- 2000-04-03 AT AT00914298T patent/ATE277893T1/de not_active IP Right Cessation
- 2000-04-03 AU AU35692/00A patent/AU3569200A/en not_active Abandoned
- 2000-04-03 HU HU0200707A patent/HUP0200707A3/hu unknown
- 2000-04-03 SK SK1301-2001A patent/SK13012001A3/sk unknown
- 2000-04-03 KR KR1020017012692A patent/KR20010102580A/ko not_active Application Discontinuation
- 2000-04-03 EE EEP200100520A patent/EE200100520A/xx unknown
- 2000-04-03 CN CN00805623A patent/CN1345307A/zh active Pending
- 2000-04-03 BR BR0009582-6A patent/BR0009582A/pt not_active IP Right Cessation
-
2001
- 2001-09-26 IS IS6087A patent/IS6087A/is unknown
- 2001-10-04 ZA ZA200108176A patent/ZA200108176B/en unknown
- 2001-10-05 NO NO20014855A patent/NO20014855L/no not_active Application Discontinuation
- 2001-11-01 BG BG106074A patent/BG106074A/xx unknown
-
2002
- 2002-06-26 HK HK02104758.2A patent/HK1044145A1/zh unknown
- 2002-11-01 US US10/286,624 patent/US6586432B2/en not_active Expired - Fee Related
-
2003
- 2003-06-30 US US10/611,052 patent/US6821973B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| CZ20013574A3 (cs) | 2002-05-15 |
| HUP0200707A2 (en) | 2002-06-29 |
| GB9907571D0 (en) | 1999-05-26 |
| DE60014343D1 (de) | 2004-11-04 |
| EP1169302B1 (en) | 2004-09-29 |
| CN1534017A (zh) | 2004-10-06 |
| DE60014343T2 (de) | 2006-03-02 |
| US20030092713A1 (en) | 2003-05-15 |
| CN1345307A (zh) | 2002-04-17 |
| CA2368240A1 (en) | 2000-10-12 |
| BR0009582A (pt) | 2001-12-26 |
| US6821973B2 (en) | 2004-11-23 |
| IL145645A0 (en) | 2002-06-30 |
| HK1044145A1 (zh) | 2002-10-11 |
| NO20014855L (no) | 2001-12-06 |
| EP1169302A1 (en) | 2002-01-09 |
| IS6087A (is) | 2001-09-26 |
| JP2002541137A (ja) | 2002-12-03 |
| TR200102875T2 (tr) | 2002-01-21 |
| US6586432B2 (en) | 2003-07-01 |
| US20040106610A1 (en) | 2004-06-03 |
| UA67839C2 (uk) | 2004-07-15 |
| PL350568A1 (en) | 2002-12-16 |
| HUP0200707A3 (en) | 2002-11-28 |
| WO2000059873A1 (en) | 2000-10-12 |
| ATE277893T1 (de) | 2004-10-15 |
| KR20010102580A (ko) | 2001-11-15 |
| NO20014855D0 (no) | 2001-10-05 |
| SK13012001A3 (sk) | 2002-04-04 |
| BG106074A (en) | 2002-05-31 |
| US6476077B1 (en) | 2002-11-05 |
| EE200100520A (et) | 2002-12-16 |
| AU3569200A (en) | 2000-10-23 |
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