ZA200102157B - Serotonergic 5HT2 agonists for treating glaucoma. - Google Patents
Serotonergic 5HT2 agonists for treating glaucoma. Download PDFInfo
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- ZA200102157B ZA200102157B ZA200102157A ZA200102157A ZA200102157B ZA 200102157 B ZA200102157 B ZA 200102157B ZA 200102157 A ZA200102157 A ZA 200102157A ZA 200102157 A ZA200102157 A ZA 200102157A ZA 200102157 B ZA200102157 B ZA 200102157B
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
- A61K31/4045—Indole-alkylamines; Amides thereof, e.g. serotonin, melatonin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Ophthalmology & Optometry (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US10106798P | 1998-09-18 | 1998-09-18 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200102157B true ZA200102157B (en) | 2003-03-05 |
Family
ID=22282920
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200102157A ZA200102157B (en) | 1998-09-18 | 2001-03-15 | Serotonergic 5HT2 agonists for treating glaucoma. |
Country Status (18)
| Country | Link |
|---|---|
| US (2) | US6664286B1 (fr) |
| EP (1) | EP1112106B1 (fr) |
| JP (1) | JP2002526443A (fr) |
| KR (1) | KR20010073153A (fr) |
| CN (1) | CN1269484C (fr) |
| AR (1) | AR020442A1 (fr) |
| AT (1) | ATE310566T1 (fr) |
| AU (1) | AU755119B2 (fr) |
| BR (1) | BR9913800A (fr) |
| CA (1) | CA2344150A1 (fr) |
| DE (1) | DE69928542T2 (fr) |
| DK (1) | DK1112106T3 (fr) |
| ES (1) | ES2252978T3 (fr) |
| HK (1) | HK1038516A1 (fr) |
| TR (1) | TR200100754T2 (fr) |
| TW (1) | TWI229602B (fr) |
| WO (1) | WO2000016761A2 (fr) |
| ZA (1) | ZA200102157B (fr) |
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| TW593302B (en) * | 2001-12-20 | 2004-06-21 | Alcon Inc | Novel benzodifuranimidazoline and benzofuranimidazoline derivatives and their use for the treatment of glaucoma |
| PL375564A1 (en) * | 2002-08-30 | 2005-11-28 | Alcon, Inc. | Substituted 5-chroman-5-yl-ethylamine compounds and their use for the treatment of glaucoma |
| EP1558238A4 (fr) * | 2002-09-24 | 2006-08-30 | Univ Virginia Commonwealth | Beta-hydroxyphenylaldylamines et utilisation de celles-ci pour traiter le glaucome |
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| US7476687B2 (en) * | 2003-11-26 | 2009-01-13 | Alcon, Inc. | Substituted furo[2,3-g]indazoles for the treatment of glaucoma |
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| US7338972B1 (en) | 2003-12-15 | 2008-03-04 | Alcon, Inc. | Substituted 1-alkylamino-1H-indazoles for the treatment of glaucoma |
| EP1744784A2 (fr) * | 2004-05-11 | 2007-01-24 | Becton, Dickinson and Company | Formulations de substances analgesiques et leurs methodes d'administration |
| EP2248524A3 (fr) | 2004-08-25 | 2011-03-09 | Takeda Pharmaceutical Company Limited | Agents preventifs/remedes pour l'incontinence de stress et procede de selecetion de ceux-ci |
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| TW200744567A (en) * | 2005-09-23 | 2007-12-16 | Alcon Inc | Phenylethylamine analogs and their use for treating glaucoma |
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| EP2789338A3 (fr) | 2007-11-15 | 2015-01-14 | Takeda Pharmaceutical Company Limited | Dérivé de pyridine condensé et son utilisation |
| US9642819B2 (en) * | 2008-07-10 | 2017-05-09 | Board Of Supervisors Of Louisiana State University And Agricultural And Mechanical | Low dosage serotonin 5-HT2A receptor agonist to suppress inflammation |
| US8299079B2 (en) | 2009-05-22 | 2012-10-30 | Kaufman Herbert E | Preparations and methods for ameliorating or reducing presbyopia |
| EP2510949A4 (fr) | 2009-12-11 | 2013-11-13 | Astellas Pharma Inc | Agent thérapeutique pour la fibromyalgie |
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| GB2571696B (en) | 2017-10-09 | 2020-05-27 | Compass Pathways Ltd | Large scale method for the preparation of Psilocybin and formulations of Psilocybin so produced |
| JPWO2019131902A1 (ja) | 2017-12-27 | 2020-12-10 | 武田薬品工業株式会社 | 腹圧性尿失禁および便失禁の治療薬 |
| CN113993523A (zh) | 2019-04-17 | 2022-01-28 | 指南针探路者有限公司 | 用赛洛西宾治疗抑郁症和其他各种病症 |
| WO2024010765A1 (fr) * | 2022-07-05 | 2024-01-11 | Board Of Supervisors Of Louisiana State University And Agricultural And Mechanical College | Compositions de traitement d'états sensibles à 5-ht2 et leurs procédés d'utilisation |
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-
1999
- 1999-09-03 JP JP2000573722A patent/JP2002526443A/ja active Pending
- 1999-09-03 WO PCT/US1999/019888 patent/WO2000016761A2/fr not_active Application Discontinuation
- 1999-09-03 CN CNB99810891XA patent/CN1269484C/zh not_active Expired - Fee Related
- 1999-09-03 KR KR1020017003191A patent/KR20010073153A/ko not_active Application Discontinuation
- 1999-09-03 ES ES99948085T patent/ES2252978T3/es not_active Expired - Lifetime
- 1999-09-03 DK DK99948085T patent/DK1112106T3/da active
- 1999-09-03 US US09/787,332 patent/US6664286B1/en not_active Expired - Lifetime
- 1999-09-03 TR TR2001/00754T patent/TR200100754T2/xx unknown
- 1999-09-03 AU AU61326/99A patent/AU755119B2/en not_active Ceased
- 1999-09-03 BR BR9913800-0A patent/BR9913800A/pt not_active Application Discontinuation
- 1999-09-03 DE DE69928542T patent/DE69928542T2/de not_active Expired - Fee Related
- 1999-09-03 CA CA002344150A patent/CA2344150A1/fr not_active Abandoned
- 1999-09-03 EP EP99948085A patent/EP1112106B1/fr not_active Expired - Lifetime
- 1999-09-03 AT AT99948085T patent/ATE310566T1/de not_active IP Right Cessation
- 1999-09-14 AR ARP990104608A patent/AR020442A1/es unknown
- 1999-09-17 TW TW088116092A patent/TWI229602B/zh not_active IP Right Cessation
-
2001
- 2001-03-15 ZA ZA200102157A patent/ZA200102157B/en unknown
- 2001-12-15 HK HK01108810A patent/HK1038516A1/xx not_active IP Right Cessation
-
2003
- 2003-05-09 US US10/434,708 patent/US20030203912A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US20030203912A1 (en) | 2003-10-30 |
| JP2002526443A (ja) | 2002-08-20 |
| EP1112106B1 (fr) | 2005-11-23 |
| CN1269484C (zh) | 2006-08-16 |
| BR9913800A (pt) | 2001-05-29 |
| AR020442A1 (es) | 2002-05-15 |
| TR200100754T2 (tr) | 2001-10-22 |
| WO2000016761A2 (fr) | 2000-03-30 |
| AU6132699A (en) | 2000-04-10 |
| WO2000016761A3 (fr) | 2000-05-25 |
| EP1112106A2 (fr) | 2001-07-04 |
| DK1112106T3 (da) | 2005-12-12 |
| CA2344150A1 (fr) | 2000-03-30 |
| AU755119B2 (en) | 2002-12-05 |
| KR20010073153A (ko) | 2001-07-31 |
| DE69928542T2 (de) | 2006-03-30 |
| CN1317979A (zh) | 2001-10-17 |
| HK1038516A1 (en) | 2002-03-22 |
| DE69928542D1 (de) | 2005-12-29 |
| ATE310566T1 (de) | 2005-12-15 |
| US6664286B1 (en) | 2003-12-16 |
| TWI229602B (en) | 2005-03-21 |
| ES2252978T3 (es) | 2006-05-16 |
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