WO2012174685A1 - Procédé de préparation d'un dérivé de 2h-1,2,3-triazole 2-substitué - Google Patents

Procédé de préparation d'un dérivé de 2h-1,2,3-triazole 2-substitué Download PDF

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Publication number
WO2012174685A1
WO2012174685A1 PCT/CN2011/001101 CN2011001101W WO2012174685A1 WO 2012174685 A1 WO2012174685 A1 WO 2012174685A1 CN 2011001101 W CN2011001101 W CN 2011001101W WO 2012174685 A1 WO2012174685 A1 WO 2012174685A1
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WO
WIPO (PCT)
Prior art keywords
formula
compound
substituted
triazole
group
Prior art date
Application number
PCT/CN2011/001101
Other languages
English (en)
Chinese (zh)
Inventor
江岳恒
阙利民
蔡彤�
林志刚
Original Assignee
苏州雅本化学股份有限公司
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 苏州雅本化学股份有限公司 filed Critical 苏州雅本化学股份有限公司
Publication of WO2012174685A1 publication Critical patent/WO2012174685A1/fr

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/04—1,2,3-Triazoles; Hydrogenated 1,2,3-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/04—1,2,3-Triazoles; Hydrogenated 1,2,3-triazoles
    • C07D249/06—1,2,3-Triazoles; Hydrogenated 1,2,3-triazoles with aryl radicals directly attached to ring atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Abstract

Procédé de préparation d'un dérivé de 2h-1,2,3-triazole 2-substitué (Formule I).
PCT/CN2011/001101 2011-06-20 2011-07-04 Procédé de préparation d'un dérivé de 2h-1,2,3-triazole 2-substitué WO2012174685A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CN201110166067.9A CN102408385B (zh) 2011-06-20 2011-06-20 一种2-取代-2h-1,2,3-三氮唑衍生物的制备方法
CN201110166067.9 2011-06-20

Publications (1)

Publication Number Publication Date
WO2012174685A1 true WO2012174685A1 (fr) 2012-12-27

Family

ID=45910775

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/CN2011/001101 WO2012174685A1 (fr) 2011-06-20 2011-07-04 Procédé de préparation d'un dérivé de 2h-1,2,3-triazole 2-substitué

Country Status (2)

Country Link
CN (1) CN102408385B (fr)
WO (1) WO2012174685A1 (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102786485B (zh) * 2012-08-24 2014-11-26 雅本化学股份有限公司 2-取代-2h-1,2,3-三氮唑衍生物及其制备方法
CN103058940B (zh) * 2012-12-14 2015-12-23 雅本化学股份有限公司 1-取代-4-溴-2h-1,2,3-三氮唑衍生物及其制备方法
CN103073513B (zh) * 2012-12-14 2015-12-02 雅本化学股份有限公司 1-取代-5-氯-2h-1,2,3-三氮唑-4-羧酸衍生物及其制备方法
AU2019261274B2 (en) * 2018-04-23 2021-10-28 Corcept Therapeutics, Inc. Methods of preparing regioselective N-alkyl triazoles

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1289326A (zh) * 1998-02-27 2001-03-28 辉瑞产品公司 用于治疗局部缺血的n－[(取代的五元二氮杂或三氮杂二不饱和环)羰基]胍衍生物
CN101389625A (zh) * 2006-02-27 2009-03-18 先正达有限公司 具有除草作用的异唑啉化合物
CN101687860A (zh) * 2007-04-23 2010-03-31 阿斯利康(瑞典)有限公司 用于治疗疼痛的新颖n-（8-杂芳基四氢萘-2-基）或n-（5-杂芳基色满-3-基）甲酰胺衍生物

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1289326A (zh) * 1998-02-27 2001-03-28 辉瑞产品公司 用于治疗局部缺血的n－[(取代的五元二氮杂或三氮杂二不饱和环)羰基]胍衍生物
CN101389625A (zh) * 2006-02-27 2009-03-18 先正达有限公司 具有除草作用的异唑啉化合物
CN101687860A (zh) * 2007-04-23 2010-03-31 阿斯利康(瑞典)有限公司 用于治疗疼痛的新颖n-（8-杂芳基四氢萘-2-基）或n-（5-杂芳基色满-3-基）甲酰胺衍生物

Also Published As

Publication number Publication date
CN102408385A (zh) 2012-04-11
CN102408385B (zh) 2014-06-18

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