UY28873A1 - Nuevos compuestos de morfina composiciones y procedimientos de preparación - Google Patents

Nuevos compuestos de morfina composiciones y procedimientos de preparación

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Publication number
UY28873A1
UY28873A1 UY28873A UY28873A UY28873A1 UY 28873 A1 UY28873 A1 UY 28873A1 UY 28873 A UY28873 A UY 28873A UY 28873 A UY28873 A UY 28873A UY 28873 A1 UY28873 A1 UY 28873A1
Authority
UY
Uruguay
Prior art keywords
morfina
new
preparation procedures
compounds compositions
compounds
Prior art date
Application number
UY28873A
Other languages
English (en)
Inventor
Paul Vincent Fish
Alan Stobie
Florian Wakenhut
Gavin Alistair Whitlock
Malcolm Christian Mackenny
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=32482498&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY28873(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of UY28873A1 publication Critical patent/UY28873A1/es

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    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
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    • C07D265/281,4-Oxazines; Hydrogenated 1,4-oxazines
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    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Diabetes (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Obesity (AREA)
  • Ophthalmology & Optometry (AREA)
  • Gynecology & Obstetrics (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Dermatology (AREA)
  • Vascular Medicine (AREA)

Abstract

La presente invención proporciona compuestos de Fórmula I: en la que R1, R2, R3, y n tienen cualquiera de los valores definidos en la memoria descriptiva, y sales farmacéuticamente aceptables de los mismos, que son útiles como agentes en el tratamiento de afecciones que incluyen trastornos urinarios, dolor, eyaculación precoz, ADHD y fibromialgia. También se proporcionan composiciones farmacéuticas que comprenden uno o más compuestos de Fórmula I.
UY28873A 2004-04-30 2005-04-27 Nuevos compuestos de morfina composiciones y procedimientos de preparación UY28873A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0409744.0A GB0409744D0 (en) 2004-04-30 2004-04-30 Novel compounds

Publications (1)

Publication Number Publication Date
UY28873A1 true UY28873A1 (es) 2005-11-30

Family

ID=32482498

Family Applications (1)

Application Number Title Priority Date Filing Date
UY28873A UY28873A1 (es) 2004-04-30 2005-04-27 Nuevos compuestos de morfina composiciones y procedimientos de preparación

Country Status (33)

Country Link
US (3) US20050250775A1 (es)
EP (1) EP1744754A1 (es)
JP (2) JP4181622B2 (es)
KR (4) KR20090006887A (es)
CN (1) CN1950089A (es)
AP (1) AP2006003767A0 (es)
AR (1) AR048934A1 (es)
AU (1) AU2005237301A1 (es)
BR (1) BRPI0510515A (es)
CA (1) CA2564990C (es)
CR (1) CR8717A (es)
DO (1) DOP2005000064A (es)
EA (1) EA200601802A1 (es)
EC (1) ECSP066958A (es)
GB (1) GB0409744D0 (es)
GE (1) GEP20084549B (es)
GT (1) GT200500098A (es)
IL (1) IL178313A0 (es)
MA (1) MA28554B1 (es)
MX (1) MXPA06012640A (es)
NI (1) NI200600257A (es)
NL (1) NL1028927C2 (es)
NO (1) NO20064282L (es)
NZ (1) NZ550054A (es)
PA (1) PA8631601A1 (es)
PE (1) PE20060305A1 (es)
SV (1) SV2005002099A (es)
TN (1) TNSN06347A1 (es)
TW (2) TWI309165B (es)
UA (1) UA86970C2 (es)
UY (1) UY28873A1 (es)
WO (1) WO2005105100A1 (es)
ZA (1) ZA200608661B (es)

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GB0409744D0 (en) * 2004-04-30 2004-06-09 Pfizer Ltd Novel compounds
JP4185154B2 (ja) 2004-04-30 2008-11-26 ワーナー−ランバート カンパニー リミテッド ライアビリティー カンパニー 中枢神経系障害治療用の置換モルホリン化合物
EP1951257A4 (en) * 2005-11-18 2008-11-05 Astrazeneca Ab CRYSTALLINE FORMS
CN101360724A (zh) * 2005-11-18 2009-02-04 阿斯利康公司 盐形式
US20090215744A1 (en) * 2005-11-18 2009-08-27 Astrazeneca Ab Solid Formulations
US8389510B2 (en) * 2005-11-18 2013-03-05 Astrazeneca Ab Crystalline forms
CN101360503A (zh) * 2005-11-18 2009-02-04 阿斯利康公司 液体制剂
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TWI438190B (zh) 2008-07-24 2014-05-21 Theravance Inc 3-(苯氧基苯基甲基)吡咯啶化合物
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