NO20064282L - Morfolinforbindelser - Google Patents

Morfolinforbindelser

Info

Publication number
NO20064282L
NO20064282L NO20064282A NO20064282A NO20064282L NO 20064282 L NO20064282 L NO 20064282L NO 20064282 A NO20064282 A NO 20064282A NO 20064282 A NO20064282 A NO 20064282A NO 20064282 L NO20064282 L NO 20064282L
Authority
NO
Norway
Prior art keywords
compounds
formula
morpholine
adhd
fibromyalgia
Prior art date
Application number
NO20064282A
Other languages
English (en)
Inventor
Alan Stobie
Paul Vincent Fish
Gavin Alistair Whitlock
Florian Wakenhut
Malcolm Christian Mackenny
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=32482498&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20064282(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of NO20064282L publication Critical patent/NO20064282L/no

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A—HUMAN NECESSITIES
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    • A61P1/18—Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
    • A—HUMAN NECESSITIES
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    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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    • C—CHEMISTRY; METALLURGY
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    • C07D265/30—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
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  • General Chemical & Material Sciences (AREA)
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  • Neurology (AREA)
  • Neurosurgery (AREA)
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  • Addiction (AREA)
  • Psychiatry (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Epidemiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Obesity (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Gynecology & Obstetrics (AREA)
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  • Dermatology (AREA)
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Abstract

Det beskrives forbindelser av formel I: hvor R1, R2 , R3 og n har enhver av verdiene definert i beskrivelsen, og farmasøytisk akseptable salter derav, som er nyttige som midler i behandling av tilstander inkluderende urinveisforstyrrelser, smerte, for tidlig ejakulering, ADHD og fibromyalgi. Det tilveiebringes også farmasøytiske materialer omfattende en eller flere forbindelser av formel 1.
NO20064282A 2004-04-30 2006-09-21 Morfolinforbindelser NO20064282L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0409744.0A GB0409744D0 (en) 2004-04-30 2004-04-30 Novel compounds
PCT/IB2005/001154 WO2005105100A1 (en) 2004-04-30 2005-04-20 Morpholine compounds

Publications (1)

Publication Number Publication Date
NO20064282L true NO20064282L (no) 2006-10-18

Family

ID=32482498

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20064282A NO20064282L (no) 2004-04-30 2006-09-21 Morfolinforbindelser

Country Status (33)

Country Link
US (3) US20050250775A1 (no)
EP (1) EP1744754A1 (no)
JP (2) JP4181622B2 (no)
KR (4) KR100896838B1 (no)
CN (1) CN1950089A (no)
AP (1) AP2006003767A0 (no)
AR (1) AR048934A1 (no)
AU (1) AU2005237301A1 (no)
BR (1) BRPI0510515A (no)
CA (1) CA2564990C (no)
CR (1) CR8717A (no)
DO (1) DOP2005000064A (no)
EA (1) EA200601802A1 (no)
EC (1) ECSP066958A (no)
GB (1) GB0409744D0 (no)
GE (1) GEP20084549B (no)
GT (1) GT200500098A (no)
IL (1) IL178313A0 (no)
MA (1) MA28554B1 (no)
MX (1) MXPA06012640A (no)
NI (1) NI200600257A (no)
NL (1) NL1028927C2 (no)
NO (1) NO20064282L (no)
NZ (1) NZ550054A (no)
PA (1) PA8631601A1 (no)
PE (1) PE20060305A1 (no)
SV (1) SV2005002099A (no)
TN (1) TNSN06347A1 (no)
TW (2) TWI309165B (no)
UA (1) UA86970C2 (no)
UY (1) UY28873A1 (no)
WO (1) WO2005105100A1 (no)
ZA (1) ZA200608661B (no)

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GB0409744D0 (en) * 2004-04-30 2004-06-09 Pfizer Ltd Novel compounds
CN101360724A (zh) * 2005-11-18 2009-02-04 阿斯利康公司 盐形式
EP1951693A4 (en) * 2005-11-18 2012-05-30 Astrazeneca Ab SOLID FORMULATIONS
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JP2009516708A (ja) * 2005-11-18 2009-04-23 アストラゼネカ・アクチエボラーグ 液体製剤
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KR101103118B1 (ko) * 2007-11-02 2012-01-04 동아제약주식회사 신규한 1,3-디히드로-5-이소벤조퓨란카르보니트릴 유도체 화합물 및 이를 함유하는 조루증 치료용 약학조성물
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