UA94902C2 - Лечение болезни паркинсона, обструктивного апное сна, деменции с тельцами леви, сосудистой деменции неимидазольными алкиламинами, которые являются лигандами h3-рецептора гистамина - Google Patents

Лечение болезни паркинсона, обструктивного апное сна, деменции с тельцами леви, сосудистой деменции неимидазольными алкиламинами, которые являются лигандами h3-рецептора гистамина

Info

Publication number
UA94902C2
UA94902C2 UAA200710712A UAA200710712A UA94902C2 UA 94902 C2 UA94902 C2 UA 94902C2 UA A200710712 A UAA200710712 A UA A200710712A UA A200710712 A UAA200710712 A UA A200710712A UA 94902 C2 UA94902 C2 UA 94902C2
Authority
UA
Ukraine
Prior art keywords
dementia
parkinson
disease
treatment
sleep apnea
Prior art date
Application number
UAA200710712A
Other languages
English (en)
Russian (ru)
Ukrainian (uk)
Inventor
Жан-Шарль Шварц
Жан-Мари Леконт
Original Assignee
Биопроже
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35169680&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UA94902(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Биопроже filed Critical Биопроже
Publication of UA94902C2 publication Critical patent/UA94902C2/ru

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4453Non condensed piperidines, e.g. piperocaine only substituted in position 1, e.g. propipocaine, diperodon
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Psychiatry (AREA)
  • Psychology (AREA)
  • Anesthesiology (AREA)
  • Pulmonology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
UAA200710712A 2005-04-01 2006-03-30 Лечение болезни паркинсона, обструктивного апное сна, деменции с тельцами леви, сосудистой деменции неимидазольными алкиламинами, которые являются лигандами h3-рецептора гистамина UA94902C2 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP05290727A EP1707203A1 (en) 2005-04-01 2005-04-01 Treatment of parkinson's disease obstructive sleep apnea, dementia with lewy bodies, vascular dementia with non-imidazole alkylamines histamine H3- receptor ligands

Publications (1)

Publication Number Publication Date
UA94902C2 true UA94902C2 (ru) 2011-06-25

Family

ID=35169680

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200710712A UA94902C2 (ru) 2005-04-01 2006-03-30 Лечение болезни паркинсона, обструктивного апное сна, деменции с тельцами леви, сосудистой деменции неимидазольными алкиламинами, которые являются лигандами h3-рецептора гистамина

Country Status (27)

Country Link
US (1) US8486947B2 (enExample)
EP (2) EP1707203A1 (enExample)
JP (3) JP5546761B2 (enExample)
KR (1) KR101308527B1 (enExample)
CN (1) CN101171009B (enExample)
AU (1) AU2006228413C1 (enExample)
BR (1) BRPI0612216B1 (enExample)
CA (1) CA2603656C (enExample)
CY (1) CY1114636T1 (enExample)
DK (1) DK1863487T4 (enExample)
EA (1) EA016007B1 (enExample)
ES (1) ES2426008T5 (enExample)
HR (1) HRP20130748T4 (enExample)
MA (1) MA29353B1 (enExample)
ME (1) ME01713B (enExample)
MX (1) MX2007012162A (enExample)
NO (1) NO343603B1 (enExample)
NZ (1) NZ561940A (enExample)
PL (1) PL1863487T5 (enExample)
PT (1) PT1863487E (enExample)
RS (1) RS52911B2 (enExample)
SG (1) SG147415A1 (enExample)
SI (1) SI1863487T2 (enExample)
TN (1) TNSN07365A1 (enExample)
UA (1) UA94902C2 (enExample)
WO (1) WO2006103546A2 (enExample)
ZA (1) ZA200708086B (enExample)

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NZ574873A (en) 2006-07-25 2012-03-30 Cephalon Inc Pyridazinone derivatives as h3 inhibitors
US8153813B2 (en) 2007-12-20 2012-04-10 Abbott Laboratories Benzothiazole and benzooxazole derivatives and methods of use
CA2712897A1 (en) 2008-01-30 2009-08-06 Pharmacopeia, Inc. Substituted spirocyclic piperidine derivatives as histamine-3 (h3) receptor ligands
FR2932479A1 (fr) 2008-06-13 2009-12-18 Servier Lab Nouveaux derives azabicycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
US9186353B2 (en) 2009-04-27 2015-11-17 Abbvie Inc. Treatment of osteoarthritis pain
WO2012037258A1 (en) 2010-09-16 2012-03-22 Abbott Laboratories Processes for preparing 1,2-substituted cyclopropyl derivatives
US9181275B2 (en) 2011-08-11 2015-11-10 Abbvie Inc. Mercaptoamidine derivatives and methods of use
WO2013151982A1 (en) 2012-04-03 2013-10-10 Arena Pharmaceuticals, Inc. Methods and compounds useful in treating pruritus, and methods for identifying such compounds
SG11201502210VA (en) * 2012-10-05 2015-04-29 Vtvx Holdings I Llc Treatment of mild and moderate alzheimer's disease
EP3391886A1 (en) 2017-04-19 2018-10-24 Novartis AG The use of a h3r inverse agonist for the treatment of shift work disorder
US20200281522A1 (en) 2019-03-06 2020-09-10 Medtronic Xomed, LLC System and method for improved obstructive sleep apnea diagnostic for implantable devices
EP4248969A1 (en) 2022-03-23 2023-09-27 Bioprojet Use of pitolisant for treating severe fatigue
WO2024201139A1 (en) 2023-03-31 2024-10-03 Bioprojet Pharma Polymorph form of pitolisant hydrochloride
TW202535385A (zh) 2023-10-16 2025-09-16 法商拜爾普羅傑特醫藥有限公司 必托里賽(pitolisant)之新穎調配物及使用方法

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Also Published As

Publication number Publication date
EP1707203A1 (en) 2006-10-04
AU2006228413B2 (en) 2011-09-15
CA2603656A1 (en) 2006-10-05
JP2014062126A (ja) 2014-04-10
CY1114636T1 (el) 2016-10-05
HRP20130748T1 (en) 2013-10-11
MA29353B1 (fr) 2008-03-03
HRP20130748T4 (hr) 2019-11-15
DK1863487T4 (da) 2019-10-14
WO2006103546A3 (en) 2007-03-01
US20090318433A1 (en) 2009-12-24
CN101171009A (zh) 2008-04-30
BRPI0612216B1 (pt) 2022-04-19
JP5546761B2 (ja) 2014-07-09
KR20080002904A (ko) 2008-01-04
EP1863487A2 (en) 2007-12-12
EP1863487B1 (en) 2013-05-29
TNSN07365A1 (fr) 2008-12-31
JP2016106142A (ja) 2016-06-16
JP5955872B2 (ja) 2016-07-20
JP2008534572A (ja) 2008-08-28
EA200702135A1 (ru) 2008-04-28
RS52911B2 (sr) 2019-11-29
PL1863487T5 (pl) 2021-08-09
DK1863487T3 (da) 2013-08-12
ME01713B (me) 2014-09-20
AU2006228413C1 (en) 2012-02-02
SI1863487T1 (sl) 2013-09-30
RS52911B (en) 2014-02-28
KR101308527B1 (ko) 2013-09-17
ZA200708086B (en) 2008-10-29
AU2006228413A1 (en) 2006-10-05
BRPI0612216A2 (pt) 2010-10-26
NO20075086L (no) 2007-12-27
SG147415A1 (en) 2008-11-28
MX2007012162A (es) 2007-11-22
PL1863487T3 (pl) 2014-10-31
EA016007B1 (ru) 2012-01-30
NO343603B1 (no) 2019-04-08
CA2603656C (en) 2015-06-16
CN101171009B (zh) 2012-11-07
SI1863487T2 (sl) 2019-11-29
NZ561940A (en) 2010-06-25
PT1863487E (pt) 2013-08-29
US8486947B2 (en) 2013-07-16
EP1863487B2 (en) 2019-07-17
ES2426008T3 (es) 2013-10-18
WO2006103546A2 (en) 2006-10-05
ES2426008T5 (es) 2020-03-20

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