UA80162C2 - Novel alkyne compounds having an mch antagonistic effect and medicaments containing these compounds - Google Patents

Novel alkyne compounds having an mch antagonistic effect and medicaments containing these compounds Download PDF

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Publication number
UA80162C2
UA80162C2 UAA200505138A UA2005005138A UA80162C2 UA 80162 C2 UA80162 C2 UA 80162C2 UA A200505138 A UAA200505138 A UA A200505138A UA 2005005138 A UA2005005138 A UA 2005005138A UA 80162 C2 UA80162 C2 UA 80162C2
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UA
Ukraine
Prior art keywords
group
chlorophenyl
pyridin
salkyl
ylethynyl
Prior art date
Application number
UAA200505138A
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English (en)
Ukrainian (uk)
Inventor
Stephan-Georg Mueller
Dirk Stenkamp
Kirsten Arndt
Gerald Juergen Roth
Ralf Richard Hermann Lotz
Thorsten Lehmann-Lintz
Martin Lenter
Philipp Lustenberger
Klaus Rudolf
Original Assignee
Boehringer Ingelheim Pharma
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Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of UA80162C2 publication Critical patent/UA80162C2/uk

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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/44—Radicals substituted by doubly-bound oxygen, sulfur, or nitrogen atoms, or by two such atoms singly-bound to the same carbon atom
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    • C07D213/48—Aldehydo radicals
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4418—Non condensed pyridines; Hydrogenated derivatives thereof having a carbocyclic group directly attached to the heterocyclic ring, e.g. cyproheptadine
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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UAA200505138A 2002-10-31 2003-10-25 Novel alkyne compounds having an mch antagonistic effect and medicaments containing these compounds UA80162C2 (en)

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