UA73144C2 - Tricyclic inhibitor of poly(adp-ribosyl)transferase, pharmaceutical composition including thereof and method for inhibiting of activness of poly(adp-ribosyl)transferase in enzymes - Google Patents

Info

Publication number

UA73144C2

UA73144C2 UA2002042574A UA2002042574A UA73144C2 UA 73144 C2 UA73144 C2 UA 73144C2 UA 2002042574 A UA2002042574 A UA 2002042574A UA 2002042574 A UA2002042574 A UA 2002042574A UA 73144 C2 UA73144 C2 UA 73144C2

Authority

UA

Ukraine

Prior art keywords

aryl

cycloalkyl

alkynyl

alkenyl

heterocycloalkyl

Prior art date

1999-08-31

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• 238000000034 method Methods 0.000 title claims description 207
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• 108090000790 Enzymes Proteins 0.000 title claims description 38
• 230000002401 inhibitory effect Effects 0.000 title claims description 25
• 239000008194 pharmaceutical composition Substances 0.000 title claims description 10
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• 125000003277 amino group Chemical group 0.000 claims description 41
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