UA5980A1 - Спосіб одержання сульфаілзаміщаних похідних фенетіламіна, а також їх кислотно-адитивних солей - Google Patents
Спосіб одержання сульфаілзаміщаних похідних фенетіламіна, а також їх кислотно-адитивних солейInfo
- Publication number
- UA5980A1 UA5980A1 UA3245545A UA3245545A UA5980A1 UA 5980 A1 UA5980 A1 UA 5980A1 UA 3245545 A UA3245545 A UA 3245545A UA 3245545 A UA3245545 A UA 3245545A UA 5980 A1 UA5980 A1 UA 5980A1
- Authority
- UA
- Ukraine
- Prior art keywords
- producing
- acid additive
- additive salts
- phenethylamine derivatives
- substituted phenethylamine
- Prior art date
Links
- BHHGXPLMPWCGHP-UHFFFAOYSA-N Phenethylamine Chemical class NCCC1=CC=CC=C1 BHHGXPLMPWCGHP-UHFFFAOYSA-N 0.000 title abstract 2
- 239000002253 acid Substances 0.000 title abstract 2
- 239000000654 additive Substances 0.000 title abstract 2
- 230000000996 additive effect Effects 0.000 title abstract 2
- 125000004397 aminosulfonyl group Chemical group NS(=O)(=O)* 0.000 title abstract 2
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- 150000003839 salts Chemical class 0.000 title abstract 2
- 239000003960 organic solvent Substances 0.000 abstract 2
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- 239000003054 catalyst Substances 0.000 abstract 1
- 239000003795 chemical substances by application Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 230000026030 halogenation Effects 0.000 abstract 1
- 238000005658 halogenation reaction Methods 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D203/00—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom
- C07D203/04—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D203/06—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D203/08—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring nitrogen atom
- C07D203/10—Radicals substituted by singly bound oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Cardiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Heart & Thoracic Surgery (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Hospice & Palliative Care (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
Предметом винаходу є спосіб одержання сульфамоїлзаміщених похідних фенетиламіну, а також їхніх кислотно-адитивних солей. Сполуку певної формули піддають взаємодії з галоїдувальним агентом в середовищі органічного розчинника, а потім при необхідності отриманий при цьому галоїдований продукт відновлюється воднем у присутності каталізатора в середовищі органічного розчинника.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP1438280A JPS56110665A (en) | 1980-02-08 | 1980-02-08 | Sulfamoyl-substituted phenetylamine derivative and its preparation |
Publications (1)
Publication Number | Publication Date |
---|---|
UA5980A1 true UA5980A1 (uk) | 1994-12-29 |
Family
ID=11859488
Family Applications (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UA3379949A UA5981A1 (uk) | 1980-02-08 | 1981-02-06 | Спосіб одержання сульфамоілзаміщеного похідного фенетіламіна і його кислотної солі |
UA3245545A UA5980A1 (uk) | 1980-02-08 | 1981-02-06 | Спосіб одержання сульфаілзаміщаних похідних фенетіламіна, а також їх кислотно-адитивних солей |
UA3382004A UA5990A1 (uk) | 1980-02-08 | 1981-02-06 | Спосіб одержання сульфамоілзаміщених похідних фенетіламіна або його солянокислої солі |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UA3379949A UA5981A1 (uk) | 1980-02-08 | 1981-02-06 | Спосіб одержання сульфамоілзаміщеного похідного фенетіламіна і його кислотної солі |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UA3382004A UA5990A1 (uk) | 1980-02-08 | 1981-02-06 | Спосіб одержання сульфамоілзаміщених похідних фенетіламіна або його солянокислої солі |
Country Status (17)
Country | Link |
---|---|
US (6) | US4373106A (uk) |
EP (1) | EP0034432B1 (uk) |
JP (1) | JPS56110665A (uk) |
AR (2) | AR227533A1 (uk) |
AT (1) | ATE7223T1 (uk) |
AU (1) | AU541720B2 (uk) |
CA (1) | CA1177849A (uk) |
DE (2) | DE19675042I2 (uk) |
ES (1) | ES499224A0 (uk) |
GR (1) | GR73827B (uk) |
IE (1) | IE50862B1 (uk) |
LU (1) | LU90000I2 (uk) |
MX (2) | MX6859E (uk) |
NL (1) | NL950014I2 (uk) |
PT (1) | PT72460B (uk) |
SU (3) | SU1082320A3 (uk) |
UA (3) | UA5981A1 (uk) |
Families Citing this family (104)
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Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3701808A (en) * | 1967-12-21 | 1972-10-31 | Allen & Hanburys Ltd | Phenylethanolamines |
ES373606A1 (es) * | 1968-11-18 | 1972-06-01 | Pfizer | Un procedimiento para la preparacion de nuevos derivados depropanolamina. |
US3878212A (en) * | 1970-04-28 | 1975-04-15 | Clemens Rufer | Blood sugar lowering sulfamoyl pyrimidines and asymmetrical carbon atom |
US4137328A (en) * | 1970-07-18 | 1979-01-30 | Pfizer Inc. | Phenyl-alkanolamine, alkylamine and α-aminoalkyl ketone derivatives as heart stimulants |
US3711545A (en) * | 1971-02-23 | 1973-01-16 | Smith Kline French Lab | Alpha-aminoalkyl-4-hydroxy-3-sulfamoylaminobenzyl alcohols |
DE2115926C3 (de) * | 1971-04-01 | 1978-05-03 | C.H. Boehringer Sohn, 6507 Ingelheim | 1 -(4-Hydroxy-3-dimethylaminosuIfamidophenyI)-2-aminoäthanderivate, Verfahren zu ihrer Herstellung und diese enthaltende Mittel |
US3860647A (en) * | 1973-08-20 | 1975-01-14 | Smithkline Corp | {60 -Aminomethyl-4-hydroxy-3-sulfamyl-benzyl alcohols and 4-hydroxy-3-sulfamyl phenethylamines |
GB1593651A (en) * | 1977-02-03 | 1981-07-22 | Allen & Hanburys Ltd | Amides |
CA1147342A (en) * | 1977-10-12 | 1983-05-31 | Kazuo Imai | Process of producing novel phenylethanolamine derivatives |
JPS5553261A (en) * | 1978-10-17 | 1980-04-18 | Yamanouchi Pharmaceut Co Ltd | New phenylethanolamine derivative and its preparation |
JPS5553262A (en) * | 1978-10-17 | 1980-04-18 | Yamanouchi Pharmaceut Co Ltd | Phenylethanolamine derivative |
JPS606330B2 (ja) * | 1978-11-30 | 1985-02-18 | 山之内製薬株式会社 | α・β両遮断剤 |
JPS56110665A (en) * | 1980-02-08 | 1981-09-01 | Yamanouchi Pharmaceut Co Ltd | Sulfamoyl-substituted phenetylamine derivative and its preparation |
US4558156A (en) * | 1980-02-08 | 1985-12-10 | Yamanouchi Pharmaceutical Co., Ltd. | Sulfamoyl-substituted phenethylamine derivatives |
DE3110573A1 (de) * | 1981-03-18 | 1982-10-21 | Bayer Ag, 5090 Leverkusen | Verfahren zur herstellung von n- und o-substituierten di- und/oder polyurethanen |
JPS5950671B2 (ja) * | 1982-08-26 | 1984-12-10 | 山之内製薬株式会社 | フェニルエタノ−ルアミン誘導体およびその製造法 |
US4558106A (en) * | 1983-03-29 | 1985-12-10 | Union Carbide Corporation | Polymerization process using metal formate to reduce the color of thermoplastic copolymers |
-
1980
- 1980-02-08 JP JP1438280A patent/JPS56110665A/ja active Granted
-
1981
- 1981-01-19 AR AR283989A patent/AR227533A1/es active
- 1981-01-23 CA CA000369230A patent/CA1177849A/en not_active Expired
- 1981-02-02 AT AT81300431T patent/ATE7223T1/de active
- 1981-02-02 DE DE1996175042 patent/DE19675042I2/de active Active
- 1981-02-02 DE DE8181300431T patent/DE3163257D1/de not_active Expired
- 1981-02-02 EP EP81300431A patent/EP0034432B1/en not_active Expired
- 1981-02-04 GR GR64051A patent/GR73827B/el unknown
- 1981-02-04 AU AU66896/81A patent/AU541720B2/en not_active Expired
- 1981-02-04 US US06/231,421 patent/US4373106A/en not_active Expired - Lifetime
- 1981-02-05 PT PT72460A patent/PT72460B/pt unknown
- 1981-02-06 IE IE236/81A patent/IE50862B1/en not_active IP Right Cessation
- 1981-02-06 ES ES499224A patent/ES499224A0/es active Granted
- 1981-02-06 UA UA3379949A patent/UA5981A1/uk unknown
- 1981-02-06 UA UA3245545A patent/UA5980A1/uk unknown
- 1981-02-06 UA UA3382004A patent/UA5990A1/uk unknown
- 1981-02-06 SU SU813245545A patent/SU1082320A3/ru active
- 1981-02-09 MX MX819298U patent/MX6859E/es unknown
-
1982
- 1982-01-21 SU SU823379949A patent/SU1181540A3/ru active
- 1982-01-29 SU SU823382004A patent/SU1248533A3/ru active
- 1982-02-26 AR AR288580A patent/AR230433A1/es active
-
1985
- 1985-07-18 US US06/756,790 patent/US4703063A/en not_active Expired - Lifetime
- 1985-11-27 US US06/803,204 patent/US4731478A/en not_active Expired - Lifetime
-
1986
- 1986-02-10 US US06/828,052 patent/US4761500A/en not_active Expired - Lifetime
-
1989
- 1989-02-14 US US07/311,366 patent/US4868216A/en not_active Expired - Lifetime
- 1989-11-13 US US07/436,125 patent/US4987152A/en not_active Expired - Lifetime
-
1992
- 1992-06-26 MX MX9203592A patent/MX9203592A/es unknown
-
1995
- 1995-08-18 NL NL950014C patent/NL950014I2/nl unknown
-
1997
- 1997-01-03 LU LU90000C patent/LU90000I2/fr unknown
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