UA124922C2 - Модулятори ядерного транспорту та їх застосування - Google Patents

Модулятори ядерного транспорту та їх застосування

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Publication number
UA124922C2
UA124922C2 UAA201710733A UAA201710733A UA124922C2 UA 124922 C2 UA124922 C2 UA 124922C2 UA A201710733 A UAA201710733 A UA A201710733A UA A201710733 A UAA201710733 A UA A201710733A UA 124922 C2 UA124922 C2 UA 124922C2
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UA
Ukraine
Prior art keywords
applications
nuclear transport
transport modulators
compounds
formula
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Application number
UAA201710733A
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English (en)
Inventor
Вінсент П. Санданаяка
Шерон Шехтер
Шерон Шачам
Діляра МакКолі
Еркан Балоглу
Original Assignee
Біоген Ма Інк.
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49448240&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UA124922(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Біоген Ма Інк. filed Critical Біоген Ма Інк.
Publication of UA124922C2 publication Critical patent/UA124922C2/uk

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4196—1,2,4-Triazoles
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
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    • A61K31/4965—Non-condensed pyrazines
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
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Abstract

Даний винахід стосується сполук формули І (І) та їх фармацевтично прийнятних солей, фармацевтичних композицій, що містять сполуки формули І, та способів застосування вказаних сполук, солей та композицій в лікуванні різних порушень, пов'язаних з активністю CRM1.
UAA201710733A 2012-05-09 2013-05-09 Модулятори ядерного транспорту та їх застосування UA124922C2 (uk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261644802P 2012-05-09 2012-05-09
US201361798188P 2013-03-15 2013-03-15

Publications (1)

Publication Number Publication Date
UA124922C2 true UA124922C2 (uk) 2021-12-15

Family

ID=49448240

Family Applications (2)

Application Number Title Priority Date Filing Date
UAA201710733A UA124922C2 (uk) 2012-05-09 2013-05-09 Модулятори ядерного транспорту та їх застосування
UAA201413015A UA118085C2 (uk) 2012-05-09 2013-05-09 Модулятори ядерного транспорту та їх застосування

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UAA201413015A UA118085C2 (uk) 2012-05-09 2013-05-09 Модулятори ядерного транспорту та їх застосування

Country Status (32)

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US (10) US9096543B2 (uk)
EP (3) EP3404027B1 (uk)
JP (5) JP6195909B2 (uk)
KR (5) KR102095429B1 (uk)
CN (1) CN104428295B (uk)
AU (5) AU2013259384B2 (uk)
BR (1) BR112014027860B8 (uk)
CA (1) CA2872190C (uk)
CL (1) CL2014003054A1 (uk)
CO (1) CO7190242A2 (uk)
CY (2) CY1120832T1 (uk)
DK (2) DK3404027T3 (uk)
EA (1) EA036639B1 (uk)
ES (2) ES2702279T3 (uk)
GE (1) GEP20237477B (uk)
HK (1) HK1209420A1 (uk)
HR (2) HRP20181838T1 (uk)
HU (2) HUE050452T2 (uk)
IN (1) IN2014DN09434A (uk)
LT (2) LT3404027T (uk)
ME (1) ME03795B (uk)
MX (1) MX364992B (uk)
NZ (1) NZ702663A (uk)
PE (1) PE20150128A1 (uk)
PL (2) PL3404027T3 (uk)
PT (2) PT3404027T (uk)
RS (2) RS58058B1 (uk)
SG (1) SG11201407268SA (uk)
SI (2) SI3404027T1 (uk)
UA (2) UA124922C2 (uk)
WO (1) WO2013170068A2 (uk)
ZA (1) ZA202004892B (uk)

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