TW201609708A - 新穎２，５－經取代之嘧啶 - Google Patents

新穎２，５－經取代之嘧啶 Download PDF

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TW201609708A
TW201609708A TW104123022A TW104123022A TW201609708A TW 201609708 A TW201609708 A TW 201609708A TW 104123022 A TW104123022 A TW 104123022A TW 104123022 A TW104123022 A TW 104123022A TW 201609708 A TW201609708 A TW 201609708A
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Taiwan
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alkyl
group
alkylene
compound
pyrimidin
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TW104123022A
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English (en)
Chinese (zh)
Inventor
英葛 柯奈茲奇
托比雅斯 克朗
芙羅利安 雅寇柏
安東尼歐 納爾迪
克利斯提安 賀斯林格
安德烈 瑋柏斯
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歌林達有限公司
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Publication of TW201609708A publication Critical patent/TW201609708A/zh

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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TW104123022A 2014-07-16 2015-07-16 新穎２，５－經取代之嘧啶 TW201609708A (zh)

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AU2015291477A1 (en) 2017-03-09
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PE20170119A1 (es) 2017-03-30
EP3169680A1 (en) 2017-05-24
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