TR201821285T4 - CCR3 antagonisti içeren farmasötik formülasyonlar. - Google Patents

CCR3 antagonisti içeren farmasötik formülasyonlar. Download PDF

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Publication number
TR201821285T4
TR201821285T4 TR2018/21285T TR201821285T TR201821285T4 TR 201821285 T4 TR201821285 T4 TR 201821285T4 TR 2018/21285 T TR2018/21285 T TR 2018/21285T TR 201821285 T TR201821285 T TR 201821285T TR 201821285 T4 TR201821285 T4 TR 201821285T4
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TR
Turkey
Prior art keywords
tablet
tablets
solvent
lubricant
premix
Prior art date
Application number
TR2018/21285T
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English (en)
Turkish (tr)
Inventor
Fetscher Alfred
Matthias Scher Jochen
Original Assignee
Alkahest Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49292482&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TR201821285(T4) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Alkahest Inc filed Critical Alkahest Inc
Publication of TR201821285T4 publication Critical patent/TR201821285T4/tr

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
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  • Veterinary Medicine (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
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  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Pain & Pain Management (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Neurology (AREA)
  • Dermatology (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Otolaryngology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Transplantation (AREA)
  • Diabetes (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
TR2018/21285T 2012-04-04 2013-04-02 CCR3 antagonisti içeren farmasötik formülasyonlar. TR201821285T4 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP12163078 2012-04-04

Publications (1)

Publication Number Publication Date
TR201821285T4 true TR201821285T4 (tr) 2019-01-21

Family

ID=49292482

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2018/21285T TR201821285T4 (tr) 2012-04-04 2013-04-02 CCR3 antagonisti içeren farmasötik formülasyonlar.

Country Status (31)

Country Link
US (3) US10213421B2 (enEXAMPLES)
EP (3) EP2833864B1 (enEXAMPLES)
JP (4) JP6320990B2 (enEXAMPLES)
KR (2) KR102138709B1 (enEXAMPLES)
CN (1) CN104203213A (enEXAMPLES)
AR (1) AR090596A1 (enEXAMPLES)
AU (1) AU2013245028B2 (enEXAMPLES)
BR (1) BR112014024479A8 (enEXAMPLES)
CA (1) CA2869058C (enEXAMPLES)
CL (1) CL2014002524A1 (enEXAMPLES)
CY (1) CY1121137T1 (enEXAMPLES)
DK (2) DK3524230T3 (enEXAMPLES)
EA (1) EA027627B1 (enEXAMPLES)
ES (2) ES2898179T3 (enEXAMPLES)
HR (1) HRP20190069T1 (enEXAMPLES)
HU (2) HUE041519T2 (enEXAMPLES)
IL (1) IL234299A (enEXAMPLES)
IN (1) IN2014DN07082A (enEXAMPLES)
LT (1) LT2833864T (enEXAMPLES)
MX (1) MX358307B (enEXAMPLES)
NZ (1) NZ628993A (enEXAMPLES)
PH (1) PH12014502241A1 (enEXAMPLES)
PL (2) PL3524230T3 (enEXAMPLES)
PT (2) PT2833864T (enEXAMPLES)
RS (1) RS58360B1 (enEXAMPLES)
SI (1) SI2833864T1 (enEXAMPLES)
SM (1) SMT201900121T1 (enEXAMPLES)
TR (1) TR201821285T4 (enEXAMPLES)
TW (1) TW201400115A (enEXAMPLES)
UY (1) UY34730A (enEXAMPLES)
WO (1) WO2013149987A1 (enEXAMPLES)

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US8278302B2 (en) 2009-04-08 2012-10-02 Boehringer Ingelheim International Gmbh Substituted piperidines as CCR3 antagonists
UA109290C2 (uk) 2010-10-07 2015-08-10 Спільні кристали і солі інгібіторів ccr3
US8680280B2 (en) 2012-04-02 2014-03-25 Boehringer Ingelheim International Gmbh Process for the manufacturing of CRR inhibitors
US20130261153A1 (en) * 2012-04-03 2013-10-03 Boehringer Ingelheim International Gmbh Use of ccr3-inhibitors
US10213421B2 (en) * 2012-04-04 2019-02-26 Alkahest, Inc. Pharmaceutical formulations comprising CCR3 antagonists
UA125658C2 (uk) 2017-04-05 2022-05-11 Алкахест Інк. Спосіб та композиція для лікування захворювання, пов'язаного з сітківкою ока, з використанням інгібітора ccr3
JP2020513005A (ja) * 2017-04-05 2020-04-30 アルカヘスト，インコーポレイテッド Ｃｃｒ３阻害剤を用いて、加齢性機能障害を治療するための方法及び組成物
US20190111042A1 (en) * 2017-10-13 2019-04-18 Alkahest, Inc. Methods and Compositions for Treating Pruritus, Xerosis, and Associated Disease Using CCR-Inhibitors
CA3097083A1 (en) 2018-05-15 2019-11-21 Alkahest, Inc. Treatment of aging-associated disease with modulators of leukotriene a4 hydrolase
WO2020069008A1 (en) * 2018-09-26 2020-04-02 Alkahest, Inc. Methods and compositions for treating aging-associated impairments using ccr3-inhibitors
EP4206153A4 (en) 2020-08-27 2024-05-15 Agc Inc. ALKALI-FREE GLASS AND PLATE GLASS
CA3221177A1 (en) 2021-11-01 2023-05-04 Meghan Kerrisk Campbell Benzodioxane modulators of leukotriene a4 hydrolase (lta4h) for prevention and treatment of aging-associated diseases

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