TN2009000481A1 - Novel peptide inhibitors of hepatitis c virus replication - Google Patents

Novel peptide inhibitors of hepatitis c virus replication

Info

Publication number
TN2009000481A1
TN2009000481A1 TNP2009000481A TN2009000481A TN2009000481A1 TN 2009000481 A1 TN2009000481 A1 TN 2009000481A1 TN P2009000481 A TNP2009000481 A TN P2009000481A TN 2009000481 A TN2009000481 A TN 2009000481A TN 2009000481 A1 TN2009000481 A1 TN 2009000481A1
Authority
TN
Tunisia
Prior art keywords
hepatitis
methods
virus replication
subject compound
peptide inhibitors
Prior art date
Application number
TNP2009000481A
Other languages
English (en)
Inventor
Steven W Andrews
Scott Seiwert
Leonid Beigelman
Lawrence Blatt
Brad Buckman
Yutong Jiang
Robert J Kaus
April L Kennedy
Timothy S Kercher
Michael A Lyon
Bin Wang
Kevin R Condroski
Original Assignee
Array Biopharma Inc
Intermune Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39743068&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TN2009000481(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Array Biopharma Inc, Intermune Inc filed Critical Array Biopharma Inc
Publication of TN2009000481A1 publication Critical patent/TN2009000481A1/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D217/00Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/22Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
    • C07D217/26Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Virology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Communicable Diseases (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Epidemiology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
TNP2009000481A 2007-05-10 2009-11-10 Novel peptide inhibitors of hepatitis c virus replication TN2009000481A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US91730007P 2007-05-10 2007-05-10
US2304108P 2008-01-23 2008-01-23
PCT/US2008/063304 WO2008141227A1 (fr) 2007-05-10 2008-05-09 Nouveaux inhibiteurs peptidiques de la réplication du virus de l'hépatite c

Publications (1)

Publication Number Publication Date
TN2009000481A1 true TN2009000481A1 (en) 2011-03-31

Family

ID=39743068

Family Applications (1)

Application Number Title Priority Date Filing Date
TNP2009000481A TN2009000481A1 (en) 2007-05-10 2009-11-10 Novel peptide inhibitors of hepatitis c virus replication

Country Status (22)

Country Link
US (1) US7932277B2 (fr)
EP (1) EP2185524A1 (fr)
JP (1) JP2010526834A (fr)
KR (1) KR20100027134A (fr)
CN (1) CN101679277A (fr)
AP (1) AP2009005057A0 (fr)
AR (1) AR066528A1 (fr)
AU (1) AU2008251425A1 (fr)
BR (1) BRPI0811447A2 (fr)
CA (1) CA2686546A1 (fr)
CL (1) CL2008001381A1 (fr)
CO (1) CO6241100A2 (fr)
EA (1) EA200971041A1 (fr)
EC (1) ECSP099792A (fr)
IL (1) IL201842A0 (fr)
MA (1) MA31497B1 (fr)
MX (1) MX2009012093A (fr)
NI (1) NI200900205A (fr)
TN (1) TN2009000481A1 (fr)
TW (1) TW200902520A (fr)
WO (1) WO2008141227A1 (fr)
ZA (1) ZA200907858B (fr)

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UA119315C2 (uk) 2012-07-03 2019-06-10 Гіліад Фармассет Елелсі Інгібітори вірусу гепатиту с
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CN101679277A (zh) 2010-03-24
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