SMT201500223B - Polimorfi e sali di n-[5-[4-(5-{[(2R,6S)-2,6-dimetil-4-morfolinil]metil}-1,3-ossazol-2-il)-1H-indazol-6-IL]-2-(metilossi)-3-piridinilÜmetansolfonammide - Google Patents
Polimorfi e sali di n-[5-[4-(5-{[(2R,6S)-2,6-dimetil-4-morfolinil]metil}-1,3-ossazol-2-il)-1H-indazol-6-IL]-2-(metilossi)-3-piridinilÜmetansolfonammideInfo
- Publication number
- SMT201500223B SMT201500223B SM201500223T SM201500223T SMT201500223B SM T201500223 B SMT201500223 B SM T201500223B SM 201500223 T SM201500223 T SM 201500223T SM 201500223 T SM201500223 T SM 201500223T SM T201500223 B SMT201500223 B SM T201500223B
- Authority
- SM
- San Marino
- Prior art keywords
- piridinilümetansolfonammide
- methyloxy
- indazol
- oxazol
- polymorphs
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Epidemiology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US38074810P | 2010-09-08 | 2010-09-08 | |
| PCT/EP2011/065419 WO2012032067A1 (en) | 2010-09-08 | 2011-09-06 | Polymorphs and salts of n- [5- [4- (5- { [(2r,6s) -2, 6 - dimethyl - 4 -morpholinyl] methyl} - 1, 3 - oxazol - 2 - yl) - 1h- inda zol-6-yl] -2- (methyloxy) - 3 - pyridinyl] methanesulfonamide |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SMT201500223B true SMT201500223B (it) | 2015-10-30 |
Family
ID=44645691
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SM201500223T SMT201500223B (it) | 2010-09-08 | 2015-09-22 | Polimorfi e sali di n-[5-[4-(5-{[(2R,6S)-2,6-dimetil-4-morfolinil]metil}-1,3-ossazol-2-il)-1H-indazol-6-IL]-2-(metilossi)-3-piridinilÜmetansolfonammide |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US8735390B2 (ja) |
| EP (1) | EP2614058B1 (ja) |
| JP (1) | JP5965402B2 (ja) |
| DK (1) | DK2614058T3 (ja) |
| ES (1) | ES2548036T3 (ja) |
| HR (1) | HRP20151017T1 (ja) |
| HU (1) | HUE026059T2 (ja) |
| PL (1) | PL2614058T3 (ja) |
| PT (1) | PT2614058E (ja) |
| RS (1) | RS54286B1 (ja) |
| SI (1) | SI2614058T1 (ja) |
| SM (1) | SMT201500223B (ja) |
| WO (1) | WO2012032067A1 (ja) |
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| ES2602972T3 (es) * | 2010-09-08 | 2017-02-23 | Glaxosmithkline Intellectual Property Development Limited | Derivados de indazol para su uso en el tratamiento de infección por virus de la gripe |
| GB201018124D0 (en) | 2010-10-27 | 2010-12-08 | Glaxo Group Ltd | Polymorphs and salts |
| JP6063870B2 (ja) | 2010-11-08 | 2017-01-18 | ライセラ・コーポレイション | ＲＯＲγ活性の阻害用のＮ−スルホニル化テトラヒドロキノリンおよび関連二環化合物および病気の治療 |
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| TW200811171A (en) | 2003-10-14 | 2008-03-01 | Glaxo Group Ltd | Muscarinic acetylcholine receptor antagonists |
| WO2005044354A1 (en) | 2003-11-03 | 2005-05-19 | Glaxo Group Limited | A fluid dispensing device |
| TW200524577A (en) | 2003-11-04 | 2005-08-01 | Glaxo Group Ltd | Muscarinic acetylcholine receptor antagonists |
| US20070111995A1 (en) | 2003-12-19 | 2007-05-17 | Allen David G | Pyrazolo [3,4-B] pyridine Compounds and Their Use as Phosphodiesterase Inhibitors |
| WO2005090352A1 (en) | 2004-03-16 | 2005-09-29 | Glaxo Group Limited | Pyrazolo[3,4-b]pyridine compound, and its use as a pde4 inhibitor |
| GB0405937D0 (en) | 2004-03-16 | 2004-04-21 | Glaxo Group Ltd | Compounds |
| GB0405933D0 (en) | 2004-03-16 | 2004-04-21 | Glaxo Group Ltd | Compounds |
| TWI363759B (en) | 2004-04-27 | 2012-05-11 | Glaxo Group Ltd | Muscarinic acetylcholine receptor antagonists |
| WO2006000401A1 (en) | 2004-06-28 | 2006-01-05 | Glaxo Group Limited | Substituted oxazines as glucocorticoid receptor modulators |
| WO2006000398A1 (en) | 2004-06-28 | 2006-01-05 | Glaxo Group Limited | 2,3-benzoxazin derivatives as non-steroidal glucocorticoid receptor modulators |
| GB0418045D0 (en) | 2004-08-12 | 2004-09-15 | Glaxo Group Ltd | Compounds |
| KR100867071B1 (ko) | 2004-10-19 | 2008-11-04 | 에프. 호프만-라 로슈 아게 | 퀴놀린 유도체 |
| US20090124588A1 (en) | 2005-01-10 | 2009-05-14 | Glaxo Group Limited | Androstane 17-Alpha-Carbonate for Use in the Treatment of Inflammatory and Allergic Conditions |
| ATE517908T1 (de) | 2005-01-10 | 2011-08-15 | Glaxo Group Ltd | Androstan-17-alpha-carbonat-derivate zur verwendung bei der behandlung allergischer und entzündlicher zustände |
| WO2009147187A1 (en) * | 2008-06-05 | 2009-12-10 | Glaxo Group Limited | 4-carboxamide indazole derivatives useful as inhibitors of p13-kinases |
| EP2406255B1 (en) * | 2009-03-09 | 2015-04-29 | Glaxo Group Limited | 4-oxadiazol-2-yl-indazoles as inhibitors of pi3 kinases |
| JO3025B1 (ar) * | 2009-04-30 | 2016-09-05 | Glaxo Group Ltd | الأندازولات المستبدلة بالأوكسازول كمثبطات كيناز pi3 |
| ES2602972T3 (es) * | 2010-09-08 | 2017-02-23 | Glaxosmithkline Intellectual Property Development Limited | Derivados de indazol para su uso en el tratamiento de infección por virus de la gripe |
-
2011
- 2011-09-06 DK DK11755311.5T patent/DK2614058T3/en active
- 2011-09-06 SI SI201130595T patent/SI2614058T1/sl unknown
- 2011-09-06 US US13/821,585 patent/US8735390B2/en active Active
- 2011-09-06 PT PT117553115T patent/PT2614058E/pt unknown
- 2011-09-06 HU HUE11755311A patent/HUE026059T2/en unknown
- 2011-09-06 RS RS20150611A patent/RS54286B1/en unknown
- 2011-09-06 EP EP11755311.5A patent/EP2614058B1/en active Active
- 2011-09-06 JP JP2013527583A patent/JP5965402B2/ja active Active
- 2011-09-06 ES ES11755311.5T patent/ES2548036T3/es active Active
- 2011-09-06 WO PCT/EP2011/065419 patent/WO2012032067A1/en active Application Filing
- 2011-09-06 PL PL11755311T patent/PL2614058T3/pl unknown
-
2015
- 2015-09-22 SM SM201500223T patent/SMT201500223B/xx unknown
- 2015-09-28 HR HRP20151017TT patent/HRP20151017T1/hr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| PL2614058T3 (pl) | 2015-12-31 |
| HUE026059T2 (en) | 2016-05-30 |
| EP2614058B1 (en) | 2015-07-08 |
| JP2013537175A (ja) | 2013-09-30 |
| EP2614058A1 (en) | 2013-07-17 |
| WO2012032067A1 (en) | 2012-03-15 |
| PT2614058E (pt) | 2015-10-27 |
| US8735390B2 (en) | 2014-05-27 |
| JP5965402B2 (ja) | 2016-08-03 |
| DK2614058T3 (en) | 2015-09-28 |
| RS54286B1 (en) | 2016-02-29 |
| HRP20151017T1 (hr) | 2015-10-23 |
| US20130165441A1 (en) | 2013-06-27 |
| ES2548036T3 (es) | 2015-10-13 |
| SI2614058T1 (sl) | 2015-10-30 |
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