SMT201500223B - Polimorfi e sali di n-[5-[4-(5-{[(2R,6S)-2,6-dimetil-4-morfolinil]metil}-1,3-ossazol-2-il)-1H-indazol-6-IL]-2-(metilossi)-3-piridinilÜmetansolfonammide - Google Patents
Polimorfi e sali di n-[5-[4-(5-{[(2R,6S)-2,6-dimetil-4-morfolinil]metil}-1,3-ossazol-2-il)-1H-indazol-6-IL]-2-(metilossi)-3-piridinilÜmetansolfonammideInfo
- Publication number
- SMT201500223B SMT201500223B SM201500223T SM201500223T SMT201500223B SM T201500223 B SMT201500223 B SM T201500223B SM 201500223 T SM201500223 T SM 201500223T SM 201500223 T SM201500223 T SM 201500223T SM T201500223 B SMT201500223 B SM T201500223B
- Authority
- SM
- San Marino
- Prior art keywords
- piridinilümetansolfonammide
- methyloxy
- indazol
- oxazol
- polymorphs
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Epidemiology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US38074810P | 2010-09-08 | 2010-09-08 | |
PCT/EP2011/065419 WO2012032067A1 (en) | 2010-09-08 | 2011-09-06 | Polymorphs and salts of n- [5- [4- (5- { [(2r,6s) -2, 6 - dimethyl - 4 -morpholinyl] methyl} - 1, 3 - oxazol - 2 - yl) - 1h- inda zol-6-yl] -2- (methyloxy) - 3 - pyridinyl] methanesulfonamide |
Publications (1)
Publication Number | Publication Date |
---|---|
SMT201500223B true SMT201500223B (it) | 2015-10-30 |
Family
ID=44645691
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SM201500223T SMT201500223B (it) | 2010-09-08 | 2015-09-22 | Polimorfi e sali di n-[5-[4-(5-{[(2R,6S)-2,6-dimetil-4-morfolinil]metil}-1,3-ossazol-2-il)-1H-indazol-6-IL]-2-(metilossi)-3-piridinilÜmetansolfonammide |
Country Status (13)
Country | Link |
---|---|
US (1) | US8735390B2 (de) |
EP (1) | EP2614058B1 (de) |
JP (1) | JP5965402B2 (de) |
DK (1) | DK2614058T3 (de) |
ES (1) | ES2548036T3 (de) |
HR (1) | HRP20151017T1 (de) |
HU (1) | HUE026059T2 (de) |
PL (1) | PL2614058T3 (de) |
PT (1) | PT2614058E (de) |
RS (1) | RS54286B1 (de) |
SI (1) | SI2614058T1 (de) |
SM (1) | SMT201500223B (de) |
WO (1) | WO2012032067A1 (de) |
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WO2006000398A1 (en) | 2004-06-28 | 2006-01-05 | Glaxo Group Limited | 2,3-benzoxazin derivatives as non-steroidal glucocorticoid receptor modulators |
GB0418045D0 (en) | 2004-08-12 | 2004-09-15 | Glaxo Group Ltd | Compounds |
CN101044135B (zh) | 2004-10-19 | 2011-11-23 | 霍夫曼-拉罗奇有限公司 | 喹啉衍生物 |
WO2006072599A2 (en) | 2005-01-10 | 2006-07-13 | Glaxo Group Limited | Androstane 17-alpha carbonate derivatives for use in the treatment of allergic and inflammatory conditions |
US20090124588A1 (en) | 2005-01-10 | 2009-05-14 | Glaxo Group Limited | Androstane 17-Alpha-Carbonate for Use in the Treatment of Inflammatory and Allergic Conditions |
ES2566339T3 (es) * | 2008-06-05 | 2016-04-12 | Glaxo Group Limited | Derivados de 4-carboxamida indazol útiles como inhibidores de PI3-quinasas |
EP2406255B1 (de) * | 2009-03-09 | 2015-04-29 | Glaxo Group Limited | 4-oxadiazol-2-ylindazole als inhibitoren von pi3-kinasen |
EP2899191B1 (de) | 2009-04-30 | 2017-08-09 | Glaxo Group Limited | Oxazolsubstituierte indazole als pi3-kinaseinhibitoren |
US9326987B2 (en) * | 2010-09-08 | 2016-05-03 | Glaxo Group Limited | Indazole derivatives for use in the treatment of influenza virus infection |
-
2011
- 2011-09-06 EP EP11755311.5A patent/EP2614058B1/de active Active
- 2011-09-06 PL PL11755311T patent/PL2614058T3/pl unknown
- 2011-09-06 SI SI201130595T patent/SI2614058T1/sl unknown
- 2011-09-06 HU HUE11755311A patent/HUE026059T2/en unknown
- 2011-09-06 JP JP2013527583A patent/JP5965402B2/ja active Active
- 2011-09-06 RS RS20150611A patent/RS54286B1/en unknown
- 2011-09-06 ES ES11755311.5T patent/ES2548036T3/es active Active
- 2011-09-06 PT PT117553115T patent/PT2614058E/pt unknown
- 2011-09-06 DK DK11755311.5T patent/DK2614058T3/en active
- 2011-09-06 WO PCT/EP2011/065419 patent/WO2012032067A1/en active Application Filing
- 2011-09-06 US US13/821,585 patent/US8735390B2/en active Active
-
2015
- 2015-09-22 SM SM201500223T patent/SMT201500223B/xx unknown
- 2015-09-28 HR HRP20151017TT patent/HRP20151017T1/hr unknown
Also Published As
Publication number | Publication date |
---|---|
EP2614058B1 (de) | 2015-07-08 |
DK2614058T3 (en) | 2015-09-28 |
ES2548036T3 (es) | 2015-10-13 |
EP2614058A1 (de) | 2013-07-17 |
JP5965402B2 (ja) | 2016-08-03 |
US8735390B2 (en) | 2014-05-27 |
SI2614058T1 (sl) | 2015-10-30 |
JP2013537175A (ja) | 2013-09-30 |
US20130165441A1 (en) | 2013-06-27 |
WO2012032067A1 (en) | 2012-03-15 |
RS54286B1 (en) | 2016-02-29 |
HUE026059T2 (en) | 2016-05-30 |
PL2614058T3 (pl) | 2015-12-31 |
PT2614058E (pt) | 2015-10-27 |
HRP20151017T1 (hr) | 2015-10-23 |
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