SK391891A3 - Xanthine derivatives and pharmaceutical composition comprising same - Google Patents

Xanthine derivatives and pharmaceutical composition comprising same Download PDF

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Publication number
SK391891A3
SK391891A3 SK3918-91A SK391891A SK391891A3 SK 391891 A3 SK391891 A3 SK 391891A3 SK 391891 A SK391891 A SK 391891A SK 391891 A3 SK391891 A3 SK 391891A3
Authority
SK
Slovakia
Prior art keywords
formula
dicyclopropylmethyl
group
compound
xanthine derivatives
Prior art date
Application number
SK3918-91A
Other languages
English (en)
Slovak (sk)
Inventor
Harald Maschler
Barbara Ann Spicer
Harry Smith
Original Assignee
Beecham Wuelfing Gmbh And Co K
Beecham Group Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Beecham Wuelfing Gmbh And Co K, Beecham Group Plc filed Critical Beecham Wuelfing Gmbh And Co K
Publication of SK391891A3 publication Critical patent/SK391891A3/sk

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
    • C07D473/06—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Biomedical Technology (AREA)
  • Cardiology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pulmonology (AREA)
  • Hospice & Palliative Care (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Immunology (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
SK3918-91A 1989-03-23 1991-12-19 Xanthine derivatives and pharmaceutical composition comprising same SK391891A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB898906792A GB8906792D0 (en) 1989-03-23 1989-03-23 Treatment and compounds

Publications (1)

Publication Number Publication Date
SK391891A3 true SK391891A3 (en) 2000-12-11

Family

ID=10653940

Family Applications (1)

Application Number Title Priority Date Filing Date
SK3918-91A SK391891A3 (en) 1989-03-23 1991-12-19 Xanthine derivatives and pharmaceutical composition comprising same

Country Status (27)

Country Link
US (4) US5981535A (de)
EP (2) EP1120417A3 (de)
JP (1) JP2510889B2 (de)
KR (1) KR0160768B1 (de)
CN (1) CN1031641C (de)
AT (1) ATE213498T1 (de)
AU (1) AU629315B2 (de)
CA (1) CA2012686C (de)
CZ (1) CZ391891A3 (de)
DE (1) DE69033915T2 (de)
DK (1) DK0389282T3 (de)
ES (1) ES2173074T3 (de)
FI (1) FI95033C (de)
GB (1) GB8906792D0 (de)
HK (1) HK1040392A1 (de)
HU (1) HU207081B (de)
IL (1) IL93832A (de)
MA (1) MA21800A1 (de)
MY (1) MY109737A (de)
NO (1) NO175592C (de)
NZ (1) NZ233021A (de)
PL (1) PL164811B1 (de)
PT (1) PT93527B (de)
SA (1) SA90100215B1 (de)
SK (1) SK391891A3 (de)
ZA (1) ZA902170B (de)
ZW (1) ZW3690A1 (de)

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Also Published As

Publication number Publication date
US5734051A (en) 1998-03-31
US6531600B1 (en) 2003-03-11
ZW3690A1 (en) 1991-02-06
MA21800A1 (fr) 1990-12-31
NO901300L (no) 1990-09-24
IL93832A0 (en) 1990-12-23
CN1047502A (zh) 1990-12-05
CZ391891A3 (en) 1993-11-17
FI95033C (fi) 1995-12-11
KR0160768B1 (ko) 1998-12-01
FI95033B (fi) 1995-08-31
EP1120417A3 (de) 2001-08-08
JP2510889B2 (ja) 1996-06-26
NO175592B (no) 1994-07-25
ZA902170B (en) 1991-03-27
EP0389282B1 (de) 2002-02-20
AU5208390A (en) 1990-09-27
HUT54155A (en) 1991-01-28
PT93527A (pt) 1990-11-07
DE69033915D1 (de) 2002-03-28
PL164811B1 (pl) 1994-10-31
IL93832A (en) 1994-07-31
HU207081B (en) 1993-03-01
CA2012686A1 (en) 1990-09-23
ATE213498T1 (de) 2002-03-15
DK0389282T3 (da) 2002-06-03
JPH02273676A (ja) 1990-11-08
NO175592C (no) 1994-11-02
US5981535A (en) 1999-11-09
SA90100215B1 (ar) 2001-10-07
NO901300D0 (no) 1990-03-21
EP1120417A2 (de) 2001-08-01
ES2173074T3 (es) 2002-10-16
DE69033915T2 (de) 2002-10-10
US6180791B1 (en) 2001-01-30
AU629315B2 (en) 1992-10-01
EP0389282A2 (de) 1990-09-26
CA2012686C (en) 1999-12-07
FI901447A0 (fi) 1990-03-22
NZ233021A (en) 1993-12-23
GB8906792D0 (en) 1989-05-10
HU901792D0 (en) 1990-06-28
HK1040392A1 (zh) 2002-06-07
EP0389282A3 (de) 1992-07-01
MY109737A (en) 1997-05-31
KR900013962A (ko) 1990-10-22
CN1031641C (zh) 1996-04-24
PT93527B (pt) 1996-08-30

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