SK3852001A3 - 4-Aminopyrrolopyrimidines as kinase inhibitors - Google Patents
4-Aminopyrrolopyrimidines as kinase inhibitors Download PDFInfo
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- SK3852001A3 SK3852001A3 SK385-2001A SK3852001A SK3852001A3 SK 3852001 A3 SK3852001 A3 SK 3852001A3 SK 3852001 A SK3852001 A SK 3852001A SK 3852001 A3 SK3852001 A3 SK 3852001A3
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- unsubstituted
- amino
- pyrrolo
- cyclopentyl
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- QORWJWZARLRLPR-UHFFFAOYSA-H tricalcium bis(phosphate) Chemical compound [Ca+2].[Ca+2].[Ca+2].[O-]P([O-])([O-])=O.[O-]P([O-])([O-])=O QORWJWZARLRLPR-UHFFFAOYSA-H 0.000 description 1
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Classifications
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
- C07F9/44—Amides thereof
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
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- A—HUMAN NECESSITIES
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- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Rheumatology (AREA)
- Emergency Medicine (AREA)
- Pulmonology (AREA)
- Obesity (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
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- Orthopedic Medicine & Surgery (AREA)
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- Hematology (AREA)
- Reproductive Health (AREA)
- Dermatology (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
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US10095498P | 1998-09-18 | 1998-09-18 | |
PCT/US1999/021536 WO2000017202A1 (fr) | 1998-09-18 | 1999-09-17 | 4-aminopyrrolopyrimidines utilisees comme inhibiteurs de kinases |
Publications (1)
Publication Number | Publication Date |
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SK3852001A3 true SK3852001A3 (en) | 2003-03-04 |
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Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
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SK385-2001A SK3852001A3 (en) | 1998-09-18 | 1999-09-17 | 4-Aminopyrrolopyrimidines as kinase inhibitors |
Country Status (22)
Country | Link |
---|---|
EP (1) | EP1114052B1 (fr) |
JP (1) | JP2002527359A (fr) |
KR (1) | KR20010085822A (fr) |
CN (1) | CN1326457A (fr) |
AT (1) | ATE310001T1 (fr) |
AU (1) | AU752474B2 (fr) |
BR (1) | BR9913888A (fr) |
CA (1) | CA2344262A1 (fr) |
CZ (1) | CZ2001959A3 (fr) |
DE (1) | DE69928414T2 (fr) |
ES (1) | ES2253930T3 (fr) |
HK (1) | HK1039325B (fr) |
HU (1) | HUP0200355A3 (fr) |
ID (1) | ID28362A (fr) |
IL (1) | IL141867A0 (fr) |
NO (1) | NO20011357L (fr) |
NZ (1) | NZ510587A (fr) |
PL (1) | PL347138A1 (fr) |
SK (1) | SK3852001A3 (fr) |
TR (1) | TR200101395T2 (fr) |
WO (1) | WO2000017202A1 (fr) |
ZA (1) | ZA200102201B (fr) |
Families Citing this family (138)
Publication number | Priority date | Publication date | Assignee | Title |
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US20030130209A1 (en) * | 1999-12-22 | 2003-07-10 | Cheresh David A. | Method of treatment of myocardial infarction |
EP1107958B1 (fr) | 1998-08-29 | 2006-08-16 | AstraZeneca AB | Composes pyrimidiniques |
JP2002523497A (ja) | 1998-08-29 | 2002-07-30 | アストラゼネカ・アクチエボラーグ | ピリミジン化合物 |
US6713474B2 (en) | 1998-09-18 | 2004-03-30 | Abbott Gmbh & Co. Kg | Pyrrolopyrimidines as therapeutic agents |
GB9828511D0 (en) | 1998-12-24 | 1999-02-17 | Zeneca Ltd | Chemical compounds |
GB9905075D0 (en) | 1999-03-06 | 1999-04-28 | Zeneca Ltd | Chemical compounds |
GB9907658D0 (en) | 1999-04-06 | 1999-05-26 | Zeneca Ltd | Chemical compounds |
US7041691B1 (en) | 1999-06-30 | 2006-05-09 | Amgen Inc. | Compounds for the modulation of PPARγ activity |
GB9919778D0 (en) | 1999-08-21 | 1999-10-27 | Zeneca Ltd | Chemical compounds |
SK288019B6 (sk) | 1999-12-24 | 2012-11-05 | Aventis Pharma Limited | Azaindoles derivatives, their use and pharmaceutical composition containing thereof |
GB0004888D0 (en) | 2000-03-01 | 2000-04-19 | Astrazeneca Uk Ltd | Chemical compounds |
GB0004890D0 (en) | 2000-03-01 | 2000-04-19 | Astrazeneca Uk Ltd | Chemical compounds |
GB0004887D0 (en) | 2000-03-01 | 2000-04-19 | Astrazeneca Uk Ltd | Chemical compounds |
GB0004886D0 (en) | 2000-03-01 | 2000-04-19 | Astrazeneca Uk Ltd | Chemical compounds |
GB0007371D0 (en) | 2000-03-28 | 2000-05-17 | Astrazeneca Uk Ltd | Chemical compounds |
WO2001072751A1 (fr) * | 2000-03-29 | 2001-10-04 | Knoll Gesellschaft Mit Beschraenkter Haftung | Pyrrolopyrimidines utilisees comme inhibiteurs de tyrosine kinases |
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GB9604361D0 (en) * | 1996-02-29 | 1996-05-01 | Pharmacia Spa | 4-Substituted pyrrolopyrimidine compounds as tyrosine kinase inhibitors |
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- 1999-09-17 TR TR2001/01395T patent/TR200101395T2/xx unknown
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- 1999-09-17 WO PCT/US1999/021536 patent/WO2000017202A1/fr not_active Application Discontinuation
- 1999-09-17 CZ CZ2001959A patent/CZ2001959A3/cs unknown
- 1999-09-17 SK SK385-2001A patent/SK3852001A3/sk unknown
- 1999-09-17 EP EP99969414A patent/EP1114052B1/fr not_active Expired - Lifetime
- 1999-09-17 JP JP2000574111A patent/JP2002527359A/ja active Pending
- 1999-09-17 AU AU60475/99A patent/AU752474B2/en not_active Ceased
- 1999-09-17 BR BR9913888-3A patent/BR9913888A/pt not_active IP Right Cessation
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- 1999-09-17 CA CA002344262A patent/CA2344262A1/fr not_active Abandoned
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HUP0200355A3 (en) | 2004-07-28 |
CZ2001959A3 (cs) | 2001-12-12 |
AU752474B2 (en) | 2002-09-19 |
AU6047599A (en) | 2000-04-10 |
ATE310001T1 (de) | 2005-12-15 |
NZ510587A (en) | 2003-11-28 |
NO20011357L (no) | 2001-05-14 |
ZA200102201B (en) | 2002-03-15 |
EP1114052A1 (fr) | 2001-07-11 |
HK1039325A1 (en) | 2002-04-19 |
CA2344262A1 (fr) | 2000-03-30 |
DE69928414D1 (de) | 2005-12-22 |
JP2002527359A (ja) | 2002-08-27 |
EP1114052B1 (fr) | 2005-11-16 |
DE69928414T2 (de) | 2006-08-03 |
NO20011357D0 (no) | 2001-03-16 |
PL347138A1 (en) | 2002-03-25 |
WO2000017202A1 (fr) | 2000-03-30 |
HUP0200355A2 (en) | 2002-06-29 |
BR9913888A (pt) | 2002-01-08 |
HK1039325B (zh) | 2006-02-24 |
CN1326457A (zh) | 2001-12-12 |
TR200101395T2 (tr) | 2001-11-21 |
IL141867A0 (en) | 2002-03-10 |
ES2253930T3 (es) | 2006-06-01 |
ID28362A (id) | 2001-05-17 |
KR20010085822A (ko) | 2001-09-07 |
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