SK286690B6 - Androstdiény, ich použitie, farmaceutická kompozícia s ich obsahom, spôsob ich prípravy a medziprodukty - Google Patents
Androstdiény, ich použitie, farmaceutická kompozícia s ich obsahom, spôsob ich prípravy a medziprodukty Download PDFInfo
- Publication number
- SK286690B6 SK286690B6 SK1813-2002A SK18132002A SK286690B6 SK 286690 B6 SK286690 B6 SK 286690B6 SK 18132002 A SK18132002 A SK 18132002A SK 286690 B6 SK286690 B6 SK 286690B6
- Authority
- SK
- Slovakia
- Prior art keywords
- group
- carbon atoms
- methyl
- alkyl
- formula
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0038—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 with an androstane skeleton, including 18- or 19-substituted derivatives, 18-nor derivatives and also derivatives where position 17-beta is substituted by a carbon atom not directly bonded to a further carbon atom and not being part of an amide group
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J3/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J17/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J3/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
- C07J3/005—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom the carbon atom being part of a carboxylic function
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J33/00—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J33/002—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0094—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 containing nitrile radicals, including thiocyanide radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0005—Oxygen-containing hetero ring
- C07J71/001—Oxiranes
- C07J71/0015—Oxiranes at position 9(11)
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pulmonology (AREA)
- Toxicology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0015876.6A GB0015876D0 (en) | 2000-06-28 | 2000-06-28 | Organic compounds |
PCT/EP2001/007249 WO2002000679A2 (fr) | 2000-06-28 | 2001-06-26 | Composes organiques |
Publications (2)
Publication Number | Publication Date |
---|---|
SK18132002A3 SK18132002A3 (sk) | 2003-08-05 |
SK286690B6 true SK286690B6 (sk) | 2009-03-05 |
Family
ID=9894607
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SK1813-2002A SK286690B6 (sk) | 2000-06-28 | 2001-06-26 | Androstdiény, ich použitie, farmaceutická kompozícia s ich obsahom, spôsob ich prípravy a medziprodukty |
Country Status (30)
Country | Link |
---|---|
US (1) | US6921757B2 (fr) |
EP (1) | EP1299409B1 (fr) |
JP (1) | JP4065399B2 (fr) |
KR (1) | KR100483865B1 (fr) |
CN (1) | CN1214038C (fr) |
AR (1) | AR030707A1 (fr) |
AT (1) | ATE292639T1 (fr) |
AU (2) | AU8389101A (fr) |
BR (1) | BR0112068A (fr) |
CA (1) | CA2412541C (fr) |
CZ (1) | CZ302513B6 (fr) |
DE (1) | DE60109931T2 (fr) |
EC (1) | ECSP014101A (fr) |
ES (1) | ES2240499T3 (fr) |
GB (1) | GB0015876D0 (fr) |
HK (1) | HK1055974A1 (fr) |
HU (1) | HUP0300783A3 (fr) |
IL (2) | IL153703A0 (fr) |
MX (1) | MXPA02012830A (fr) |
MY (1) | MY129523A (fr) |
NO (1) | NO324055B1 (fr) |
NZ (1) | NZ523194A (fr) |
PE (1) | PE20020179A1 (fr) |
PL (1) | PL207722B1 (fr) |
PT (1) | PT1299409E (fr) |
RU (1) | RU2277100C2 (fr) |
SK (1) | SK286690B6 (fr) |
TW (1) | TWI232868B (fr) |
WO (1) | WO2002000679A2 (fr) |
ZA (1) | ZA200300202B (fr) |
Families Citing this family (111)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AR028948A1 (es) | 2000-06-20 | 2003-05-28 | Astrazeneca Ab | Compuestos novedosos |
US6858593B2 (en) | 2000-08-05 | 2005-02-22 | Smithkline Beecham Corporation | Anti-inflammatory androstane derivative compositions |
US6777400B2 (en) | 2000-08-05 | 2004-08-17 | Smithkline Beecham Corporation | Anti-inflammatory androstane derivative compositions |
US6759398B2 (en) * | 2000-08-05 | 2004-07-06 | Smithkline Beecham Corporation | Anti-inflammatory androstane derivative |
US6750210B2 (en) | 2000-08-05 | 2004-06-15 | Smithkline Beecham Corporation | Formulation containing novel anti-inflammatory androstane derivative |
US6858596B2 (en) * | 2000-08-05 | 2005-02-22 | Smithkline Beecham Corporation | Formulation containing anti-inflammatory androstane derivative |
US6787532B2 (en) | 2000-08-05 | 2004-09-07 | Smithkline Beecham Corporation | Formulation containing anti-inflammatory androstane derivatives |
US6777399B2 (en) * | 2000-08-05 | 2004-08-17 | Smithkline Beecham Corporation | Anti-inflammatory androstane derivative compositions |
AU7576001A (en) * | 2000-08-05 | 2002-02-18 | Glaxo Group Ltd | 6.alpha., 9.alpha.-difluoro-17.alpha.-`(2-furanylcarboxyl) oxy]-11.beta.-hydroxy-16.alpha.-methyl-3-oxo-androst-1,4,-diene-17-carbothioic acid s-fluoromethyl ester as an anti-inflammatory agent |
GB0019172D0 (en) | 2000-08-05 | 2000-09-27 | Glaxo Group Ltd | Novel compounds |
UA77656C2 (en) | 2001-04-07 | 2007-01-15 | Glaxo Group Ltd | S-fluoromethyl ester of 6-alpha, 9-alpha-difluoro-17-alpha-[(2-furanylcarbonyl)oxy]-11-beta-hydroxy-16- alpha-methyl-3-oxoandrosta-1,4-dien-17-beta-carbothioacid as anti-inflammatory agent |
EP1383786B1 (fr) * | 2001-04-30 | 2008-10-15 | Glaxo Group Limited | Derives anti-inflammatoires d'androstane 17.beta.-carbothioate ester avec un groupe cyclique en position 17.alpha |
DE60227254D1 (de) * | 2001-06-12 | 2008-08-07 | Glaxo Group Ltd | Neue anti inflammatorische 17.alpha.-heterozyklische ester von 17.beta.-carbothioat androstan derivativen |
GB0125259D0 (en) * | 2001-10-20 | 2001-12-12 | Glaxo Group Ltd | Novel compounds |
WO2003042229A1 (fr) * | 2001-11-12 | 2003-05-22 | Glaxo Group Limited | Esters heterocycliques non aromatiques de furan-2-one esters de 17 $g(b) carboxyl ou 17 $g(b) carbothio glucocorticoides |
GB0127160D0 (en) * | 2001-11-12 | 2002-01-02 | Glaxo Group Ltd | Novel compounds |
WO2003048181A1 (fr) * | 2001-12-01 | 2003-06-12 | Glaxo Group Limited | 17.alpha.-esters cycliques de 16-methylpregnan-3,20-dione en tant qu'agents anti-inflammatoires |
WO2003072592A1 (fr) * | 2002-01-15 | 2003-09-04 | Glaxo Group Limited | 17 alpha esters cycloalkyle/cycloalcenyle d'alkyle ou haloalkyle-androst-4-en-3-on-11 beta, 17 alpha-diol 17 beta-carboxylates comme agents anti-inflammatoires |
WO2003062259A2 (fr) * | 2002-01-21 | 2003-07-31 | Glaxo Group Limited | Nouveaux composes |
GB0202216D0 (en) * | 2002-01-31 | 2002-03-20 | Glaxo Group Ltd | Novel compounds |
AU2003244451A1 (en) * | 2002-02-04 | 2003-09-02 | Glaxo Group Limited | Amorphous fluticasone 2-furoate, pharmaceutical compositions thereof and its conversion to the crystalline unsolvated form |
US20050175545A1 (en) * | 2002-02-04 | 2005-08-11 | Keith Biggadike | Formulation for inhalation comprising a glucocorticoid and a beta 2-adrenoreceptor agonist |
GB0202635D0 (en) * | 2002-02-05 | 2002-03-20 | Glaxo Wellcome Mfg Pte Ltd | Formulation containing novel anti-inflammatory androstane derivative |
GB2389530B (en) | 2002-06-14 | 2007-01-10 | Cipla Ltd | Pharmaceutical compositions |
GB0217504D0 (en) * | 2002-07-29 | 2002-09-04 | Novartis Ag | Organic compounds |
WO2004071383A2 (fr) * | 2003-02-11 | 2004-08-26 | Boehringer Ingelheim International Gmbh | Nouvelles compositions pharmaceutiques a base d'anticholinergiques et d'inhibiteurs de la synthese ou de l'activite du facteur de necrose des tumeurs alpha |
TW200519106A (en) | 2003-05-02 | 2005-06-16 | Novartis Ag | Organic compounds |
GB0316290D0 (en) * | 2003-07-11 | 2003-08-13 | Glaxo Group Ltd | Novel compounds |
GB0401334D0 (en) | 2004-01-21 | 2004-02-25 | Novartis Ag | Organic compounds |
US7507745B2 (en) | 2004-02-20 | 2009-03-24 | Boehringer Ingelheim International Gmbh | Pharmaceutical compositions based on fluorenecarboxylic acid esters and soluble TNF receptor fusion proteins |
US8182792B2 (en) | 2004-03-23 | 2012-05-22 | Novartis Ag | Pharmaceutical compositions |
GB0410712D0 (en) | 2004-05-13 | 2004-06-16 | Novartis Ag | Organic compounds |
GB0411056D0 (en) | 2004-05-18 | 2004-06-23 | Novartis Ag | Organic compounds |
DE102004025985A1 (de) * | 2004-05-21 | 2005-12-15 | Schering Ag | Estriol- und Estetrol-Prodrugs |
DE102004025966A1 (de) * | 2004-05-21 | 2005-12-15 | Schering Ag | Estradiol-Prodrugs |
GT200500281A (es) | 2004-10-22 | 2006-04-24 | Novartis Ag | Compuestos organicos. |
GB0424284D0 (en) | 2004-11-02 | 2004-12-01 | Novartis Ag | Organic compounds |
GB0426164D0 (en) | 2004-11-29 | 2004-12-29 | Novartis Ag | Organic compounds |
ATE517908T1 (de) | 2005-01-10 | 2011-08-15 | Glaxo Group Ltd | Androstan-17-alpha-carbonat-derivate zur verwendung bei der behandlung allergischer und entzündlicher zustände |
GB0507165D0 (en) * | 2005-04-08 | 2005-05-18 | Glaxo Group Ltd | Novel crystalline pharmaceutical product |
GB0507577D0 (en) | 2005-04-14 | 2005-05-18 | Novartis Ag | Organic compounds |
GB0510390D0 (en) | 2005-05-20 | 2005-06-29 | Novartis Ag | Organic compounds |
TW200738634A (en) | 2005-08-02 | 2007-10-16 | Astrazeneca Ab | New salt |
CA2618089A1 (fr) | 2005-08-08 | 2007-02-15 | Argenta Discovery Ltd. | Derives bicyclo[2,2]hept-7-ylamine et leurs utilisations |
GB0516313D0 (en) | 2005-08-08 | 2005-09-14 | Argenta Discovery Ltd | Azole derivatives and their uses |
EP2532679B1 (fr) | 2005-10-21 | 2017-04-12 | Novartis AG | Anticorps humains dirigés contre l'IL -13 et utilisations thérapeutiques |
GB0523656D0 (en) * | 2005-11-21 | 2005-12-28 | Novartis Ag | Organic compounds |
GB0523654D0 (en) * | 2005-11-21 | 2005-12-28 | Novartis Ag | Organic compounds |
GB0526244D0 (en) | 2005-12-22 | 2006-02-01 | Novartis Ag | Organic compounds |
GB0601951D0 (en) | 2006-01-31 | 2006-03-15 | Novartis Ag | Organic compounds |
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EP1894568A1 (fr) * | 2006-08-31 | 2008-03-05 | Novartis AG | Composées pharmaceutiques destinées au traitement des maladies inflammatoires ou obstructives des bronches |
ATE502943T1 (de) | 2006-09-29 | 2011-04-15 | Novartis Ag | Pyrazolopyrimidine als pi3k-lipidkinasehemmer |
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KR20090094460A (ko) | 2006-12-19 | 2009-09-07 | 아스트라제네카 아베 | 무스카린 수용체 길항제로서 퀴누클리디놀 유도체 |
DE602007011670D1 (de) | 2007-01-10 | 2011-02-10 | Irm Llc | Verbindungen und zusammensetzungen als kanal-aktivierende proteasehemmer |
EP2117541A1 (fr) | 2007-02-09 | 2009-11-18 | Irm Llc | Composés et compositions en tant qu'inhibiteurs de la protéase activatrice de canaux |
EA200901489A1 (ru) | 2007-05-07 | 2010-04-30 | Новартис Аг | Органические соединения |
AU2008334629B2 (en) | 2007-12-10 | 2012-04-12 | Novartis Ag | Organic compounds |
WO2009087224A1 (fr) | 2008-01-11 | 2009-07-16 | Novartis Ag | Pyrimidines utilisés en tant qu'inhibiteurs de kinase |
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EP2300010B1 (fr) | 2008-06-10 | 2015-03-04 | Novartis AG | Dérivés de pyrazine en tant que bloqueur du canal sodique epithelial |
WO2010067102A1 (fr) | 2008-12-09 | 2010-06-17 | Astrazeneca Ab | Dérivés de diazaspiro[5.5]undécane et composés associés utilisés comme antagonistes des récepteurs muscariniques et agonistes des récepteurs bêta adrénergiques dans le traitement des affections pulmonaires |
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IN2012DN01453A (fr) | 2009-08-20 | 2015-06-05 | Novartis Ag | |
CA2777245A1 (fr) | 2009-10-22 | 2011-04-28 | Vertex Pharmaceuticals Incorporated | Compositions destinees au traitement de la mucoviscidose et d'autres maladies chroniques |
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US8247436B2 (en) | 2010-03-19 | 2012-08-21 | Novartis Ag | Pyridine and pyrazine derivative for the treatment of CF |
UY33597A (es) | 2010-09-09 | 2012-04-30 | Irm Llc | Compuestos y composiciones como inhibidores de la trk |
WO2012034095A1 (fr) | 2010-09-09 | 2012-03-15 | Irm Llc | Composés et compositions comme inhibiteurs de trk |
US8372845B2 (en) | 2010-09-17 | 2013-02-12 | Novartis Ag | Pyrazine derivatives as enac blockers |
EP2673277A1 (fr) | 2011-02-10 | 2013-12-18 | Novartis AG | Composés de [1, 2, 4]triazolo [4, 3 -b]pyridazine en tant qu'inhibiteurs de la tyrosine kinase c-met |
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WO2012116217A1 (fr) | 2011-02-25 | 2012-08-30 | Irm Llc | Composés et compositions en tant qu'inhibiteurs de trk |
US8883819B2 (en) | 2011-09-01 | 2014-11-11 | Irm Llc | Bicyclic heterocycle derivatives for the treatment of pulmonary arterial hypertension |
EP2755976B1 (fr) | 2011-09-15 | 2018-07-18 | Novartis AG | 3-(quinolin-6-ylthio)-[1,2,4]triazolo[4,3-a]pyradines substituées en position 6 à activité tyrosine kinase |
WO2013038378A1 (fr) | 2011-09-16 | 2013-03-21 | Novartis Ag | Dérivés pyridinamides |
EP2755967B1 (fr) | 2011-09-16 | 2015-10-21 | Novartis AG | Composés hétérocycliques destinés au traitement de la mucosviscidose |
WO2013038373A1 (fr) | 2011-09-16 | 2013-03-21 | Novartis Ag | Dérivés pyrimidinamides |
WO2013038390A1 (fr) | 2011-09-16 | 2013-03-21 | Novartis Ag | Hétérocyclyle carboxamides n-substitués |
WO2013038381A1 (fr) | 2011-09-16 | 2013-03-21 | Novartis Ag | Dérivés d'amide pyridine/pyrazine |
EP2793893A4 (fr) | 2011-11-23 | 2015-07-08 | Intellikine Llc | Régimes de traitement améliorés utilisant des inhibiteurs de mtor |
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CN104245701A (zh) | 2012-04-03 | 2014-12-24 | 诺华有限公司 | 有酪氨酸激酶抑制剂的组合产品和其应用 |
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WO2014151147A1 (fr) | 2013-03-15 | 2014-09-25 | Intellikine, Llc | Combinaison d'inhibiteurs de kinase et ses utilisations |
EP3007697B1 (fr) | 2013-06-14 | 2020-09-02 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Inhibiteurs du rac1 permettant d'induire la bronchodilatation |
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BR112016024533A8 (pt) | 2014-04-24 | 2021-03-30 | Novartis Ag | derivados de amino pirazina como inibidores de fosfatidilinositol 3-cinase ou sal, seu uso, e composição e combinação farmacêuticas |
WO2016011658A1 (fr) | 2014-07-25 | 2016-01-28 | Novartis Ag | Polythérapie |
AU2015294889B2 (en) | 2014-07-31 | 2018-03-15 | Novartis Ag | Combination therapy |
EP3703065A1 (fr) | 2015-01-20 | 2020-09-02 | Novartis AG | Déverrouillage d'application au moyen d'un dispositif physique, et transfert de données entre ces éléments |
PL3111978T3 (pl) | 2015-07-03 | 2022-01-24 | Novartis Ag | Inhalator przystosowany do odczytu informacji przechowywanych w środkach przechowywania danych pojemnika |
CN108129537B (zh) * | 2017-12-19 | 2022-03-01 | 广州健康元呼吸药物工程技术有限公司 | 一种糖皮质激素异构体及其制备方法和用途 |
WO2020250116A1 (fr) | 2019-06-10 | 2020-12-17 | Novartis Ag | Dérivé de pyridine et de pyrazine pour le traitement de la fk, de la bpco et de la bronchiectasie |
US20220306617A1 (en) | 2019-08-28 | 2022-09-29 | Novartis Ag | Substituted 1,3-phenyl heteroaryl derivatives and their use in the treatment of disease |
TW202140550A (zh) | 2020-01-29 | 2021-11-01 | 瑞士商諾華公司 | 使用抗tslp抗體治療炎性或阻塞性氣道疾病之方法 |
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US3639434A (en) * | 1967-02-02 | 1972-02-01 | Boots Pure Drug Co Ltd | 17-acyloxysteroids and their manufacture |
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GB1438940A (en) * | 1972-07-19 | 1976-06-09 | Glaxo Lab Ltd | 17beta-haloalkoxycarbonyl-17alpha-oxysteroids |
NL7502252A (nl) * | 1974-02-27 | 1975-08-29 | Pierrel Spa | Werkwijze voor het bereiden van een geneesmid- del met anti-inflammatoire werking, gevormd ge- neesmiddel verkregen volgens deze werkwijze alsmede werkwijze voor het bereiden van in het geneesmiddel gebruikte nieuwe steroiden. |
CH628355A5 (de) * | 1976-02-24 | 1982-02-26 | Ciba Geigy Ag | Verfahren zur herstellung neuer androstadien-17beta-carbonsaeuren und ihrer ester und salze. |
ATE8790T1 (de) * | 1981-02-02 | 1984-08-15 | Schering Corporation | Aromatische heterocyclische steroidester, verfahren zu ihrer herstellung und pharmazeutische zusammensetzungen, die sie enthalten. |
US4607028A (en) * | 1983-08-18 | 1986-08-19 | Ciba-Geigy Corporation | Novel carboxylic acid esters |
PE44995A1 (es) | 1994-01-27 | 1995-12-18 | Schering Corp | Furoato de mometasona para el tratamiento de las enfermedades pulmonares y de las vias respiratorias |
JPH08291073A (ja) * | 1995-04-22 | 1996-11-05 | Kissei Pharmaceut Co Ltd | 医薬品組成物及びその製造方法 |
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2000
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2001
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- 2001-06-26 KR KR10-2002-7017949A patent/KR100483865B1/ko not_active IP Right Cessation
- 2001-06-26 EP EP01962783A patent/EP1299409B1/fr not_active Expired - Lifetime
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- 2001-06-26 AT AT01962783T patent/ATE292639T1/de active
- 2001-06-26 PE PE2001000620A patent/PE20020179A1/es not_active Application Discontinuation
- 2001-06-26 BR BR0112068-9A patent/BR0112068A/pt not_active IP Right Cessation
- 2001-06-26 WO PCT/EP2001/007249 patent/WO2002000679A2/fr active IP Right Grant
- 2001-06-26 CZ CZ20024203A patent/CZ302513B6/cs not_active IP Right Cessation
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MM4A | Patent lapsed due to non-payment of maintenance fees |
Effective date: 20140626 |