SK286473B6 - Farmaceutická kompozícia s predĺženým uvoľňovanímalebo dvojitým režimom uvoľňovania obsahujúca inhibítor cGMP PDE-5, spôsob jej prípravy a použitie inhibítora cGMP PDE-5 - Google Patents

Farmaceutická kompozícia s predĺženým uvoľňovanímalebo dvojitým režimom uvoľňovania obsahujúca inhibítor cGMP PDE-5, spôsob jej prípravy a použitie inhibítora cGMP PDE-5 Download PDF

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Publication number
SK286473B6
SK286473B6 SK519-2001A SK5192001A SK286473B6 SK 286473 B6 SK286473 B6 SK 286473B6 SK 5192001 A SK5192001 A SK 5192001A SK 286473 B6 SK286473 B6 SK 286473B6
Authority
SK
Slovakia
Prior art keywords
inhibitor
cgmp pde
pharmaceutical composition
release
composition according
Prior art date
Application number
SK519-2001A
Other languages
English (en)
Slovak (sk)
Other versions
SK5192001A3 (en
Inventor
Elizabeth King
Ross James Macrae
Original Assignee
Pfizer Ireland Pharmaceuticals
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27269526&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SK286473(B6) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GBGB9823192.1A external-priority patent/GB9823192D0/en
Priority claimed from GBGB9825117.6A external-priority patent/GB9825117D0/en
Priority claimed from GBGB9826392.4A external-priority patent/GB9826392D0/en
Application filed by Pfizer Ireland Pharmaceuticals filed Critical Pfizer Ireland Pharmaceuticals
Publication of SK5192001A3 publication Critical patent/SK5192001A3/sk
Publication of SK286473B6 publication Critical patent/SK286473B6/sk

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846Poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Neurosurgery (AREA)
  • Gynecology & Obstetrics (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
SK519-2001A 1998-10-23 1999-10-04 Farmaceutická kompozícia s predĺženým uvoľňovanímalebo dvojitým režimom uvoľňovania obsahujúca inhibítor cGMP PDE-5, spôsob jej prípravy a použitie inhibítora cGMP PDE-5 SK286473B6 (sk)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GBGB9823192.1A GB9823192D0 (en) 1998-10-23 1998-10-23 Pharmaceutical formulations
GBGB9825117.6A GB9825117D0 (en) 1998-11-16 1998-11-16 Pharmaceutical formulations
GBGB9826392.4A GB9826392D0 (en) 1998-11-27 1998-11-27 Pharmaceutical formulations
PCT/IB1999/001619 WO2000024383A1 (fr) 1998-10-23 1999-10-04 Formulations pharmaceutiques a liberation controlee contenant un inhibiteur de pde-5 de cgmp

Publications (2)

Publication Number Publication Date
SK5192001A3 SK5192001A3 (en) 2002-09-10
SK286473B6 true SK286473B6 (sk) 2008-11-06

Family

ID=27269526

Family Applications (1)

Application Number Title Priority Date Filing Date
SK519-2001A SK286473B6 (sk) 1998-10-23 1999-10-04 Farmaceutická kompozícia s predĺženým uvoľňovanímalebo dvojitým režimom uvoľňovania obsahujúca inhibítor cGMP PDE-5, spôsob jej prípravy a použitie inhibítora cGMP PDE-5

Country Status (44)

Country Link
US (1) US6964780B1 (fr)
EP (1) EP1123088B1 (fr)
JP (1) JP2002528408A (fr)
KR (1) KR20010075659A (fr)
CN (1) CN1324233A (fr)
AP (1) AP2001002125A0 (fr)
AT (1) ATE340562T1 (fr)
AU (1) AU756509B2 (fr)
BG (1) BG65323B1 (fr)
BR (1) BR9914718A (fr)
CA (1) CA2348086C (fr)
CO (1) CO5160262A1 (fr)
CR (1) CR6326A (fr)
CY (1) CY1106239T1 (fr)
CZ (1) CZ20011427A3 (fr)
DE (1) DE69933383T2 (fr)
DK (1) DK1123088T3 (fr)
DZ (1) DZ2923A1 (fr)
EA (1) EA004068B1 (fr)
EE (1) EE200100235A (fr)
ES (1) ES2272082T3 (fr)
GT (1) GT199900184A (fr)
HK (1) HK1041818A1 (fr)
HR (1) HRP20010285A2 (fr)
HU (1) HUP0104318A3 (fr)
ID (1) ID28232A (fr)
IL (1) IL141764A (fr)
IS (1) IS5865A (fr)
MA (1) MA26700A1 (fr)
MX (1) MXPA01004011A (fr)
MY (1) MY130727A (fr)
NO (1) NO20011933L (fr)
NZ (1) NZ510275A (fr)
OA (1) OA11664A (fr)
PA (1) PA8484301A1 (fr)
PE (1) PE20001286A1 (fr)
PL (1) PL195789B1 (fr)
PT (1) PT1123088E (fr)
SK (1) SK286473B6 (fr)
TR (1) TR200101103T2 (fr)
TW (1) TW577756B (fr)
UA (1) UA67802C2 (fr)
UY (1) UY25765A1 (fr)
WO (1) WO2000024383A1 (fr)

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Also Published As

Publication number Publication date
HK1041818A1 (zh) 2002-07-26
AU756509B2 (en) 2003-01-16
SK5192001A3 (en) 2002-09-10
KR20010075659A (ko) 2001-08-09
US6964780B1 (en) 2005-11-15
EA200100298A1 (ru) 2001-08-27
JP2002528408A (ja) 2002-09-03
BR9914718A (pt) 2001-07-10
DZ2923A1 (fr) 2004-03-01
PL195789B1 (pl) 2007-10-31
CO5160262A1 (es) 2002-05-30
BG105465A (bg) 2001-12-29
CR6326A (es) 2004-02-23
AP2001002125A0 (en) 2001-04-04
EA004068B1 (ru) 2003-12-25
HRP20010285A2 (en) 2002-06-30
PE20001286A1 (es) 2000-11-22
CY1106239T1 (el) 2011-06-08
IS5865A (is) 2001-02-27
DE69933383D1 (de) 2006-11-09
OA11664A (en) 2005-01-07
DK1123088T3 (da) 2007-01-02
UY25765A1 (es) 2001-08-27
AU5878799A (en) 2000-05-15
NO20011933D0 (no) 2001-04-19
NZ510275A (en) 2003-07-25
MA26700A1 (fr) 2004-12-20
HUP0104318A3 (en) 2003-12-29
EE200100235A (et) 2002-08-15
WO2000024383A1 (fr) 2000-05-04
CZ20011427A3 (cs) 2001-10-17
BG65323B1 (bg) 2008-02-29
UA67802C2 (uk) 2004-07-15
CA2348086C (fr) 2007-01-23
CA2348086A1 (fr) 2000-05-04
ATE340562T1 (de) 2006-10-15
TR200101103T2 (tr) 2001-09-21
EP1123088A1 (fr) 2001-08-16
PT1123088E (pt) 2007-01-31
EP1123088B1 (fr) 2006-09-27
CN1324233A (zh) 2001-11-28
PA8484301A1 (es) 2000-09-29
DE69933383T2 (de) 2007-02-01
HUP0104318A2 (hu) 2002-03-28
MY130727A (en) 2007-07-31
IL141764A (en) 2008-06-05
ES2272082T3 (es) 2007-04-16
ID28232A (id) 2001-05-10
IL141764A0 (en) 2002-03-10
MXPA01004011A (es) 2003-03-10
NO20011933L (no) 2001-06-25
PL347476A1 (en) 2002-04-08
TW577756B (en) 2004-03-01
GT199900184A (es) 2001-04-14

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