EE200100235A - cGMP PDE-5 inhibiitorit sisaldavad kontrollitud vabanemisega farmatseutilised formulatsioonid - Google Patents

cGMP PDE-5 inhibiitorit sisaldavad kontrollitud vabanemisega farmatseutilised formulatsioonid

Info

Publication number
EE200100235A
EE200100235A EEP200100235A EEP200100235A EE200100235A EE 200100235 A EE200100235 A EE 200100235A EE P200100235 A EEP200100235 A EE P200100235A EE P200100235 A EEP200100235 A EE P200100235A EE 200100235 A EE200100235 A EE 200100235A
Authority
EE
Estonia
Prior art keywords
inhibitor
controlled release
pharmaceutical formulations
formulations containing
release pharmaceutical
Prior art date
Application number
EEP200100235A
Other languages
English (en)
Inventor
King Elizabeth
James Macrae Ross
Original Assignee
Pfizer Research And Development Company, N.V./S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27269526&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EE200100235(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GBGB9823192.1A external-priority patent/GB9823192D0/en
Priority claimed from GBGB9825117.6A external-priority patent/GB9825117D0/en
Priority claimed from GBGB9826392.4A external-priority patent/GB9826392D0/en
Application filed by Pfizer Research And Development Company, N.V./S.A. filed Critical Pfizer Research And Development Company, N.V./S.A.
Publication of EE200100235A publication Critical patent/EE200100235A/et

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846—Poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Gynecology & Obstetrics (AREA)
  • Neurology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
EEP200100235A 1998-10-23 1999-10-04 cGMP PDE-5 inhibiitorit sisaldavad kontrollitud vabanemisega farmatseutilised formulatsioonid EE200100235A (et)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GBGB9823192.1A GB9823192D0 (en) 1998-10-23 1998-10-23 Pharmaceutical formulations
GBGB9825117.6A GB9825117D0 (en) 1998-11-16 1998-11-16 Pharmaceutical formulations
GBGB9826392.4A GB9826392D0 (en) 1998-11-27 1998-11-27 Pharmaceutical formulations
PCT/IB1999/001619 WO2000024383A1 (en) 1998-10-23 1999-10-04 Controlled-release pharmaceutical formulations containing a cgmp pde-5 inhibitor

Publications (1)

Publication Number Publication Date
EE200100235A true EE200100235A (et) 2002-08-15

Family

ID=27269526

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200100235A EE200100235A (et) 1998-10-23 1999-10-04 cGMP PDE-5 inhibiitorit sisaldavad kontrollitud vabanemisega farmatseutilised formulatsioonid

Country Status (44)

Country Link
US (1) US6964780B1 (et)
EP (1) EP1123088B1 (et)
JP (1) JP2002528408A (et)
KR (1) KR20010075659A (et)
CN (1) CN1324233A (et)
AP (1) AP2001002125A0 (et)
AT (1) ATE340562T1 (et)
AU (1) AU756509B2 (et)
BG (1) BG65323B1 (et)
BR (1) BR9914718A (et)
CA (1) CA2348086C (et)
CO (1) CO5160262A1 (et)
CR (1) CR6326A (et)
CY (1) CY1106239T1 (et)
CZ (1) CZ20011427A3 (et)
DE (1) DE69933383T2 (et)
DK (1) DK1123088T3 (et)
DZ (1) DZ2923A1 (et)
EA (1) EA004068B1 (et)
EE (1) EE200100235A (et)
ES (1) ES2272082T3 (et)
GT (1) GT199900184A (et)
HK (1) HK1041818A1 (et)
HR (1) HRP20010285A2 (et)
HU (1) HUP0104318A3 (et)
ID (1) ID28232A (et)
IL (1) IL141764A (et)
IS (1) IS5865A (et)
MA (1) MA26700A1 (et)
MX (1) MXPA01004011A (et)
MY (1) MY130727A (et)
NO (1) NO20011933L (et)
NZ (1) NZ510275A (et)
OA (1) OA11664A (et)
PA (1) PA8484301A1 (et)
PE (1) PE20001286A1 (et)
PL (1) PL195789B1 (et)
PT (1) PT1123088E (et)
SK (1) SK286473B6 (et)
TR (1) TR200101103T2 (et)
TW (1) TW577756B (et)
UA (1) UA67802C2 (et)
UY (1) UY25765A1 (et)
WO (1) WO2000024383A1 (et)

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DE60236850D1 (de) * 2001-02-15 2010-08-12 Mitsubishi Tanabe Pharma Corp Tabletten, die in der mundhöhle schnell zerfallen
US10675280B2 (en) 2001-10-20 2020-06-09 Sprout Pharmaceuticals, Inc. Treating sexual desire disorders with flibanserin
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JP5793828B2 (ja) 2006-08-14 2015-10-14 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング フリバンセリンの製剤及びその製造方法
EP2056797A2 (en) 2006-08-25 2009-05-13 Boehringer Ingelheim International GmbH Controlled release system and method for manufacturing the same
EP1925307A1 (en) * 2006-11-03 2008-05-28 Emotional Brain B.V. Use of 3-alpha-androstanediol in the treatment of sexual dysfunction
US20080226715A1 (en) * 2007-03-16 2008-09-18 Albert Cha Therapeutic compositions and methods
CN101711153A (zh) * 2007-06-13 2010-05-19 拜耳先灵制药股份公司 用于治疗听觉损伤的pde抑制剂
CL2008002693A1 (es) 2007-09-12 2009-10-16 Boehringer Ingelheim Int Uso de flibanserina para el tratamiento de sintomas vasomotores seleccionados de sofocos, sudores nocturnos, cambios de estado de animo e irritabilidad
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EP2374460A4 (en) * 2008-12-12 2013-08-21 Rhein Siegfried Sa De Cv SILDENAFIL COMPOSITION WITH PULSED RELEASE AND METHOD FOR PRODUCING THIS COMPOSITION
KR101004205B1 (ko) * 2008-12-17 2010-12-24 동아제약주식회사 유데나필 함유 서방성 제제를 제조하기 위한 제어방출 조성물
EA015250B9 (ru) * 2010-11-19 2013-10-30 Тева Фармасьютикал Индастриз, Лтд. Таблетка силденафила, обеспечивающая модифицированную фармакокинетику, и способ ее изготовления
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WO2017168174A1 (en) * 2016-04-02 2017-10-05 N4 Pharma Uk Limited New pharmaceutical forms of sildenafil
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Also Published As

Publication number Publication date
HUP0104318A3 (en) 2003-12-29
AP2001002125A0 (en) 2001-04-04
EA004068B1 (ru) 2003-12-25
AU756509B2 (en) 2003-01-16
JP2002528408A (ja) 2002-09-03
CR6326A (es) 2004-02-23
CO5160262A1 (es) 2002-05-30
CA2348086A1 (en) 2000-05-04
MY130727A (en) 2007-07-31
BG105465A (bg) 2001-12-29
IS5865A (is) 2001-02-27
NO20011933D0 (no) 2001-04-19
AU5878799A (en) 2000-05-15
UY25765A1 (es) 2001-08-27
HUP0104318A2 (hu) 2002-03-28
DE69933383D1 (de) 2006-11-09
DK1123088T3 (da) 2007-01-02
PL195789B1 (pl) 2007-10-31
GT199900184A (es) 2001-04-14
NZ510275A (en) 2003-07-25
HK1041818A1 (zh) 2002-07-26
EP1123088B1 (en) 2006-09-27
IL141764A (en) 2008-06-05
BG65323B1 (bg) 2008-02-29
CZ20011427A3 (cs) 2001-10-17
DE69933383T2 (de) 2007-02-01
ATE340562T1 (de) 2006-10-15
EA200100298A1 (ru) 2001-08-27
BR9914718A (pt) 2001-07-10
NO20011933L (no) 2001-06-25
IL141764A0 (en) 2002-03-10
CY1106239T1 (el) 2011-06-08
TR200101103T2 (tr) 2001-09-21
PT1123088E (pt) 2007-01-31
PA8484301A1 (es) 2000-09-29
WO2000024383A1 (en) 2000-05-04
PE20001286A1 (es) 2000-11-22
UA67802C2 (uk) 2004-07-15
EP1123088A1 (en) 2001-08-16
MA26700A1 (fr) 2004-12-20
MXPA01004011A (es) 2003-03-10
ID28232A (id) 2001-05-10
CA2348086C (en) 2007-01-23
ES2272082T3 (es) 2007-04-16
US6964780B1 (en) 2005-11-15
TW577756B (en) 2004-03-01
OA11664A (en) 2005-01-07
SK286473B6 (sk) 2008-11-06
SK5192001A3 (en) 2002-09-10
CN1324233A (zh) 2001-11-28
PL347476A1 (en) 2002-04-08
DZ2923A1 (fr) 2004-03-01
HRP20010285A2 (en) 2002-06-30
KR20010075659A (ko) 2001-08-09

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