PA8484301A1 - Formulaciones farmaceuticas de liberacion controlada - Google Patents

Formulaciones farmaceuticas de liberacion controlada

Info

Publication number
PA8484301A1
PA8484301A1 PA19998484301A PA8484301A PA8484301A1 PA 8484301 A1 PA8484301 A1 PA 8484301A1 PA 19998484301 A PA19998484301 A PA 19998484301A PA 8484301 A PA8484301 A PA 8484301A PA 8484301 A1 PA8484301 A1 PA 8484301A1
Authority
PA
Panama
Prior art keywords
pharmaceutical formulations
controlled liberation
liberation
controlled
formulations
Prior art date
Application number
PA19998484301A
Other languages
English (en)
Inventor
Elizabeth King
Ross James Macrae
Original Assignee
Warner Lambert Exp Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27269526&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PA8484301(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GBGB9823192.1A external-priority patent/GB9823192D0/en
Priority claimed from GBGB9825117.6A external-priority patent/GB9825117D0/en
Priority claimed from GBGB9826392.4A external-priority patent/GB9826392D0/en
Application filed by Warner Lambert Exp Ltd filed Critical Warner Lambert Exp Ltd
Publication of PA8484301A1 publication Critical patent/PA8484301A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846Poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Abstract

LA INVENCION PROPORCIONA FORMULACIONES FARMACEUTICAS DE LIBERACION CONTROLADA PARA ADMINISTRACION ORAL QUE CONTIENEN UN INHIBIDOR GMPC PDE-5. LAS FORMULACIONES SON UTILES, ENTRE OTROS, EN EL TRATAMIENTO O PREVENCION DE LA DISFUNCION SEXUAL.
PA19998484301A 1998-10-23 1999-10-18 Formulaciones farmaceuticas de liberacion controlada PA8484301A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB9823192.1A GB9823192D0 (en) 1998-10-23 1998-10-23 Pharmaceutical formulations
GBGB9825117.6A GB9825117D0 (en) 1998-11-16 1998-11-16 Pharmaceutical formulations
GBGB9826392.4A GB9826392D0 (en) 1998-11-27 1998-11-27 Pharmaceutical formulations

Publications (1)

Publication Number Publication Date
PA8484301A1 true PA8484301A1 (es) 2000-09-29

Family

ID=27269526

Family Applications (1)

Application Number Title Priority Date Filing Date
PA19998484301A PA8484301A1 (es) 1998-10-23 1999-10-18 Formulaciones farmaceuticas de liberacion controlada

Country Status (44)

Country Link
US (1) US6964780B1 (es)
EP (1) EP1123088B1 (es)
JP (1) JP2002528408A (es)
KR (1) KR20010075659A (es)
CN (1) CN1324233A (es)
AP (1) AP2001002125A0 (es)
AT (1) ATE340562T1 (es)
AU (1) AU756509B2 (es)
BG (1) BG65323B1 (es)
BR (1) BR9914718A (es)
CA (1) CA2348086C (es)
CO (1) CO5160262A1 (es)
CR (1) CR6326A (es)
CY (1) CY1106239T1 (es)
CZ (1) CZ20011427A3 (es)
DE (1) DE69933383T2 (es)
DK (1) DK1123088T3 (es)
DZ (1) DZ2923A1 (es)
EA (1) EA004068B1 (es)
EE (1) EE200100235A (es)
ES (1) ES2272082T3 (es)
GT (1) GT199900184A (es)
HK (1) HK1041818A1 (es)
HR (1) HRP20010285A2 (es)
HU (1) HUP0104318A3 (es)
ID (1) ID28232A (es)
IL (1) IL141764A (es)
IS (1) IS5865A (es)
MA (1) MA26700A1 (es)
MX (1) MXPA01004011A (es)
MY (1) MY130727A (es)
NO (1) NO20011933L (es)
NZ (1) NZ510275A (es)
OA (1) OA11664A (es)
PA (1) PA8484301A1 (es)
PE (1) PE20001286A1 (es)
PL (1) PL195789B1 (es)
PT (1) PT1123088E (es)
SK (1) SK286473B6 (es)
TR (1) TR200101103T2 (es)
TW (1) TW577756B (es)
UA (1) UA67802C2 (es)
UY (1) UY25765A1 (es)
WO (1) WO2000024383A1 (es)

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AU2002230217B2 (en) 2001-02-15 2005-02-17 Tanabe Seiyaku Co., Ltd. Tablets quickly disintegrated in oral cavity
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EP1896076A2 (en) * 2005-06-27 2008-03-12 Daniel Drai Compositions and methods for enhancement of sexual function
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KR20080056250A (ko) * 2005-09-29 2008-06-20 바이엘 헬스케어 아게 비뇨기 장애의 치료를 위한 pde 억제제 및 이들의 조합
EP1945214A1 (en) 2005-10-29 2008-07-23 Boehringer Ingelheim International GmbH Benzimidazolone derivatives for the treatment of premenstrual and other female sexual disorders
EP1790343A1 (en) * 2005-11-11 2007-05-30 Emotional Brain B.V. Pharmaceuticals formulations and uses thereof in the treatment of female sexual dysfunction
DE602007004615D1 (de) 2006-06-30 2010-03-18 Boehringer Ingelheim Pharma Flibanserin zur behandlung von harninkontinenz und assoziierten erkrankungen
CA2660476C (en) 2006-08-14 2015-11-17 Boehringer Ingelheim International Gmbh Formulations of flibanserin and method for manufacturing the same
CA2661613C (en) 2006-08-25 2016-01-26 Boehringer Ingelheim International Gmbh Controlled release system and method for manufacturing the same
EP1925307A1 (en) * 2006-11-03 2008-05-28 Emotional Brain B.V. Use of 3-alpha-androstanediol in the treatment of sexual dysfunction
WO2008115797A1 (en) * 2007-03-16 2008-09-25 Pavo, Inc. Therapeutic compositions and methods
JP2010532319A (ja) * 2007-06-13 2010-10-07 バイエル・シェーリング・ファルマ・アクチェンゲゼルシャフト 聴覚障害の処置用のpde阻害剤
PE20091188A1 (es) 2007-09-12 2009-08-31 Boehringer Ingelheim Int Compuesto 1-[2-(4-(3-trifluorometil-fenil)piperazin-1-il)etil]-2,3-dihidro-1h-benzimidazol-2-ona (flibanserina), sus sales de adicion y composiciones farmaceuticas que los contienen
US20110033506A1 (en) * 2008-02-08 2011-02-10 Adel Penhasi Combination dosage form of low-dose modafinil and low-dose sildenafil
EP2374460A4 (en) * 2008-12-12 2013-08-21 Rhein Siegfried Sa De Cv SILDENAFIL COMPOSITION WITH PULSED RELEASE AND METHOD FOR PRODUCING THIS COMPOSITION
KR101004205B1 (ko) * 2008-12-17 2010-12-24 동아제약주식회사 유데나필 함유 서방성 제제를 제조하기 위한 제어방출 조성물
EA015250B9 (ru) * 2010-11-19 2013-10-30 Тева Фармасьютикал Индастриз, Лтд. Таблетка силденафила, обеспечивающая модифицированную фармакокинетику, и способ ее изготовления
BR112013029199B1 (pt) 2011-05-13 2022-02-08 Eb Ip Hybritabs B.V. Dispositivo de distribuição de dois fármacos
WO2013016144A1 (en) * 2011-07-22 2013-01-31 Pom Wonderful, Llc Compositions comprising pomegranate polyphenols in combination with erectile dysfunction-treating compounds, and methods of treating erectile dysfunction therewith
WO2017168174A1 (en) * 2016-04-02 2017-10-05 N4 Pharma Uk Limited New pharmaceutical forms of sildenafil
CN113995727B (zh) * 2021-11-08 2023-04-07 山东鲁抗医药股份有限公司 一种5型磷酸二酯酶抑制剂片剂及其制备方法

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Also Published As

Publication number Publication date
BG105465A (bg) 2001-12-29
CR6326A (es) 2004-02-23
CN1324233A (zh) 2001-11-28
EA200100298A1 (ru) 2001-08-27
WO2000024383A1 (en) 2000-05-04
PE20001286A1 (es) 2000-11-22
EP1123088A1 (en) 2001-08-16
NO20011933L (no) 2001-06-25
AU5878799A (en) 2000-05-15
EE200100235A (et) 2002-08-15
MXPA01004011A (es) 2003-03-10
UY25765A1 (es) 2001-08-27
EA004068B1 (ru) 2003-12-25
CZ20011427A3 (cs) 2001-10-17
NZ510275A (en) 2003-07-25
PL195789B1 (pl) 2007-10-31
AU756509B2 (en) 2003-01-16
DE69933383D1 (de) 2006-11-09
KR20010075659A (ko) 2001-08-09
BR9914718A (pt) 2001-07-10
US6964780B1 (en) 2005-11-15
HUP0104318A3 (en) 2003-12-29
DE69933383T2 (de) 2007-02-01
MY130727A (en) 2007-07-31
CA2348086A1 (en) 2000-05-04
PL347476A1 (en) 2002-04-08
CY1106239T1 (el) 2011-06-08
IS5865A (is) 2001-02-27
CO5160262A1 (es) 2002-05-30
AP2001002125A0 (en) 2001-04-04
HUP0104318A2 (hu) 2002-03-28
PT1123088E (pt) 2007-01-31
HK1041818A1 (zh) 2002-07-26
NO20011933D0 (no) 2001-04-19
DK1123088T3 (da) 2007-01-02
TR200101103T2 (tr) 2001-09-21
GT199900184A (es) 2001-04-14
OA11664A (en) 2005-01-07
MA26700A1 (fr) 2004-12-20
ATE340562T1 (de) 2006-10-15
EP1123088B1 (en) 2006-09-27
SK286473B6 (sk) 2008-11-06
DZ2923A1 (fr) 2004-03-01
TW577756B (en) 2004-03-01
CA2348086C (en) 2007-01-23
JP2002528408A (ja) 2002-09-03
ES2272082T3 (es) 2007-04-16
IL141764A (en) 2008-06-05
UA67802C2 (uk) 2004-07-15
HRP20010285A2 (en) 2002-06-30
BG65323B1 (bg) 2008-02-29
SK5192001A3 (en) 2002-09-10
IL141764A0 (en) 2002-03-10
ID28232A (id) 2001-05-10

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