SK165795A3 - 3-phenylizoquinoline-1(2h)-one derivatives, preparation method and pharmaceutical compounds containing these derivatives - Google Patents

3-phenylizoquinoline-1(2h)-one derivatives, preparation method and pharmaceutical compounds containing these derivatives Download PDF

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Publication number
SK165795A3
SK165795A3 SK1657-95A SK165795A SK165795A3 SK 165795 A3 SK165795 A3 SK 165795A3 SK 165795 A SK165795 A SK 165795A SK 165795 A3 SK165795 A3 SK 165795A3
Authority
SK
Slovakia
Prior art keywords
formula
methyl
compound
compounds
carbon atoms
Prior art date
Application number
SK1657-95A
Other languages
English (en)
Slovak (sk)
Inventor
Mireille Sevrin
Benoit Marabout
Jacques Froissant
Catherine Guinot
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of SK165795A3 publication Critical patent/SK165795A3/sk

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D217/00Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/22Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D217/00Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/22Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
    • C07D217/24Oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/16Otologicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
SK1657-95A 1994-12-29 1995-12-28 3-phenylizoquinoline-1(2h)-one derivatives, preparation method and pharmaceutical compounds containing these derivatives SK165795A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9415837A FR2728900B1 (fr) 1994-12-29 1994-12-29 Derives de 3-phenylisoquinolein-1(2h)-one, leur preparation et leur application en therapeutique

Publications (1)

Publication Number Publication Date
SK165795A3 true SK165795A3 (en) 1996-07-03

Family

ID=9470390

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1657-95A SK165795A3 (en) 1994-12-29 1995-12-28 3-phenylizoquinoline-1(2h)-one derivatives, preparation method and pharmaceutical compounds containing these derivatives

Country Status (22)

Country Link
US (1) US5665733A (de)
EP (1) EP0719764B1 (de)
JP (1) JPH08239365A (de)
KR (1) KR960022472A (de)
CN (1) CN1131150A (de)
AR (1) AR002016A1 (de)
AT (1) ATE172966T1 (de)
AU (1) AU698595B2 (de)
BR (1) BR9506106A (de)
CA (1) CA2166234A1 (de)
CO (1) CO4700298A1 (de)
CZ (1) CZ348995A3 (de)
DE (1) DE69505780D1 (de)
FI (1) FI956298A (de)
FR (1) FR2728900B1 (de)
HU (1) HU215394B (de)
IL (1) IL116590A0 (de)
NO (1) NO955326L (de)
NZ (1) NZ280765A (de)
PL (1) PL312079A1 (de)
SK (1) SK165795A3 (de)
ZA (1) ZA9511046B (de)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2750427B1 (fr) * 1996-06-28 1998-08-07 Synthelabo Derives de 1-oxo-1, 2-dihydroisoquinoleine-4-propanamide, leur preparation et leur application en therapeutique
FR2772758B1 (fr) * 1997-12-22 2000-02-04 Synthelabo Derives de 1-oxo-1,2-dihydroisoquinoleine-4-propanamide, leur preparation et leur application en therapeutique
ATE496893T1 (de) * 2002-12-20 2011-02-15 X Ceptor Therapeutics Inc Isochinolinonderivate und deren verwendung als medikamente
GB0420722D0 (en) * 2004-09-17 2004-10-20 Addex Pharmaceuticals Sa Novel allosteric modulators
EP2064185B1 (de) * 2006-08-10 2011-06-08 Ferrer Internacional, S.A. 1h-chinolin-4-on-verbindungen mit affinität zum gaba-rezeptor, verfahren, anwendungen und zusammensetzungen
EP1886996A1 (de) * 2006-08-10 2008-02-13 Ferrer Internacional, S.A. 1H-Chinolin-4-on Verbindungen mit Affinität für den GABA Rezeptor, Prozesse, Verwendungen und Zusammensetzungen
EP2387564A1 (de) 2009-01-15 2011-11-23 Rutgers, The State University of New Jersey Benzo[c]phenanthridine als antimikrobielle mittel
WO2010127307A1 (en) 2009-04-30 2010-11-04 Rutgers, The State University Of New Jersey Antimicrobial agents
FR2956816B1 (fr) * 2010-03-01 2012-05-18 Univ Joseph Fourier Utilisation de quinolones pour la preparation de medicaments, nouvelles quinolones et leur procede de synthese
WO2011156626A1 (en) 2010-06-09 2011-12-15 Rutgers, The State University Of New Jersey Antimicrobial agents
CA2803890A1 (en) 2010-06-25 2011-12-29 Rutgers, The State University Of New Jersey Antimicrobial agents
US9822108B2 (en) 2012-01-13 2017-11-21 Rutgers, The State University Of New Jersey Antimicrobial agents
EP2828245A1 (de) 2012-03-21 2015-01-28 Rutgers, The State University of New Jersey Antimikrobiotika
US9458150B2 (en) 2013-11-08 2016-10-04 Rutgers, The State University Of New Jersey Antimicrobial agents
US10513528B2 (en) 2016-02-25 2019-12-24 Taxis Pharmaceuticals, Inc. Synthetic processes and intermediates
US10774093B2 (en) 2017-03-30 2020-09-15 Taxis Pharmaceuticals, Inc. Synthetic processes and synthetic intermediates
EP4126858A1 (de) * 2020-03-26 2023-02-08 Richter Gedeon Nyrt. Dihydro-2-pyrrolo[3,4-c pyridin-derivate als gabaa a5 rezeptormodulatoren
TW202202495A (zh) * 2020-03-26 2022-01-16 匈牙利商羅特格登公司 作為gamma-胺基丁酸A受體次單元alpha 5受體調節劑之㖠啶及吡啶并〔3,4-c〕嗒𠯤衍生物

Also Published As

Publication number Publication date
HUT74187A (en) 1996-11-28
FI956298A0 (fi) 1995-12-28
CN1131150A (zh) 1996-09-18
KR960022472A (ko) 1996-07-18
CZ348995A3 (en) 1996-07-17
AR002016A1 (es) 1998-01-07
DE69505780D1 (de) 1998-12-10
CA2166234A1 (en) 1996-06-30
HU215394B (hu) 1998-12-28
HU9503848D0 (en) 1996-02-28
EP0719764A1 (de) 1996-07-03
NO955326D0 (no) 1995-12-28
PL312079A1 (en) 1996-07-08
ZA9511046B (en) 1996-07-11
FR2728900B1 (fr) 1997-01-31
FI956298A (fi) 1996-06-30
FR2728900A1 (fr) 1996-07-05
JPH08239365A (ja) 1996-09-17
BR9506106A (pt) 1997-12-23
AU698595B2 (en) 1998-11-05
CO4700298A1 (es) 1998-12-29
US5665733A (en) 1997-09-09
AU4071295A (en) 1996-07-04
NZ280765A (en) 1996-08-27
ATE172966T1 (de) 1998-11-15
IL116590A0 (en) 1996-03-31
EP0719764B1 (de) 1998-11-04
NO955326L (no) 1996-07-01

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