SK120895A3 - Pyridine derivatives, process for preparing the same and intermediate products in this process and pharmaceutical compositions containing them - Google Patents

Pyridine derivatives, process for preparing the same and intermediate products in this process and pharmaceutical compositions containing them Download PDF

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Publication number
SK120895A3
SK120895A3 SK1208-95A SK120895A SK120895A3 SK 120895 A3 SK120895 A3 SK 120895A3 SK 120895 A SK120895 A SK 120895A SK 120895 A3 SK120895 A3 SK 120895A3
Authority
SK
Slovakia
Prior art keywords
group
carbon atoms
formula
alkylene
pyridyl
Prior art date
Application number
SK1208-95A
Other languages
English (en)
Slovak (sk)
Inventor
Michael G Wayne
Michael J Smithers
John W Rayner
Alan W Faull
Robert J Pearce
Andrew G Brewster
Richard E Shute
Stuart D Mills
Peter W R Caulkett
Original Assignee
Zeneca Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB939306453A external-priority patent/GB9306453D0/en
Priority claimed from GB939325605A external-priority patent/GB9325605D0/en
Application filed by Zeneca Ltd filed Critical Zeneca Ltd
Publication of SK120895A3 publication Critical patent/SK120895A3/sk

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Electrochromic Elements, Electrophoresis, Or Variable Reflection Or Absorption Elements (AREA)
  • Electroluminescent Light Sources (AREA)
  • Emulsifying, Dispersing, Foam-Producing Or Wetting Agents (AREA)
  • Pyrrole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
SK1208-95A 1993-03-29 1994-03-28 Pyridine derivatives, process for preparing the same and intermediate products in this process and pharmaceutical compositions containing them SK120895A3 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB939306453A GB9306453D0 (en) 1993-03-29 1993-03-29 Heterocyclic derivatives
GB939325605A GB9325605D0 (en) 1993-12-15 1993-12-15 Heterocyclic derivatives
PCT/GB1994/000647 WO1994022834A1 (en) 1993-03-29 1994-03-28 Heterocyclic derivatives as platelet aggregation inhibitors

Publications (1)

Publication Number Publication Date
SK120895A3 true SK120895A3 (en) 1996-06-05

Family

ID=26302668

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1208-95A SK120895A3 (en) 1993-03-29 1994-03-28 Pyridine derivatives, process for preparing the same and intermediate products in this process and pharmaceutical compositions containing them

Country Status (26)

Country Link
US (1) US5556977A (https=)
EP (2) EP0691959B1 (https=)
JP (1) JPH08508291A (https=)
KR (1) KR100231089B1 (https=)
CN (1) CN1120334A (https=)
AT (2) ATE202345T1 (https=)
AU (1) AU692438B2 (https=)
BR (1) BR9406613A (https=)
CA (1) CA2156070A1 (https=)
CZ (1) CZ250995A3 (https=)
DE (2) DE69427548T2 (https=)
DK (2) DK0691959T3 (https=)
ES (2) ES2119184T3 (https=)
FI (1) FI954616L (https=)
GB (1) GB9406143D0 (https=)
GR (2) GR3027751T3 (https=)
HU (2) HUT72088A (https=)
IL (1) IL109144A (https=)
NO (1) NO305244B1 (https=)
NZ (1) NZ262941A (https=)
PL (1) PL310889A1 (https=)
PT (1) PT825184E (https=)
SK (1) SK120895A3 (https=)
TW (1) TW276254B (https=)
WO (1) WO1994022834A1 (https=)
ZW (1) ZW4294A1 (https=)

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GB9902989D0 (en) 1999-02-11 1999-03-31 Zeneca Ltd Heterocyclic derivatives
CA2370742A1 (en) * 1999-04-19 2000-10-26 Coelacanth Corporation Ppar-(gamma) agonists as agents for the treatment of type ii diabetes
US6310081B1 (en) 1999-05-10 2001-10-30 American Home Products Corporation Biphenyl sulfonyl aryl carboxylic acids useful in the treatment of insulin resistance and hyperglycemia
DE60144284D1 (de) 2000-11-01 2011-05-05 Millennium Pharm Inc Stickstoffhaltige heterozyklische verbindungen und verfahren zu deren herstellung
DE202011000090U1 (de) 2011-01-14 2011-04-21 E-LEAD ELECTRONIC CO., LTD., Shengang Shiang Fahrzeug-Audiosystem mit auswechselbarem Plug-In-Computer
MX2020003242A (es) 2017-09-22 2020-09-18 Jubilant Epipad LLC Compuestos heterociclicos como inhibidores de pad.
AU2018352142B2 (en) 2017-10-18 2022-08-25 Jubilant Epipad LLC Imidazo-pyridine compounds as PAD inhibitors
KR20200085836A (ko) 2017-11-06 2020-07-15 주빌런트 프로델 엘엘씨 Pd1/pd-l1 활성화 억제제로서의 피리미딘 유도체
BR112020010322A2 (pt) 2017-11-24 2020-11-17 Jubilant Episcribe Llc composto da fórmula i; composto da fórmula ia; composto da fórmula ib; processo de preparação de compostos da fórmula i; composição farmacêutica; método para o tratamento e/ou prevenção de várias doenças; uso dos compostos; método para o tratamento de câncer; e método para o tratamento e/ou prevenção de uma afecção mediada por prmt5 ou um distúrbio proliferativo ou câncer
SG11202008950PA (en) 2018-03-13 2020-10-29 Jubilant Prodel LLC Bicyclic compounds as inhibitors of pd1/pd-l1 interaction/activation

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Also Published As

Publication number Publication date
IL109144A0 (en) 1994-06-24
EP0691959B1 (en) 1998-07-22
GR3036640T3 (en) 2001-12-31
HU211336A9 (en) 1995-11-28
FI954616A7 (fi) 1995-09-28
WO1994022834A1 (en) 1994-10-13
KR100231089B1 (ko) 1999-11-15
DK0691959T3 (da) 1999-04-26
CN1120334A (zh) 1996-04-10
PL310889A1 (en) 1996-01-08
CA2156070A1 (en) 1994-10-13
FI954616A0 (fi) 1995-09-28
ATE202345T1 (de) 2001-07-15
HUT72088A (en) 1996-03-28
IL109144A (en) 2000-02-29
AU6288994A (en) 1994-10-24
DE69427548T2 (de) 2002-04-18
JPH08508291A (ja) 1996-09-03
HU9502290D0 (en) 1995-10-30
ZW4294A1 (en) 1994-12-21
DE69411900T2 (de) 1998-12-10
NO305244B1 (no) 1999-04-26
DK0825184T3 (da) 2001-09-10
GB9406143D0 (en) 1994-05-18
FI954616L (fi) 1995-09-28
NZ262941A (en) 1997-07-27
PT825184E (pt) 2001-11-30
CZ250995A3 (en) 1996-01-17
US5556977A (en) 1996-09-17
NO953837L (no) 1995-09-28
TW276254B (https=) 1996-05-21
DE69411900D1 (de) 1998-08-27
EP0691959A1 (en) 1996-01-17
BR9406613A (pt) 1996-02-06
DE69427548D1 (de) 2001-07-26
ES2159798T3 (es) 2001-10-16
EP0825184B1 (en) 2001-06-20
ES2119184T3 (es) 1998-10-01
ATE168678T1 (de) 1998-08-15
EP0825184A1 (en) 1998-02-25
NO953837D0 (no) 1995-09-28
GR3027751T3 (en) 1998-11-30
AU692438B2 (en) 1998-06-11

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